Zobrazeno 1 - 10
of 12
pro vyhledávání: '"Marilenia De Matteo"'
Autor:
Isabelle Bonomo, Giulia Assoni, Valeria La Pietra, Giulia Canarutto, Elisa Facen, Greta Donati, Chiara Zucal, Silvia Genovese, Mariachiara Micaelli, Anna Pérez-Ràfols, Sergio Robbiati, Dimitris L. Kontoyannis, Marilenia De Matteo, Marco Fragai, Pierfausto Seneci, Luciana Marinelli, Daniela Arosio, Silvano Piazza, Alessandro Provenzani
Publikováno v:
Disease Models & Mechanisms, Vol 16, Iss 3 (2023)
Externí odkaz:
https://doaj.org/article/f46f5530b8b347c99a98e099c85d727f
Publikováno v:
Results in Chemistry, Vol 4, Iss , Pp 100654- (2022)
An efficient synthetic route was set up to prepare in good scale M-108, a novel bicycle derivative recently identified as a potent and selective G9a inhibitor, potentially useful as anti-fibroadipogenic agent. In particular, a facile three-steps sequ
Externí odkaz:
https://doaj.org/article/541b77a011324d9aa43adcccd223c3a1
Autor:
Alessia Petrocchi, Alessandro Grillo, Luca Ferrante, Pietro Randazzo, Adolfo Prandi, Marilenia De Matteo, Costanza Iaccarino, Monica Bisbocci, Antonella Cellucci, Cristina Alli, Martina Nibbio, Vincenzo Pucci, Jérôme Amaudrut, Christian Montalbetti, Carlo Toniatti, Romano Di Fabio
Publikováno v:
ACS Medicinal Chemistry Letters. 14:645-651
Autor:
Isabelle Bonomo, Giulia Assoni, Valeria La Pietra, Giulia Canarutto, Elisa Facen, Greta Donati, Chiara Zucal, Silvia Genovese, Mariachiara Micaelli, Anna Pérez-Ràfols, Sergio Robbiati, Dimitris L. Kontoyannis, Marilenia De Matteo, Marco Fragai, Pierfausto Seneci, Luciana Marinelli, Daniela Arosio, Silvano Piazza, Alessandro Provenzani
Lipopolysaccharide exposure to macrophages induces an inflammatory response that is heavily regulated at the transcriptional and post-transcriptional levels. HuR (ELAVL1) is an RNA binding protein that binds and regulates the maturation and half-life
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::41301d83518b6abcd82afc44a44b97b0
https://doi.org/10.1101/2023.01.16.524289
https://doi.org/10.1101/2023.01.16.524289
Autor:
Leda Ivanova Bencheva, Lorena Donnici, Luca Ferrante, Adolfo Prandi, Roberta Sinisi, Marilenia De Matteo, Pietro Randazzo, Matteo Conti, Pietro Di Lucia, Elisa Bono, Leonardo Giustini, Maria Vittoria Orsale, Alexandros Patsilinakos, Edith Monteagudo, Matteo Iannacone, Vincenzo Summa, Luca G. Guidotti, Raffaele De Francesco, Romano Di Fabio
Publikováno v:
Bioorganicmedicinal chemistry letters. 73
Chronic hepatitis B (CHB) is a major worldwide public health problem and novel anti-HBV therapies preventing liver disease progression to cirrhosis and hepatocellular carcinoma are urgently needed. Over the last several years, capsid assembly modulat
Autor:
Pietro Randazzo, Roberta Sinisi, Davide Gornati, Stefania Bertuolo, Leda Bencheva, Marilenia De Matteo, Martina Nibbio, Edith Monteagudo, Lorenzo Turcano, Valeria Bianconi, Giovanna Peruzzi, Vincenzo Summa, Alberto Bresciani, Chiara Mozzetta, Romano Di Fabio
Publikováno v:
Bioorganicmedicinal chemistry letters. 72
A new series of in vitro potent and highly selective histone methyl transferase enzyme G9a inhibitors was obtained. In particular, compound 2a, one the most potent G9a inhibitor identified, was endowed with >130-fold selectivity over GLP and excellen
Autor:
Adolfo Prandi, Luca Ferrante, Maria Veneziano, Mariana Gallo, Marco Ferrara, Leda Ivanova Bencheva, Antonella Cellucci, Nausicaa Mazzocchi, Pierfausto Seneci, Silvano Ronzoni, Andrea Menegon, Roberta Sinisi, Pietro Randazzo, Vincenzo Summa, Marilenia De Matteo, Romano Di Fabio
[Image: see text] Acid-sensing ion channels (ASICs) are a family of ion channels permeable to cations and largely responsible for the onset of acid-evoked ion currents both in neurons and in different types of cancer cells, thus representing a potent
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8c8a3bad6284485d88304e25bccd2e07
http://hdl.handle.net/11588/828238
http://hdl.handle.net/11588/828238
Autor:
Andrea Caprini, Daniele Lecis, Ilaria Motto, Amira Khaled, Cristina Battaglia, Martino Bolognesi, Francesca Vasile, Aldo Bianchi, Federica Cossu, Federica Servida, Moira Marizzoni, Elena de Franco, Pierfausto Seneci, Vincenzo Rizzo, Carmelo Drago, Leonardo Manzoni, Donatella Potenza, Marilenia De Matteo, Elisa Turlizzi, Mario Milani, Domenico Delia, Elisabetta Moroni, Eloise Mastrangelo, Maurizio Varrone, Laura Belvisi, Carlo Scolastico
