Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Maria Carmela Fulco"'
Autor:
Giulio Dondio, Saverio Minucci, Roberto Boggio, Giacomo Carenzi, Agnese Abate, Mario Varasi, Marco Giulio Rozio, Ciro Mercurio, Roberto Dal Zuffo, Chiara Bigogno, Maria Carmela Fulco, Florian Thaler, Tiziana Cataudella, Antonello Mai
Publikováno v:
Journal of Medicinal Chemistry. 54:3051-3064
New spiro[chromane-2,4'-piperidine] and spiro[benzofuran-2,4'-piperidine] hydroxamic acid derivatives as HDAC inhibitors have been identified by combining privileged structures with a hydroxamic acid moiety as zinc binding group. The compounds were e
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4f41905394ac094b5e80673f4d267b9
https://doi.org/10.1021/jm200146u
https://doi.org/10.1021/jm200146u
Publikováno v:
Tetrahedron. 65:7092-7098
The metal-catalyzed reactions of neopentyl α-diazomethanesulfonate (DAMS) and diisopropyl α-diazomethanephosphonate (DIDAMP) with furan, 2-methylfuran and 2-methoxyfuran are reported. The products consist mostly of ω-acyl-substituted sulfono- or p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5117d5474515f39c72badc3b5de97b5f
https://doi.org/10.1016/j.tet.2009.06.040
https://doi.org/10.1016/j.tet.2009.06.040
Autor:
Raffaella Amici, Ciro Mercurio, Andrea Colombo, Maria Carmela Fulco, Luca Sartori, Florian Thaler, Giulio Dondio, Saverio Minucci, Stefania Gagliardi, Roberto Boggio, Loris Moretti, Giacomo Carenzi, Agnese Abate, Mario Varasi
Publikováno v:
European journal of medicinal chemistry. 108
In the last decades, inhibitors of histone deacetylases (HDAC) have become an important class of anti-cancer agents. In a previous study we described the synthesis of spiro[chromane-2,4'-piperidine]hydroxamic acid derivatives able to inhibit histone
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b08d2569a3404a6df65d91fa433e2125
https://pubmed.ncbi.nlm.nih.gov/26629860
https://pubmed.ncbi.nlm.nih.gov/26629860
Autor:
Antimo Gioiello, Francesco Venturoni, Simon Zlotsky, Asiya Khamidullina, Roberto Pellicciari, Maria Carmela Fulco
Publikováno v:
ChemInform. 41
A facile one-pot procedure for the synthesis of pyrazole-5-carboxylates by 1,3-dipolar cycloaddition of ethyl diazoacetate is described. Cycloadditions with α-methylene carbonyl compounds utilizing 1,8-diazabicyclo[5.4.0]undec-7-ene as base and acet
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e77f5aea9287c26a119c017f7b72f564
https://doi.org/10.1002/chin.201006112
https://doi.org/10.1002/chin.201006112
Publikováno v:
ChemInform. 40
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9aed00ccb27f74aa9d6f44c18f541a42
https://doi.org/10.1002/chin.200952049
https://doi.org/10.1002/chin.200952049
Autor:
Roberto Pellicciari, Burcu Çaliskan Ergün, Maria Carmela Fulco, Maura Marinozzi, Roccaldo Sardella, Benedetto Natalini
The first series of conformationally constrained analogues of homotaurine is reported. The partial constriction of the skeleton Was realized through the insertion of a cyclopropyl ring, between the alpha,beta- and beta,gamma-positions, thus affording
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::47d859c0ee81da7c0add2d14b171a54f
https://avesis.gazi.edu.tr/publication/details/ceed9357-ac05-491b-9ebe-92c47c9e1931/oai
https://avesis.gazi.edu.tr/publication/details/ceed9357-ac05-491b-9ebe-92c47c9e1931/oai
Autor:
Asiya Khamidullina, Roberto Pellicciari, Maria Carmela Fulco, Antimo Gioiello, Francesco Venturoni, Simon Zlotsky
A facile one-pot procedure for the synthesis of pyrazole-5-carboxylates by 1,3-dipolar cycloaddition of ethyl diazoacetate is described. Cycloadditions with α-methylene carbonyl compounds utilizing 1,8-diazabicyclo[5.4.0]undec-7-ene as base and acet
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b98e40ec8e310d49dc314ff466c38dc0
http://hdl.handle.net/11391/108656
http://hdl.handle.net/11391/108656
Autor:
Maria Carmela Fulco, Antonio Macchiarulo, Christian Thomsen, Julia Gafarova, Søren Møller Nielsen, Maura Marinozzi, Gianluca Giorgi, Roberto Pellicciari, Michaela Serpi
Bioisosteric replacements of the distal acidic group of L-glutamic acid (L-Glu, 1) and conformational constraining of its carbon skeleton, have been widely exploited to discover competitive modulators of glutamate receptors. Noteworthy, L-homocysteic
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ff5b2cfa779392d7a8d22bc044cb6609
http://hdl.handle.net/11391/31758
http://hdl.handle.net/11391/31758
Autor:
Antonio Macchiarulo, Roberto Pellicciari, Clemens Novak, Mette Brunsgaard Hermit, Rosanna Filosa, Thomas N. Sager, Tine B. Stensbøl, Benedetto Natalini, Søren Møller Nielsen, Maria Carmela Fulco, Maura Marinozzi, Christian Thomsen
The first series of 2'-substituted 2-(3'-carboxybicyclo-[1.1.1]pentyl)glycine derivatives, (2R)- and (2S)-(2',2'-dichloro-3'-carboxybicycto[1.1.1]pentyl)glycine (10) and (11), and 2-(2'-chloro-3'-carboxybicyclo[1.1.1]pentyl)glycine (12) were synthesi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d6bddff862213e1f46ff91e6d1df174
http://hdl.handle.net/11591/335042
http://hdl.handle.net/11591/335042