Zobrazeno 1 - 10
of 24
pro vyhledávání: '"Matheson, CJ"'
Autor:
Matheson, CJ, Coxon, CR, Bayliss, R, Boxall, K, Carbain, B, Fry, AM, Hardcastle, IR, Harnor, SJ, Mas-Droux, C, Newell, DR, Richards, MW, Sivaprakasam, M, Turner, D, Griffin, RJ, Golding, BT, Cano, C
Renewed interest in covalent inhibitors of enzymes implicated in disease states has afforded several agents targeted at protein kinases of relevance to cancers. We now report the design, synthesis and biological evaluation of 6-ethynylpurines that ac
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=core_ac_uk__::50079741394e01f4bd1b1137f16bfc2a
https://eprints.whiterose.ac.uk/160431/19/d0md00074d.pdf
https://eprints.whiterose.ac.uk/160431/19/d0md00074d.pdf
Autor:
Coxon, CR, Wong, C, Bayliss, RWA, Boxall, K, Carr, KH, Fry, AM, Hardcastle, IR, Matheson, CJ, Newell, DR, Sivaprakasam, M, Thomas, H, Turner, D, Yeoh, S, Wang, LZ, Griffin, RJ, Golding, BT, Cano, C
Publikováno v:
Oncotarget
Nek2 (NIMA-related kinase 2) is a cell cycle-dependent serine/threonine protein kinase that regulates centrosome separation at the onset of mitosis. Overexpression of Nek2 is common in human cancers and\ud suppression can restrict tumor cell growth a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::2a81c9e348a99e3a06a93c16991f5ec9
Autor:
Warfield BM; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States.
Publikováno v:
Data in brief [Data Brief] 2021 Sep 25; Vol. 38, pp. 107433. Date of Electronic Publication: 2021 Sep 25 (Print Publication: 2021).
Autor:
Warfield BM; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., McArthur DG; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States.
Publikováno v:
ACS chemical neuroscience [ACS Chem Neurosci] 2021 Sep 15; Vol. 12 (18), pp. 3477-3486. Date of Electronic Publication: 2021 Sep 02.
N-Substituted pyrrolopyrimidines and purines as p90 ribosomal S6 protein kinase-2 (RSK2) inhibitors.
Autor:
Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Warfield BM; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA. Electronic address: philip.reigan@cuanschutz.edu.
Publikováno v:
Bioorganic & medicinal chemistry [Bioorg Med Chem] 2021 Jul 01; Vol. 41, pp. 116220. Date of Electronic Publication: 2021 May 19.
Autor:
Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Minhajuddin M; Division of Hematology, University of Colorado Anschutz Medical Campus, 12700 E 19th Avenue, Aurora, CO, 80045, USA., Jordan CT; Division of Hematology, University of Colorado Anschutz Medical Campus, 12700 E 19th Avenue, Aurora, CO, 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA. Electronic address: philip.reigan@cuanschutz.edu.
Publikováno v:
European journal of medicinal chemistry [Eur J Med Chem] 2020 Jul 01; Vol. 197, pp. 112316. Date of Electronic Publication: 2020 Apr 16.
Autor:
Matheson CJ; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Coxon CR; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Bayliss R; School of Molecular and Cellular Biology , The Astbury Centre for Structural Molecular Biology , University of Leeds , UK.; Section of Structural Biology , The Institute of Cancer Research , Sutton , UK., Boxall K; Cancer Research UK Cancer Therapeutics Unit , The Institute of Cancer Research , Sutton , UK., Carbain B; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Fry AM; School of Molecular and Cellular Biology , The Astbury Centre for Structural Molecular Biology , University of Leeds , UK., Hardcastle IR; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Harnor SJ; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Mas-Droux C; Section of Structural Biology , The Institute of Cancer Research , Sutton , UK., Newell DR; Cancer Research UK Newcastle Drug Discovery Unit , Translational and Clinical Research Institute , Newcastle University Centre for Cancer , Faculty of Medical Sciences , Newcastle University , Newcastle upon Tyne , UK., Richards MW; School of Molecular and Cellular Biology , The Astbury Centre for Structural Molecular Biology , University of Leeds , UK., Sivaprakasam M; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Turner D; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Griffin RJ; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Golding BT; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060., Cano C; Cancer Research UK Newcastle Drug Discovery Unit , Chemistry, School of Natural and Environmental Sciences , Newcastle University , Newcastle upon Tyne , UK . Email: celine.cano@ncl.ac.uk ; Tel: +44 (0)191 208 7060.
Publikováno v:
RSC medicinal chemistry [RSC Med Chem] 2020 May 22; Vol. 11 (6), pp. 707-731. Date of Electronic Publication: 2020 May 22 (Print Publication: 2020).
Autor:
Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, USA., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, USA. Electronic address: philip.reigan@cuanschutz.edu.
Publikováno v:
Bioorganic & medicinal chemistry [Bioorg Med Chem] 2020 Mar 01; Vol. 28 (5), pp. 115303. Date of Electronic Publication: 2020 Jan 12.
Autor:
Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA.
Publikováno v:
Data in brief [Data Brief] 2020 Feb 28; Vol. 29, pp. 105347. Date of Electronic Publication: 2020 Feb 28 (Print Publication: 2020).
Autor:
Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA.
Publikováno v:
ChemMedChem [ChemMedChem] 2018 Aug 20; Vol. 13 (16), pp. 1681-1694. Date of Electronic Publication: 2018 Jul 11.