Výsledky vyhledávání - "Mathieu Danel"

Akademický článek

Synthesis, In Silico, and In Vitro Evaluation of Anti-Leishmanial Activity of Oxadiazoles and Indolizine Containing Compounds Flagged against Anti-Targets

Autor: Strahinja Stevanovic, Milan Sencanski, Mathieu Danel, Christophe Menendez, Roumaissa Belguedj, Abdelmalek Bouraiou, Katarina Nikolic, Sandrine Cojean, Philippe M. Loiseau, Sanja Glisic, Michel Baltas, Alfonso T. García-Sosa

Publikováno v: Molecules, Vol 24, Iss 7, p 1282 (2019)

Due to the lack of approved vaccines against human leishmaniasis and the limitations of the current chemotherapy inducing side effects and drug resistance, development of new, effective chemotherapeutic agents is essential. This study describes the s

Externí odkaz: https://doaj.org/article/df39e0b494e14ea1ae0280a0c717ab36

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A Coumarin-Based Analogue of Thiacetazone as Dual Covalent Inhibitor and Potential Fluorescent Label of HadA in Mycobacterium tuberculosis

Autor: Antonio Peixoto, Monika Záhorszká, Jana Korduláková, Mathieu Danel, Fernanda Goncalves, Elodie Vega, Asma Farjallah, Maria Rosalia Pasca, Mary Jackson, Giulia Degiacomi, Laurent R. Chiarelli, Cendrine Seguin, Martin Forbak, Christian Lherbet, Stefan Chassaing, Chantal Carayon, Souhir Abid, Marco Fumagalli, Anna E. Grzegorzewicz

Publikováno v: ACS Infectious Diseases
ACS Infectious Diseases, American Chemical Society, 2021, 7 (3), pp.552-565. ⟨10.1021/acsinfecdis.0c00325⟩
ACS Infectious Diseases, 2021, 7 (3), pp.552-565. ⟨10.1021/acsinfecdis.0c00325⟩

International audience; A novel coumarin-based molecule, designed as a fluorescent surrogate of a thiacetazone-derived antitubercular agent, was quickly and easily synthesized from readily available starting materials. This small molecule, coined Cou

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9a5b5cd98cba63d79872ca55f29014c7
https://hal.archives-ouvertes.fr/hal-03209886/document

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Chan–Lam-Type C–N Cross-Coupling Reactions under Base- and Ligand-Free CuI-Zeolite Catalysis

Autor: Mathieu Danel, Randa Sakly, Tony Garnier, Stefan Chassaing, Patrick Pale

Publikováno v: Synthesis. 49:1223-1230

Various representative copper(I)-exchanged zeolites were investigated for their catalytic potential in Chan–Lam cross-coupling reactions. CuI-USY appeared as the best catalyst and proved to efficiently promote C–N cross-coupling processes under a

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::c3ce1256f025723f2b4be036885d401a
https://doi.org/10.1055/s-0036-1588652

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Synthesis and multistate characterization of bis-flavylium dications – symmetric resorcinol- and phloroglucinol-type derivatives as stochastic systems

Autor: João Avó, Tony Garnier, Stefan Chassaing, Mathieu Danel, Fernando Pina, Nuno Basílio

Publikováno v: RSC Advances. 6:69698-69707

Two symmetric bis-flavylium dications were readily synthesized and further evaluated for their multistate profile. Both systems were shown to be fully stochastic and behave like a single compound suggesting that the two flavylium moieties do not comm

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::3cc1ede1f8979159c1336bc68b6b4a08
https://doi.org/10.1039/c6ra12017b

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Copper(I)-USY as a Ligand-Free and Recyclable Catalyst for Ullmann-Type O-, N-, S-, and C-Arylation Reactions: Scope and Application to Total Synthesis

Autor: Patrick Pale, Tony Garnier, Stefan Chassaing, Valérie Bénéteau, Anthony Pujol, Mathieu Danel, Valentin Magné

Publikováno v: The Journal of organic chemistry. 83(12)

The copper(I)-doped zeolite CuI-USY proved to be a versatile, efficient, and recyclable catalyst for various Ullmann-type coupling reactions. Easy to prepare and cheap, this catalytic material enables the arylation and heteroarylation of diverse O-,

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::33a97daf2f13805bfbc326b2b18b7528
https://pubmed.ncbi.nlm.nih.gov/29790337

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6,6′-Dimethyl-2,2′-bipyridine-4-ester: A pivotal synthon for building tethered bipyridine ligands

Autor: Nadine Leygue, Fabien Havas, Mathieu Danel, Claude Picard, Béatrice Mestre, Chantal Galaup

Publikováno v: Tetrahedron. 65:7673-7686

We describe an efficient and scalable synthesis of 4-carbomethoxy-6,6′-dimethyl-2,2′-bipyridine starting from easily available substituted 2-halopyridines and based on the application of modified Negishi cross-coupling conditions. This compound i

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::1c5c1ef062443b1012b6ccef7fb227bf
https://doi.org/10.1016/j.tet.2009.06.111

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New Amino Endoperoxides Belonging to the Antimalarial G-Factor Series

Autor: Christiane André-Barrès, Virginie Bernat, Cécile Givelet, Henri Vial, Mathieu Danel

Publikováno v: European Journal of Organic Chemistry. 2007:3095-3101

In the search for new antimalarial endoperoxides we developed a direct route for the preparation of new amino compounds belonging to the G-factor series. During the synthesis, a significant difference in reactivity between two series of diastereoisom

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::1eda6840ef1d777241a88cd53d24f523
https://doi.org/10.1002/ejoc.200700086

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A convenient synthesis of 6,6′-dimethyl-2,2′-bipyridine-4-ester and its application to the preparation of bifunctional lanthanide chelators

Autor: Mathieu Danel, Chantal Galaup, Fabien Havas, Pierre Tisnès, Claude Picard

Publikováno v: Tetrahedron Letters. 48:999-1002

We describe a convenient scalable synthesis of 4-carbomethoxy-6,6′-dimethyl-2,2′-bipyridine based on the application of modified Negishi cross-coupling conditions. The use of this building block in the preparation of a number of dissymmetrically

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::5315fef080ee3f57fb7cc532671c2355
https://doi.org/10.1016/j.tetlet.2006.12.012

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Cu I –USY as a Ligand-Free and Recyclable Catalytic System for the Ullmann-Type Diaryl Ether Synthesis

Autor: Tony Garnier, Stefan Chassaing, Valentin Magné, Mathieu Danel, Patrick Pale

Publikováno v: Organic Letters
Organic Letters, American Chemical Society, 2015, 17 (18), pp.4494-4497. ⟨10.1021/acs.orglett.5b02167⟩

The catalytic potential of copper(I)-exchanged zeolites was evaluated in the Ullmann-type synthesis of diaryl ethers. Among four investigated zeolites (i.e., USY, MOR, β, and ZSM5), Cu(I)-USY was the best catalyst and proved efficient under ligand-f

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::34ac96408d34e05f7fd25b7ddade6314
https://hal.archives-ouvertes.fr/hal-02062181

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