New Generation Dopaminergic Agents. 6. Structure−Activity Relationship Studies of a Series of 4-(Aminoethoxy)indole and 4-(Aminoethoxy)indolone Derivatives Based on the Newly Discovered 3-Hydroxyphenoxyethylamine D2 Template

Autor: Mewshaw, R. E., Webb, M. B., Marquis, K. L., McGaughey, G. B., Shi, X., Wasik, T., Scerni, R., Brennan, J. A., Andree, T. H.

Publikováno v: Journal of Medicinal Chemistry; June 3, 1999, Vol. 42 Issue: 11 p2007-2020, 14p

pi-Stacking interactions. Alive and well in proteins.

Autor: McGaughey, G B, Gagné, M, Rappé, A K

Publikováno v: Journal of Biological Chemistry; June 1998, Vol. 273 Issue: 25 p15458-63, 6p

ChemInform Abstract: New Generation Dopaminergic Agents. Part 5. Heterocyclic Bioisosteres That Exploit the 3-OH-N¹-Phenylpiperazine Dopaminergic Template.

Autor: MEWSHAW, R. E., VERWIJS, A., SHI, X., MCGAUGHEY, G. B., NELSON, J. A., MAZANDARANI, H., BRENNAN, J. A., MARQUIS, K. L., COUPET, J., ANDREE, T. H.

Publikováno v: ChemInform; Feb1999, Vol. 30 Issue 8, pno-no, 1p

HIV-1 vaccine development: constrained peptide immunogens show improved binding to the anti-HIV-1 gp41 MAb.

Autor: McGaughey GB; Department of Molecular Systems, Merck Research Laboratories, P.O. Box 4, West Point, Pennsylvania 19486, USA. michael_bogusky@merck.com, Citron M, Danzeisen RC, Freidinger RM, Garsky VM, Hurni WM, Joyce JG, Liang X, Miller M, Shiver J, Bogusky MJ

Publikováno v: Biochemistry [Biochemistry] 2003 Mar 25; Vol. 42 (11), pp. 3214-23.

New generation dopaminergic agents. 6. Structure-activity relationship studies of a series of 4-(aminoethoxy)indole and 4-(aminoethoxy)indolone derivatives based on the newly discovered 3-hydroxyphenoxyethylamine D2 template.

Autor: Mewshaw RE; Global Chemical Sciences and CNS Disorders Departments, Wyeth-Ayerst Research Laboratories, CN 8000, Princeton, New Jersey 08543-8000, USA., Webb MB, Marquis KL, McGaughey GB, Shi X, Wasik T, Scerni R, Brennan JA, Andree TH

Publikováno v: Journal of medicinal chemistry [J Med Chem] 1999 Jun 03; Vol. 42 (11), pp. 2007-20.