Zobrazeno 1 - 10
of 324
pro vyhledávání: '"Matheson, CJ"'
Autor:
Matheson, CJ, Coxon, CR, Bayliss, R, Boxall, K, Carbain, B, Fry, AM, Hardcastle, IR, Harnor, SJ, Mas-Droux, C, Newell, DR, Richards, MW, Sivaprakasam, M, Turner, D, Griffin, RJ, Golding, BT, Cano, C
Renewed interest in covalent inhibitors of enzymes implicated in disease states has afforded several agents targeted at protein kinases of relevance to cancers. We now report the design, synthesis and biological evaluation of 6-ethynylpurines that ac
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=core_ac_uk__::50079741394e01f4bd1b1137f16bfc2a
https://eprints.whiterose.ac.uk/160431/19/d0md00074d.pdf
https://eprints.whiterose.ac.uk/160431/19/d0md00074d.pdf
Autor:
Coxon, CR, Wong, C, Bayliss, RWA, Boxall, K, Carr, KH, Fry, AM, Hardcastle, IR, Matheson, CJ, Newell, DR, Sivaprakasam, M, Thomas, H, Turner, D, Yeoh, S, Wang, LZ, Griffin, RJ, Golding, BT, Cano, C
Publikováno v:
Oncotarget
Nek2 (NIMA-related kinase 2) is a cell cycle-dependent serine/threonine protein kinase that regulates centrosome separation at the onset of mitosis. Overexpression of Nek2 is common in human cancers and\ud suppression can restrict tumor cell growth a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::2a81c9e348a99e3a06a93c16991f5ec9
Autor:
Warfield BM; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO 80045, United States.
Publikováno v:
Data in brief [Data Brief] 2021 Sep 25; Vol. 38, pp. 107433. Date of Electronic Publication: 2021 Sep 25 (Print Publication: 2021).
Autor:
Warfield BM; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., McArthur DG; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, Colorado 80045, United States.
Publikováno v:
ACS chemical neuroscience [ACS Chem Neurosci] 2021 Sep 15; Vol. 12 (18), pp. 3477-3486. Date of Electronic Publication: 2021 Sep 02.
N-Substituted pyrrolopyrimidines and purines as p90 ribosomal S6 protein kinase-2 (RSK2) inhibitors.
Autor:
Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Warfield BM; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA. Electronic address: philip.reigan@cuanschutz.edu.
Publikováno v:
Bioorganic & medicinal chemistry [Bioorg Med Chem] 2021 Jul 01; Vol. 41, pp. 116220. Date of Electronic Publication: 2021 May 19.
Wee1 inhibitor PD0166285 sensitized TP53 mutant lung squamous cell carcinoma to cisplatin via STAT1.
Autor:
Li, Qi1,2 (AUTHOR), Yang, Wenjie3 (AUTHOR), Zhang, Qingyi4 (AUTHOR), Zhang, Daoming5 (AUTHOR), Deng, Jun6 (AUTHOR), Chen, Binxin1,2 (AUTHOR), Li, Ping2 (AUTHOR), Zhang, Huanqi5 (AUTHOR), Jiang, Yiming5 (AUTHOR), Li, Yangling2,5 (AUTHOR), Zhang, Bo7,8 (AUTHOR) zhangbo1009@zju.edu.cn, Lin, Nengming1,2 (AUTHOR) lnm1013@zju.edu.cn
Publikováno v:
Cancer Cell International. 9/13/2024, Vol. 24 Issue 1, p1-17. 17p.
Autor:
Chen, Rong1 (AUTHOR), Liu, Hengfang2 (AUTHOR), Meng, Weikang2 (AUTHOR), Sun, Jingyu2 (AUTHOR) bengbenghenhao@163.com
Publikováno v:
Scientific Reports. 9/9/2024, Vol. 14 Issue 1, p1-18. 18p.
Autor:
Su, Xin1,2 (AUTHOR), Li, Jian1,2 (AUTHOR), Xu, Xiao1,2 (AUTHOR), Ye, Youbao1,2 (AUTHOR), Wang, Cailiu1,2 (AUTHOR), Pang, Guanglong1,2 (AUTHOR), Liu, Wenxiu1,2 (AUTHOR), Liu, Ang1,2 (AUTHOR), Zhao, Changchun1,2 (AUTHOR), Hao, Xiangyong2 (AUTHOR) Haoxy-2008@163.com
Publikováno v:
Journal of Translational Medicine. 8/9/2024, Vol. 22 Issue 1, p1-43. 43p.
Autor:
Gruszka, Renata1 (AUTHOR) renata.gruszka@biol.uni.lodz.pl, Zakrzewski, Jakub2 (AUTHOR), Nowosławska, Emilia3 (AUTHOR), Grajkowska, Wiesława4 (AUTHOR), Zakrzewska, Magdalena5 (AUTHOR)
Publikováno v:
Scientific Reports. 8/2/2024, Vol. 14 Issue 1, p1-10. 10p.
Autor:
Matheson CJ; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Casalvieri KA; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Backos DS; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA., Minhajuddin M; Division of Hematology, University of Colorado Anschutz Medical Campus, 12700 E 19th Avenue, Aurora, CO, 80045, USA., Jordan CT; Division of Hematology, University of Colorado Anschutz Medical Campus, 12700 E 19th Avenue, Aurora, CO, 80045, USA., Reigan P; Department of Pharmaceutical Sciences, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of Colorado Anschutz Medical Campus, 12850 East Montview Boulevard, Aurora, CO, 80045, USA. Electronic address: philip.reigan@cuanschutz.edu.
Publikováno v:
European journal of medicinal chemistry [Eur J Med Chem] 2020 Jul 01; Vol. 197, pp. 112316. Date of Electronic Publication: 2020 Apr 16.