Zobrazeno 1 - 10
of 50
pro vyhledávání: '"Michelyne, Haroun"'
Autor:
Michelyne Haroun, Maria Fesatidou, Anthi Petrou, Christophe Tratrat, Panagiotis Zagaliotis, Antonis Gavalas, Katharigatta N. Venugopala, Hafedh Kochkar, Promise M. Emeka, Nancy S. Younis, Dalia Ahmed Elmaghraby, Mervt M. Almostafa, Muhammad Shahzad Chohan, Ioannis S. Vizirianakis, Aliki Papadimitriou-Tsantarliotou, Athina Geronikaki
Publikováno v:
Molecules, Vol 28, Iss 8, p 3416 (2023)
Major obstacles faced by the use of nonsteroidal anti-inflammatory drugs (NSAID) are their gastrointestinal toxicity induced by non-selective inhibition of both cyclooxygenases (COX) 1 and 2 and their cardiotoxicity associated with a certain class of
Externí odkaz:
https://doaj.org/article/18a59193f9924d31ac5c5a1b48fac4bf
Autor:
Katharigatta N. Venugopala, Sandeep Chandrashekharappa, Pran Kishore Deb, Christophe Tratrat, Melendhran Pillay, Deepak Chopra, Nizar A. Al-Shar’i, Wafa Hourani, Lina A. Dahabiyeh, Pobitra Borah, Rahul D. Nagdeve, Susanta K. Nayak, Basavaraj Padmashali, Mohamed A. Morsy, Bandar E. Aldhubiab, Mahesh Attimarad, Anroop B. Nair, Nagaraja Sreeharsha, Michelyne Haroun, Sheena Shashikanth, Viresh Mohanlall, Raghuprasad Mailavaram
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 1471-1486 (2021)
A series of 1,2,3-trisubstituted indolizines (2a–2f, 3a–3d, and 4a–4c) were screened for in vitro whole-cell anti-tubercular activity against the susceptible H37Rv and multidrug-resistant (MDR) Mycobacterium tuberculosis (MTB) strains. Compound
Externí odkaz:
https://doaj.org/article/317149f295104f1dbe7c0e6553495828
Autor:
Michelyne Haroun, Anthi Petrou, Christophe Tratrat, Aggeliki Kolokotroni, Maria Fesatidou, Panagiotis Zagaliotis, Antonis Gavalas, Katharigatta N. Venugopala, Nagaraja Sreeharsha, Anroop B. Nair, Heba Sadek Elsewedy, Athina Geronikaki
Publikováno v:
Molecules, Vol 27, Iss 23, p 8137 (2022)
A series of previously synthesized 5-benzyliden-2-(5-methylthiazole-2-ylimino)thiazoli- din-4-one were evaluated for their anti-inflammatory activity on the basis of PASS predictive outcomes. The predictive compounds were found to demonstrate moderat
Externí odkaz:
https://doaj.org/article/633e7aebcc864b4eadfedf76439abe3c
Autor:
Nagaraja Sreeharsha, Samathoti Prasanthi, Satyavarapu Veera Venkata Naga Satya Mahalakshmi, Prakash S. Goudanavar, Nimbagal Raghavendra Naveen, Buduru Gowthami, Santosh Fattepur, Girish Meravanige, Syed Mohammed Basheeruddin Asdaq, Md. Khalid Anwer, Bandar Aldhubiab, Mohammed Monirul Islam, Mohammed Habeebuddin, Mallikarjun Telsang, Mazen Al Gharsan, Michelyne Haroun
Publikováno v:
Molecules, Vol 27, Iss 22, p 7914 (2022)
A brand-new nano-crystal (NC) version of the hydrophobic drug Paclitaxel (PT) were formulated for cancer treatment. A stable NC formulation for the administration of PT was created using the triblock co-polymer Pluronic F127. To achieve maximum entra
Externí odkaz:
https://doaj.org/article/f75fe324ecf048c9a3407b3e9c2081f6
Autor:
Katharigatta N. Venugopala, Nizar A. Al-Shar’i, Lina A. Dahabiyeh, Wafa Hourani, Pran Kishore Deb, Melendhran Pillay, Bashaer Abu-Irmaileh, Yasser Bustanji, Sandeep Chandrashekharappa, Christophe Tratrat, Mahesh Attimarad, Anroop B. Nair, Nagaraja Sreeharsha, Pottathil Shinu, Michelyne Haroun, Mahmoud Kandeel, Abdulmalek Ahmed Balgoname, Rashmi Venugopala, Mohamed A. Morsy
Publikováno v:
Antibiotics, Vol 11, Iss 7, p 831 (2022)
