Palosuran inhibits binding to primate UT receptors in cell membranes but demonstrates differential activity in intact cells and vascular tissues.

Autor: Behm, D. J.¹ david.j.behm@gsk.com, McAtee, J. J.², Dodson, J. W.², Neeb, M. J.², Fries, H. E.³, Evans, C. A.³, Hernandez, R. R.⁴, Hoffman, K. D.⁴, Harrison, S. M.⁵, Lai, J. M.¹, Wu, C.¹, Aiyar, N. V.¹, Ohlstein, E. H.¹, Douglas, S. A.¹

Publikováno v: British Journal of Pharmacology. Oct2008, Vol. 155 Issue 3, p374-386. 13p. 1 Diagram, 6 Charts, 8 Graphs.

Synthesis and Biological Evaluation of 2‘,3‘-Didehydro-2‘,3‘-dideoxy-5- fluorocytidine (D4FC) Analogues:  Discovery of Carbocyclic Nucleoside Triphosphates with Potent Inhibitory Activity against HIV-1 Reverse Transcriptase¹

Autor: Shi, J., McAtee, J. J., Wirtz, S. Schlueter, Tharnish, P., Juodawlkis, A., Liotta, D. C., Schinazi, R. F.

Publikováno v: Journal of Medicinal Chemistry; March 11, 1999, Vol. 42 Issue: 5 p859-867, 9p

First and second generation total synthesis of the teicoplanin aglycon.

Autor: Boger DL; Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA., Kim SH, Mori Y, Weng JH, Rogel O, Castle SL, McAtee JJ

Publikováno v: Journal of the American Chemical Society [J Am Chem Soc] 2001 Mar 07; Vol. 123 (9), pp. 1862-71.