Publikováno v:
Bioorganic & Medicinal Chemistry. 17:5834-5856
Novel proapoptotic Smac mimics/IAPs inhibitors have been designed, synthesized and characterized. Computational models and structural studies (crystallography, NMR) have elucidated the SAR of this class of inhibitors, and have permitted further optim
Autor:
Lucia Battistini, Daniela Arosio, Michelandrea De Cesare, Paola Carta, Carlo Scolastico, Giovanni Casiraghi, Michael Pilkington-Miksa, Laura Belvisi, Franco Zunino, Eugenio Scanziani, Leonardo Manzoni, Gloria Rassu, Marilenia De Matteo, Paola Perego, Vittoria Castiglioni, Paola Burreddu, Franca Zanardi, Nives Carenini, Francesca Vasile
Publikováno v:
Bioconjugate chemistry 23 (2012): 1610–1622. doi:10.1021/bc300164t
info:cnr-pdr/source/autori:Michael Pilkington-Miksa; Daniela Arosio; Lucia Battistini; Laura Belvisi; Marilenia De Matteo; Francesca Vasile; Paola Burreddu; Paola Carta; Gloria Rassu; Paola Perego; Nives Carenini; Franco Zunino; Michelandrea De Cesare; Vittoria Castiglioni; Eugenio Scanziani; Carlo Scolastico; Giovanni Casiraghi; Franca Zanardi; and Leonardo Manzoni/titolo:Design, Synthesis, and Biological Evaluation of Novel cRGD-Paclitaxel Conjugates for Integrin-Assisted Drug Delivery/doi:10.1021%2Fbc300164t/rivista:Bioconjugate chemistry/anno:2012/pagina_da:1610/pagina_a:1622/intervallo_pagine:1610–1622/volume:23
info:cnr-pdr/source/autori:Michael Pilkington-Miksa; Daniela Arosio; Lucia Battistini; Laura Belvisi; Marilenia De Matteo; Francesca Vasile; Paola Burreddu; Paola Carta; Gloria Rassu; Paola Perego; Nives Carenini; Franco Zunino; Michelandrea De Cesare; Vittoria Castiglioni; Eugenio Scanziani; Carlo Scolastico; Giovanni Casiraghi; Franca Zanardi; and Leonardo Manzoni/titolo:Design, Synthesis, and Biological Evaluation of Novel cRGD-Paclitaxel Conjugates for Integrin-Assisted Drug Delivery/doi:10.1021%2Fbc300164t/rivista:Bioconjugate chemistry/anno:2012/pagina_da:1610/pagina_a:1622/intervallo_pagine:1610–1622/volume:23
The efficacy of taxane-based antitumor therapy is limited by several drawbacks which result in a poor therapeutic index. Thus, the development of approaches that favor selective delivery of taxane drugs (e.g., paclitaxel, PTX) to the disease area rep
Autor:
Pierfausto Seneci, Francesca Vasile, Laura Belvisi, Vincenzo Rizzo, Carmelo Drago, Federica Servida, Leonardo Manzoni, Luca Ferrante, C. Scolastico, Aldo Bianchi, Gabriele Timpano, Donatella Potenza, Annalisa Conti, Eloise Mastrangelo, Marilenia De Matteo, Paola Perego
Publikováno v:
Bioorganic & medicinal chemistry
(2012): 6687–6708. doi:10.1016/j.bmc.2012.09.020
info:cnr-pdr/source/autori:Leonardo Manzoni; Laura Belvisi; Aldo Bianchi; Annalisa Conti; Carmelo Drago; Marilenia de Matteo; Luca Ferrante; Eloise Mastrangelo; Paola Perego; Donatella Potenza; Carlo Scolastico; Federica Servida; Gabriele Timpano; Francesca Vasile; Vincenzo Rizzo; Pierfausto Seneci/titolo:Homo-and heterodimeric Smac mimetics%2FIAP inhibitors as in vivo-active pro-apoptotic agents. Part I: Synthesis/doi:10.1016%2Fj.bmc.2012.09.020/rivista:Bioorganic & medicinal chemistry (Print)/anno:2012/pagina_da:6687/pagina_a:6708/intervallo_pagine:6687–6708/volume
(2012): 6687–6708. doi:10.1016/j.bmc.2012.09.020
info:cnr-pdr/source/autori:Leonardo Manzoni; Laura Belvisi; Aldo Bianchi; Annalisa Conti; Carmelo Drago; Marilenia de Matteo; Luca Ferrante; Eloise Mastrangelo; Paola Perego; Donatella Potenza; Carlo Scolastico; Federica Servida; Gabriele Timpano; Francesca Vasile; Vincenzo Rizzo; Pierfausto Seneci/titolo:Homo-and heterodimeric Smac mimetics%2FIAP inhibitors as in vivo-active pro-apoptotic agents. Part I: Synthesis/doi:10.1016%2Fj.bmc.2012.09.020/rivista:Bioorganic & medicinal chemistry (Print)/anno:2012/pagina_da:6687/pagina_a:6708/intervallo_pagine:6687–6708/volume
Novel pro-apoptotic, homo- and heterodimeric Smac mimetics/IAPs inhibitors based on the N-AVPI-like 4-substituted 1-aza-2-oxobicyclo[5.3.0]decane scaffold were prepared from monomeric structures connected through a head-head (8), tail-tail (9) or hea