Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Michela Di Mattia"'
Autor:
Ilaria D’Acquarica, Francesco Gasparrini, Dorina Kotoni, Marco Pierini, Claudio Villani, Walter Cabri, Michela Di Mattia, Fabrizio Giorgi
Publikováno v:
Molecules, Vol 15, Iss 3, Pp 1309-1323 (2010)
Since its identification in the early 1970s, artemisinin, as well as semi-synthetic derivatives and synthetic trioxanes, have been used in malaria therapy. Reduction of artemisinin by NaBH4 produced dihydroartemisinin (DHA), and yielded a new stereoc
Externí odkaz:
https://doaj.org/article/990ad2397d0e4bdf87d5820bcb0baf29
Autor:
Francesco Gasparrini, Patrizia Simone, M.G. Quaglia, Fabrizio Giorgi, Marta Di Iorio, Andrea Mazzanti, Ilaria D'Acquarica, Walter Cabri, Marco Pierini, Michela Di Mattia, Claudio Villani
Publikováno v:
The Journal of Organic Chemistry. 76:4831-4840
Artemisinin or qinghaosu has now largely given way to the more potent dihydroartemisinin (DHA, 1) and its derivatives in the treatment of drug-resistant malaria, in combination with other classical antimalarial drugs. DHA is obtained by NaBH(4) reduc
Feed additives in animal nutrition: Quantification of a new adrenergic drug by hyphenated techniques
Autor:
Gianfranco Brambilla, Beatrice Bocca, Claudia Cartoni, Marialinda Felli, Bruno Neri, Maurizio Fiori, Mario Vincenzo Russo, Michela Di Mattia
Publikováno v:
Journal of Separation Science. 26:363-368
Zilpaterol, (±)-trans-4,5,6,7-tetrahydro-7-hydroxy-6-(isopropylamino) imidazo [4,5,1-jk]-[1]benzazepin-2(1H)-one, is an adrenergic agonist drug licensed in Mexico and South Africa as feed additive for cattle at slaughter age. In contrast, the EU leg
Autor:
Patrizia Simone, Fabrizio Giorgi, Walter Cabri, Michela Di Mattia, Francesco Gasparrini, Ilaria D'acquarica, Andrea Mazzanti, Marco Pierini, M.G. Quaglia, Marta Di Iorio, Claudio Villani
Artemisinin (Qinghaosu, 1) is a sesquiterpene lactone endoperoxide isolated from Artemisia annua L. that Chinese herbalists have traditionally used to treat malaria. Reduction of artemisinin by NaBH(4) produced dihydroartemisinin (DHA, 2) and yielded
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2b8b9a2d9af8481e0240dda5c28eb204
http://hdl.handle.net/11573/354195
http://hdl.handle.net/11573/354195
Autor:
Dorina Kotoni, Claudio Villani, Ilaria D'Acquarica, Walter Cabri, Fabrizio Giorgi, Marco Pierini, Francesco Gasparrini, Michela Di Mattia
Publikováno v:
Molecules
Molecules, Vol 15, Iss 3, Pp 1309-1323 (2010)
Molecules, Vol 15, Iss 3, Pp 1309-1323 (2010)
Since its identification in the early 1970s, artemisinin, as well as semi-synthetic derivatives and synthetic trioxanes, have been used in malaria therapy. Reduction of artemisinin by NaBH(4) produced dihydroartemisinin (DHA), and yielded a new stere
Autor:
Gianluca Giorgi, Samantha Zanoli, Michela Di Mattia, Anna Ramunno, Giuseppe Campiani, Stefania Butini, Sandra Gemma, Alberto Bergamini, Salvatore Sanna Coccone, Giuseppe Borrelli, Sandro Cosconati, Luciana Marinelli, Margherita Brindisi, Alberta Samuele, Bruno Galletti, Ettore Novellino, Giovanni Maga, Silvana Lalli
Starting from the prototypic compound 4, we describe new, potent, and broad-spectrum pyrrolobenzo(py-rido)oxazepinones antivirals. A biochemical and enzymological investigation was performed for defining their mechanism of inhibition at either recomb
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::454e0a9f045019b65519412b67085301
http://hdl.handle.net/11365/3650
http://hdl.handle.net/11365/3650
Autor:
Francesco Gasparrini, Ilaria D'Acquarica, Silvana Lalli, Alessia Ciogli, Bruno Galletti, Marco Pierini, Michela Di Mattia, Patrizia Simone, Fabrizio Giorgi, Walter Cabri
We developed a cryo-HPLC/UV method for the simultaneous determination of artemisinin (1), alpha-dihydroartemisinin (2 alpha), beta-dihydroartemisinin (2 beta). and a ubiquitous thermal decomposition product of 2 (designated as diketoaldehyde, 3), sta
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5e8b5819e1e2ede5ea775b2a30046017
http://hdl.handle.net/11585/756766
http://hdl.handle.net/11585/756766
Autor:
Stefania Butini, Margherita Brindisi, Sandro Cosconati, Luciana Marinelli, Giuseppe Borrelli, Salvatore Sanna Coccone, Anna Ramunno, Giuseppe Campiani, Ettore Novellino, Samantha Zanoli, Alberta Samuele, Gianluca Giorgi, Alberto Bergamini, Michela Di Mattia, Silvana Lalli, Bruno Galletti, Sandra Gemma, Giovanni Maga
Publikováno v:
Journal of Medicinal Chemistry; Feb2009, Vol. 52 Issue 4, p1224-1228, 5p
Autor:
Beatrice Bocca, Claudia Cartoni, Michela Di Mattia, Maurizio Fiori, Marialinda Felli, Bruno Neri, Mario Vincenzo Russo
Publikováno v:
Journal of Separation Science; Apr2003, Vol. 26 Issue 5, p363-368, 6p