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Autor:
Miriam Carr, Daniela M. Zisterer, Niamh M. O’Boyle, Balázs Sarkadi, Mary J. Meegan, Aisling Croke, David Lloyd, Seema M. Nathwani, Peig Carroll, Lisa M. Greene, Mark Lawler, Anthony M. McElligott, Eibhlin Conneally, Niall O. Keely, Sandra A. Bright, Maria Gagliardi, Lisa M. O’Connor, Darren Fayne
Publikováno v:
Journal of Pharmacology and Experimental Therapeutics. 335:302-313
Combretastatin-A4 (CA-4) is a natural derivative of the African willow tree Combretum caffrum. CA-4 is one of the most potent antimitotic components of natural origin, but it is, however, intrinsically unstable. A novel series of CA-4 analogs incorpo
Autor:
McKeown JP; School of Pharmacy and Pharmaceutical Sciences, Panoz Institute, Trinity College, The University of Dublin, East End 4/5, Dublin 2, D02 PN40 Dublin, Ireland.; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Byrne AJ; School of Pharmacy and Pharmaceutical Sciences, Panoz Institute, Trinity College, The University of Dublin, East End 4/5, Dublin 2, D02 PN40 Dublin, Ireland.; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Bright SA; School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Charleton CE; School of Pharmacy and Pharmaceutical Sciences, Panoz Institute, Trinity College, The University of Dublin, East End 4/5, Dublin 2, D02 PN40 Dublin, Ireland.; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Kandwal S; Molecular Design Group, School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland.; Molecular Design Group, School of Chemical Sciences, Dublin City University, Glasnevin, D09 V209 Dublin, Ireland.; DCU Life Sciences Institute, Dublin City University, Glasnevin, D09 V209 Dublin, Ireland., Čmelo I; Molecular Design Group, School of Chemical Sciences, Dublin City University, Glasnevin, D09 V209 Dublin, Ireland.; DCU Life Sciences Institute, Dublin City University, Glasnevin, D09 V209 Dublin, Ireland., Twamley B; School of Chemistry, Trinity College Dublin, Dublin 2, D02 P3X2 Dublin, Ireland., McElligott AM; Discipline of Haematology, School of Medicine, Trinity Translational Medicine Institute, St. James's Hospital and Trinity College, Dublin 8, D08 W9RT Dublin, Ireland., Fayne D; Molecular Design Group, School of Chemical Sciences, Dublin City University, Glasnevin, D09 V209 Dublin, Ireland.; DCU Life Sciences Institute, Dublin City University, Glasnevin, D09 V209 Dublin, Ireland., O'Boyle NM; School of Pharmacy and Pharmaceutical Sciences, Panoz Institute, Trinity College, The University of Dublin, East End 4/5, Dublin 2, D02 PN40 Dublin, Ireland.; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Williams DC; School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Meegan MJ; School of Pharmacy and Pharmaceutical Sciences, Panoz Institute, Trinity College, The University of Dublin, East End 4/5, Dublin 2, D02 PN40 Dublin, Ireland.; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland.
Publikováno v:
Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2024 Aug 05; Vol. 17 (8). Date of Electronic Publication: 2024 Aug 05.
Autor:
Byrne AJ; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Bright SA; School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., McKeown JP; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Bergin A; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Twamley B; School of Chemistry, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., McElligott AM; Discipline of Haematology, School of Medicine, Trinity Translational Medicine Institute, St. James's Hospital and Trinity College, Dublin 8, D08 W9RT Dublin, Ireland., Noorani S; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Kandwal S; School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Fayne D; School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., O'Boyle NM; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Williams DC; School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland., Meegan MJ; School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse St, Dublin 2, D02 R590 Dublin, Ireland.
Publikováno v:
Molecules (Basel, Switzerland) [Molecules] 2023 Dec 14; Vol. 28 (24). Date of Electronic Publication: 2023 Dec 14.
Autor:
Brophy S; The John Durkan Leukaemia Laboratory, Trinity Translational Medicine Institute, Trinity College and St James's Hospital, Dublin, Ireland., Amet R; The John Durkan Leukaemia Laboratory, Trinity Translational Medicine Institute, Trinity College and St James's Hospital, Dublin, Ireland., Foy-Stones H; Cryobiology Laboratory Stem Cell Facility, St James's Hospital, Dublin, Ireland., Gardiner N; Cryobiology Laboratory Stem Cell Facility, St James's Hospital, Dublin, Ireland., McElligott AM; The John Durkan Leukaemia Laboratory, Trinity Translational Medicine Institute, Trinity College and St James's Hospital, Dublin, Ireland. tony.mcelligott@tcd.ie.; Trinity St. James's Cancer Institute, Trinity College and St James's Hospital, Dublin, Ireland. tony.mcelligott@tcd.ie.
Publikováno v:
Methods in molecular biology (Clifton, N.J.) [Methods Mol Biol] 2023; Vol. 2645, pp. 179-187.