Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Marie-Agnes Lassoie"'
Autor:
Laurent Knerr, Marie-Agnes Lassoie, Valérie Verbois, Fabienne Broeders, Gérald Guillaumet, Laurent Provins, Abdoulaye Gassama, Stéphanie Norsikian, Françoise de Laveleye-Defais, Philippe Collart, Laurent Defrère, Laszlo Kiss, Luc Quere, Jean-Marie Nicolas, Jean-Claude Hayez, Thierry Demaude, Sylvain Routier
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 17:142-146
A new series of 2,6-quinolinyl derivatives was prepared leading to potent low nanomolar VLA-4/VCAM-1 antagonists.
Autor:
Bernard Christophe, T. Taverne, Patrick Pasau, Jean-Pierre Hénichart, Christophe Genicot, Florence Moureau, Luc Quere, Laurence Goossens, B. J. Van Keulen, Michel Gillard, Marie-Agnes Lassoie, Philippe Collart, Thomas Ryckmans, F. Stiernet, Jean-Marie Nicolas, Michel Neuwels
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 13:437-442
Benzyloxyphenethylpiperazines are a new class of high affinity NK1 receptor antagonists. Oral bioavailability and selectivity can be fine tuned by the nature of the substituents on the basic nitrogen atom. Addition of substituents with a carboxylic a
Autor:
Jean‐Pierre Henichart, Nathalie Mestdagh, Raymond Houssin, Corinne Audouin, Marie-Agnes Lassoie
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 11:845-848
N-Aminoindoline derivatives were prepared and their 5-lipoxygenase inhibitory activities were evaluated in vitro and compared with those of phenidone and NDGA. Compound 4 presents the most effective 5-LO inhibition.
Autor:
Florence Moureau, Jean-Pierre Hénichart, Michel Neuwels, Raymond Houssin, Marie-Agnes Lassoie, Didier Berckmans, Edmond Differding, Solo Goldstein
Publikováno v:
Letters in Peptide Science. 2:125-134
Nine potent and selective substance P receptor antagonists (NK1 -) were analyzed with respect to their conformational space, with the aim to suggest probable conformations adopted at the receptor site and superposition rules for each structure (pharm
Autor:
Corinne Audouin, Jean‐Pierre Henichart, Marie-Agnes Lassoie, Nathalie Mestdagh, Raymond Houssin
Publikováno v:
ChemInform. 32
N-Aminoindoline derivatives were prepared and their 5-lipoxygenase inhibitory activities were evaluated in vitro and compared with those of phenidone and NDGA. Compound 4 presents the most effective 5-LO inhibition.