Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Michal Šarkan"'
Autor:
Ľudevít Kádaši, Michal Šarkan, Klaudia Kyselicová, Csaba Bognar, Radoslav Beňuš, Marian Baldovic, Lukáš Šebest
Publikováno v:
Biologia. 71:613-619
DNA was extracted using a Silica Bead Extraction kit from bone samples taken from a Slavonic-Avar individual found at the archaeological site of Cifer-Pac. The analysed skeletal remains from the grave number 62/79 belong to a young adult male (20–3
Autor:
Rohit Tiwari, Katarína Mikušová, Giorgia Mori, Michal Šarkan, Allen G. Oliver, Laurent R. Chiarelli, Scott G. Franzblau, Ivana Centárová, Marvin J. Miller, Patricia A. Miller, Sang-Hyun Cho
Publikováno v:
ACS Medicinal Chemistry Letters. 7:266-270
Electron deficient nitroaromatic compounds such as BTZ043 and its closest congener, PBTZ169, and related agents are a promising new class of anti-TB compounds. Herein we report the design and syntheses of 1,3-benzothiazinone azide (BTZ-N3) and relate
Autor:
Ruben C. Hartkoorn, Anthony Vocat, Katarína Mikušová, Elena Kazakova, João Neres, Trent M. Conroy, O. B. Ryabova, Jérémie Piton, Michal Šarkan, Vadim Makarov, Stanislav Huszár, Gaëlle S. Kolly, Stewart T. Cole
8-Nitro-benzothiazinones (BTZs), such as BTZ043 and PBTZ169, inhibit decaprenylphosphoryl-β- d -ribose 2′-oxidase (DprE1) and display nanomolar bactericidal activity against Mycobacterium tuberculosis in vitro . Structure-activity relationship (SA
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::30730f59186b1402cb4ef1f895a65322
https://infoscience.epfl.ch/record/213880
https://infoscience.epfl.ch/record/213880
Autor:
Anthony Vocat, Jan Němeček, Věra Klimešová, Ivana Centárová, Michal Šarkan, Jiřina Stolaříková, Ivona Pavkova, Júlia Zemanová, Kateřina Vávrová, Katarína Mikušová, Stewart T. Cole, Alexandr Hrabálek, Patrik Čonka, Galina Karabanovich, Jaroslav Roh, Rita Székely, Tomáš Smutný, Petr Pavek, Marcela Vejsova
Herein, we report the discovery and structure activity relationships of 5-substituted-2-[(3,5-dinitrobenzyl)-sulfanyl]-1,3,4-oxadiazoles and 1,3,4-thiadiazoles as a new class of antituberculosis agents. The majority of these compounds exhibited outst
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f7f30a60187d8a3d4d646eae257ee63b
https://infoscience.epfl.ch/record/219388
https://infoscience.epfl.ch/record/219388
Autor:
Katarína Mikušová, Veronika Mokosova, Miroslav Brecik, Stewart T. Cole, Emoeke Kilacskova, Raju Mukherjee, Adela Bobovská, João Neres, Ivana Centárová, Jana Korduláková, Stanislav Huszár, Michal Šarkan, Zuzana Svetlíková, Gaëlle S. Kolly
The flavo-enzyme DprE1 catalyzes a key epimerization step in the decaprenyl-phosphoryl d-arabinose (DPA) pathway, which is essential for mycobacterial cell wall biogenesis and targeted by several new tuberculosis drug candidates. Here, using differen
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f63164c0af086c942318eef104bf68ec
https://infoscience.epfl.ch/record/212241
https://infoscience.epfl.ch/record/212241