Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Masakatsu Sugahara"'
Autor:
Takashi, Goi, Tatsuo, Nakajima, Yoshiyuki, Komatsu, Atsushi, Kawata, Shuhei, Yamakoshi, Okimasa, Okada, Masakatsu, Sugahara, Asami, Umeda, Yoko, Takada, Jun, Murakami, Rikiya, Ohashi, Tomoko, Watanabe, Koichi, Fukase
Publikováno v:
ACS Med Chem Lett
[Image: see text] Inhibition of hypoxia-inducible factor prolyl hydroxylase domain (HIF-PHD) promotes erythropoietin (EPO) production by stabilizing the HIFα subunit. Thieno[2,3-d]pyrimidine 8 identified based on X-ray crystal structure analysis was
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::933a2a8fe3fc1119a71ecc9b4ca917e6
https://pubmed.ncbi.nlm.nih.gov/32676148
https://pubmed.ncbi.nlm.nih.gov/32676148
Autor:
Takashi Goi, Tatsuo Nakajima, Yoshiyuki Komatsu, Atsushi Kawata, Shuhei Yamakoshi, Okimasa Okada, Masakatsu Sugahara, Asami Umeda, Yoko Takada, Jun Murakami, Rikiya Ohashi, Tomoko Watanabe, Koichi Fukase
Publikováno v:
ACS Medicinal Chemistry Letters; 7/9/2020, Vol. 11 Issue 7, p1416-1420, 5p
Publikováno v:
Journal of the Chemical Society, Perkin Transactions 1. :768-773
A synthetic study of a 1-arylnaphthalene lignan having a heteroaryl group, such as the pyridyl group, at the C(1) position was conducted in detail. The Diels–Alder reaction of 1-pyridylisobenzofuran precursor 1 with dimethyl maleate or dimethyl fum
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::deeb28ed54b133f770873ad851c38b41
https://doi.org/10.1039/b110265f
https://doi.org/10.1039/b110265f
Autor:
Tsuyoshi Ogiku, Yasunori Moritani, Tameo Iwasaki, Masakatsu Sugahara, Yoshihiro Terakawa, Tatsuzo Ukita
Publikováno v:
ChemInform. 29
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::81874ab5e063422031799a79d87cff47
https://doi.org/10.1002/chin.199821093
https://doi.org/10.1002/chin.199821093
Publikováno v:
ChemInform. 33
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f591cdd5bfe8283ed60608b14eb3df13
https://doi.org/10.1002/chin.200232037
https://doi.org/10.1002/chin.200232037
Autor:
Tooru Kuroda, Kazuhiko Kondo, Tatsuzo Ukita, Masakatsu Sugahara, Hideshi Shimadzu, Yasunori Moritani
Publikováno v:
Chemical and Pharmaceutical Bulletin. 48:589-591
6,7-Diethoxy-1-[1-(2-methoxyethyl)-2-oxo-1,2-dihydropyridin- 4-yl]naphthalene-2,3-dimethanol [T-440, (1)] is a potential anti-asthmatic agent based on selective phosphodiesterase 4 inhibition. It was necessary for the further evaluation of 1 to devel
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::47b9d23e36b8e8c50f591b10cb8f0fb3
https://doi.org/10.1248/cpb.48.589
https://doi.org/10.1248/cpb.48.589
Autor:
Hideo Kikkawa, Tooru Kuroda, Yoshihiro Terakawa, Kazuaki Naito, Katsuo Ikezawa, Tatsuzo Ukita, Kazuteru Wada, Aya Nakata, Masakatsu Sugahara
Publikováno v:
ChemInform. 34
A novel series of 1-pyridylisoquinoline and 1-pyridyldihydroisoquinoline derivatives has been prepared. These compounds showed potent PDE4 inhibitory activities and a broad margin between the K(i) value of the rolipram binding affinity and the IC(50)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5d3d0ce6dc473c62438d03228116ee2e
https://doi.org/10.1002/chin.200341147
https://doi.org/10.1002/chin.200341147
Autor:
Tooru Kuroda, Tatsuzo Ukita, Masakatsu Sugahara, Yasunori Moritani, Kazuhiko Kondo, Hideshi Shimadzu
Publikováno v:
ChemInform. 31
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::94b218d18f72b01cd3bcc5ee8c431d69
https://doi.org/10.1002/chin.200038147
https://doi.org/10.1002/chin.200038147