Zobrazeno 1 - 10 of 28 pro vyhledávání: '"Matteo, Falsini"'
1
Akademický článek
The role of 5-arylalkylamino- and 5-piperazino- moieties on the 7-aminopyrazolo[4,3-d]pyrimidine core in affecting adenosine A1 and A2A receptor affinity and selectivity profiles
Autor: Lucia Squarcialupi, Marco Betti, Daniela Catarzi, Flavia Varano, Matteo Falsini, Annalisa Ravani, Silvia Pasquini, Fabrizio Vincenzi, Veronica Salmaso, Mattia Sturlese, Katia Varani, Stefano Moro, Vittoria Colotta
Publikováno v: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 32, Iss 1, Pp 248-263 (2017)
New 7-amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives, substituted at the 5-position with aryl(alkyl)amino- and 4-substituted-piperazin-1-yl- moieties, were synthesized with the aim of targeting human (h) adenosine A1 and/or A2A receptor subtypes
Externí odkaz: https://doaj.org/article/3becb9391fc64475b2620dd24841af0a
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2
Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A
Autor: Tasia, Amelia, Jacobus P D, van Veldhoven, Matteo, Falsini, Rongfang, Liu, Laura H, Heitman, Gerard J P, van Westen, Elena, Segala, Grégory, Verdon, Robert K Y, Cheng, Robert M, Cooke, Daan, van der Es, Adriaan P, IJzerman
Publikováno v: Journal of Medicinal Chemistry
In this study, we determined the crystal structure of an engineered human adenosine A2A receptor bound to a partial agonist and compared it to structures cocrystallized with either a full agonist or an antagonist/inverse agonist. The interaction betw
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::d1106f4cb522305aba0e4d49b33d5633
https://pubmed.ncbi.nlm.nih.gov/33764785
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3
Crystal structure and subsequent ligand design of a nonriboside partial agonist bound to the adenosine A2A receptor
Autor: Tasia Amelia, Robert K. Y. Cheng, Gerard J. P. van Westen, Rongfang Liu, Elena Segala, Robert M. Cooke, Laura H. Heitman, Jacobus P. D. van Veldhoven, Daan van der Es, Matteo Falsini, Grégory Verdon, Adriaan P. IJzerman
Publikováno v: Journal of Medicinal Chemistry, 64(7), 3827-3842. American Chemical Society (ACS)
Journal of Medicinal Chemistry
In this study, we determined the crystal structure of an engineered human adenosine A2A receptor bound to a partial agonist and compared it to structures cocrystallized with either a full agonist or an antagonist/inverse agonist. The interaction betw
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a3eaee9ee24339f7b4772a78e3323223
http://hdl.handle.net/1887/3204468
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5
The role of 5-arylalkylamino- and 5-piperazino- moieties on the 7-aminopyrazolo[4,3-d]pyrimidine core in affecting adenosine A1 and A2A receptor affinity and selectivity profiles
Autor: Silvia Pasquini, Veronica Salmaso, Matteo Falsini, Stefano Moro, Daniela Catarzi, Annalisa Ravani, Fabrizio Vincenzi, Lucia Squarcialupi, Mattia Sturlese, Flavia Varano, Katia Varani, Marco Betti, Vittoria Colotta
Publikováno v: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 32, Iss 1, Pp 248-263 (2017)
New 7-amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives, substituted at the 5-position with aryl(alkyl)amino- and 4-substituted-piperazin-1-yl- moieties, were synthesized with the aim of targeting human (h) adenosine A1 and/or A2A receptor subtypes
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fdf7dd71d812ffdd28de7a08f7657a04
https://doi.org/10.1080/14756366.2016.1247060
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6
Solutions for Seal Gas Leakages Recovery in Methane Compression: Integration into Processing Lines or Gas Valorization Systems
Autor: Matteo Falsini, Luca Scarbolo, Sergio Cipriani, Filippo Conforti
Publikováno v: Day 2 Wed, September 04, 2019.
Recovery and valorization of wasted gas associated to methane processing (i.e. leakages from rotating equipment and flared gas) has usually been avoided due to the inherently limited amount of gas of these streams. Moreover, the technical complexitie
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::5c17b8d2d206e434c7ebd2be72b46d56
https://doi.org/10.2118/195759-ms
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8
Smart Integration of Natural Gas Valorization Systems and Flexible Plant Installation in Existing and Low Capacity Gas Production Sites
Autor: Filippo Conforti, Matteo Falsini
Publikováno v: Day 2 Tue, May 07, 2019.
The increasing demand of energy efficiency, the evolution of emission regulatory and the limited investments allocation, increases the attractiveness for flexible gas valorization systems [GGFR]. Gas valorization system can be considered all the tech
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::17940e67033fcfef652b417856643408
https://doi.org/10.4043/29551-ms
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