Zobrazeno 1 - 10
of 106
pro vyhledávání: '"Milan Potáček"'
Publikováno v:
ARKIVOC, Vol 2001, Iss 2, Pp 146-162 (2002)
Externí odkaz:
https://doaj.org/article/86b258717e414677b9b535c13dbd1071
Publikováno v:
Molecules, Vol 21, Iss 2, p 187 (2016)
This paper describes the synthesis of precursors with a benzo[b]furan skeleton for the intramolecular 1,3-dipolar cycloaddition of azomethine ylides prepared from N-substituted 3-allyl-aminobenzo[b]furan-2-aldehydes and secondary amines derived from
Externí odkaz:
https://doaj.org/article/4aefb824f77c43b88a5c39df09c60c0f
Publikováno v:
Acta Crystallographica Section E, Vol 65, Iss 6, Pp o1307-o1307 (2009)
In the title salt, C12H20NO+·CH3SO3−, the [1-(1-adamantylamino)ethylidene]oxonium cations and methanesulfonate anions are linked into chains along the a axis via O—H...O and N—H...O hydrogen bonds. All non-H atoms of the acetamido group are es
Externí odkaz:
https://doaj.org/article/a74bb21d67ef4b1a8ae4b128fb4c1e0a
Autor:
Jiří Brynda, Ullrich Jahn, Milan Potáček, Anna Hlavačková, Vlastimil Král, M. Kugler, Pavlína Řezáčová, Jiří Schimer, Milan Dejmek, Pavel Šácha, Jan Tykvart, Jan Konvalinka, Lukáš Tenora, Václav Navrátil, Jitka Zemanova, Pavel Majer
Publikováno v:
SLAS Discovery. 25:1026-1037
The DNA-linked inhibitor antibody assay (DIANA) has been recently validated for ultrasensitive enzyme detection and for quantitative evaluation of enzyme inhibitor potency. Here we present its adaptation for high-throughput screening of human carboni
Publikováno v:
The Journal of Organic Chemistry. 81:11841-11856
C-H activation of position 3 of a substituted pyrazole ring catalyzed by palladium(II) was straightforward and convenient for arylated or heteroarylated 5,5-dimethyl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazoles. Moreover, we introduced simple protection of
Publikováno v:
Synthesis. 48:2429-2437
The paper describes synthesis of two regioisomeric 2-amino-3-formyl and 3-amino-2-formyl substituted derivatives of tetrahydrobenzo[b] thiophene and their preparation for subsequent thermally-initiated reactions with secondary amines for generation o
Autor:
Milan Potáček, Juraj Galeta
Publikováno v:
Journal of Molecular Catalysis A: Chemical. 395:87-92
Superbasic properties of caged proton sponges (PSs) – substituted diazatetracyclo[4.4.0.13,10.15,8]dodecanes (DTDs) – were utilized in Knoevenagel and Claisen–Schmidt condensations, the Pudovik reaction, and Michael addition. This investigation
Autor:
Dominique Harakat, Milan Potáček, Juraj Galeta, Jean-Philippe Bouillon, Francois‐Xavier Harnisch
Publikováno v:
Journal of Fluorine Chemistry. 158:38-43
Blocked hydrazines were prepared by the reaction of diethyl hydrazinophosphate with fluorinated aldehydes applying Zwierzak’s method and then introduced into the reaction with 3-substituted homoallenyl aldehydes. The resulting non-symmetrical fluor
Autor:
Pavlína Pospíšilová, Pavel Majer, Vladimír Kryštof, Eva Řezníčková, Radek Jorda, Milan Potáček, Juraj Galeta, Karel Berka, Lukáš Tenora
Publikováno v:
European journal of medicinal chemistry. 127
A series of 2,3,4-substituted 5,5-dimethyl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazoles (DPPs) was synthesized and evaluated for their ALK5 inhibition activity. The most potent compounds displayed submicromolar IC50 values for ALK5. Preliminary profiling o
Publikováno v:
ChemInform. 47