A series of 2,3-dihydroquinazolin-4(1H)-one derivatives (3a–3m) was screened for in vitro whole-cell antitubercular activity against the tubercular strain H37Rv and multidrug-resistant (MDR) Mycobacterium tuberculosis (MTB) strains. Compounds 3l an
Externí odkaz:
https://doaj.org/article/6cf9acd88ee14653afc00830d58d75af
Autor:
Michelyne Haroun, Santosh S. Chobe, Rajasekhar Reddy Alavala, Savita M. Mathure, Risy Namratha Jamullamudi, Charushila K. Nerkar, Vijay Kumar Gugulothu, Christophe Tratrat, Mohammed Monirul Islam, Katharigatta N. Venugopala, Mohammed Habeebuddin, Mallikarjun Telsang, Nagaraja Sreeharsha, Md. Khalid Anwer
Publikováno v:
Molecules, Vol 27, Iss 12, p 3757 (2022)
Considering the importance of benzothiazepine pharmacophore, an attempt was carried out to synthesize novel 1,5-benzothiazepine derivatives using polyethylene glycol-400 (PEG-400)-mediated pathways. Initially, different chalcones were synthesized and
Externí odkaz:
https://doaj.org/article/f9a0fe7beef040fcbf57ec2267aec8e1
Autor:
Geronikaki Athina, Christophe Tratrat, Anthi Petrou, Maria Fesatidou, Michelyne Haroun, Katharigatta Venugopala, Nagaraja Sreeharsha, Jad Chemali
Publikováno v:
Current Topics in Medicinal Chemistry. 23:520-538
Abstract: Viral infections range from self-limiting to more serious and fatal infections; therefore, some viral infections are of great public health concern worldwide, e.g., Hepatitis B virus, Hepatitis C virus, and HIV. Recently, the world faced a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b18d8f253af3972cd7064651b5dea7db
https://doi.org/10.2174/1568026623666230325153927
https://doi.org/10.2174/1568026623666230325153927
Autor:
Katharigatta N. Venugopala, Pottathil Shinu, Christophe Tratrat, Pran Kishore Deb, Raquel M. Gleiser, Sandeep Chandrashekharappa, Deepak Chopra, Mahesh Attimarad, Anroop B. Nair, Nagaraja Sreeharsha, Fawzi M. Mahomoodally, Michelyne Haroun, Mahmoud Kandeel, Syed Mohammed Basheeruddin Asdaq, Viresh Mohanlall, Nizar A. Al-Shar’i, Mohamed A. Morsy
Publikováno v:
Molecules, Vol 27, Iss 9, p 2676 (2022)
Alteration of insect growth regulators by the action of inhibitors is becoming an attractive strategy to combat disease-transmitting insects. In the present study, we investigated the larvicidal effect of 1,2,3-triazolyl-pyrimidinone derivatives agai
Externí odkaz:
https://doaj.org/article/93c72a09147b4eaa9ec3e683e05a5128
Autor:
Christophe Tratrat, Anthi Petrou, Athina Geronikaki, Marija Ivanov, Marina Kostić, Marina Soković, Ioannis S. Vizirianakis, Nikoleta F. Theodoroula, Michelyne Haroun
Publikováno v:
Molecules, Vol 27, Iss 6, p 1930 (2022)
Herein, we report computational and experimental evaluations of the antimicrobial activity of twenty one 2,3-diaryl-thiazolidin-4-ones. All synthesized compounds exhibited an antibacterial activity against six Gram-positive and Gram-negative bacteria
Externí odkaz:
https://doaj.org/article/f8bb2151bf9d4c1e95d0422c5f1ec871
Autor:
Michelyne Haroun, Christophe Tratrat, Anthi Petrou, Athina Geronikaki, Marija Ivanov, Ana Ćirić, Marina Soković, Sreeharsha Nagaraja, Katharigatta Narayanaswamy Venugopala, Anroop Balachandran Nair, Heba S. Elsewedy, Hafedh Kochkar
Publikováno v:
Molecules, Vol 26, Iss 13, p 4061 (2021)
Background: Infectious diseases still affect large populations causing significant morbidity and mortality. Bacterial and fungal infections for centuries were the main factors of death and disability of millions of humans. Despite the progress in the
Externí odkaz:
https://doaj.org/article/0f62d5fd50d4408dbcf8ec1b77089a30