Zobrazeno 1 - 10
of 43
pro vyhledávání: '"Maria A, Siracusa"'
Autor:
Loredana Salerno, Maria N. Modica, Valeria Pittalà, Giuseppe Romeo, Maria A. Siracusa, Claudia Di Giacomo, Valeria Sorrenti, Rosaria Acquaviva
Publikováno v:
The Scientific World Journal, Vol 2014 (2014)
Eggplant fruit is a very rich source of polyphenol compounds endowed with antioxidant properties. The aim of this study was to extract polyphenols from eggplant entire fruit, pulp, or skin, both fresh and dry, and compare results between conventional
Externí odkaz:
https://doaj.org/article/22f1d2c827374ac9bcd7c86796e86743
Autor:
Mario Salmona, Maria Angela Siracusa, Giuseppe Romeo, Maria N. Modica, Loredana Salerno, Alfredo Cagnotto, Sebastiano Intagliata, Valeria Pittalà
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 26:4052-4056
In this work we report the discovery of new homo and hetero bis-piperazinyl-1-propanone derivatives as selective ligands for 5-HT7 over 5-HT1A receptor. These newly synthesized compounds possess a 4-arylpiperazine linked through an acyl spacer to ano
Autor:
Giuseppe Amico, Livia Basile, Loredana Salerno, Salvatore Guccione, Valeria Pittalà, Maria N. Modica, Maria Angela Siracusa, Agostino Marrazzo, Giuseppe Romeo
Publikováno v:
Journal of Advances in Medical and Pharmaceutical Sciences. 5:1-10
Autor:
Mario Salmona, Valeria Pittalà, Sebastiano Intagliata, Alfredo Cagnotto, Maria Angela Siracusa, Loredana Salerno, Giuseppe Romeo, Maria N. Modica
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 25:1427-1430
New long-chain 4-substituted piperazines linked to a thienopyrimidine or a quinazoline system were synthesized and tested for their binding properties on human cloned 5-HT1A and 5-HT7 serotonin receptors. Some structural modifications, concerning tre
Autor:
Maria Angela Siracusa, Loredana Salerno, Claudia Di Giacomo, Valeria Sorrenti, Valeria Pittalà, Giuseppe Romeo, Maria N. Modica, Rosaria Acquaviva
Publikováno v:
The Scientific World Journal, Vol 2014 (2014)
The Scientific World Journal
The Scientific World Journal
Eggplant fruit is a very rich source of polyphenol compounds endowed with antioxidant properties. The aim of this study was to extract polyphenols from eggplant entire fruit, pulp, or skin, both fresh and dry, and compare results between conventional
Autor:
Maria N. Modica, Mario Salmona, Sebastiano Intagliata, Valeria Pittalà, Alfredo Cagnotto, Maria Angela Siracusa, Loredana Salerno, Rafał Kurczab, Giuseppe Romeo
Based on our earlier studies of structure activity relationships on 4-substituted piperazine derivatives, in this work we synthesized a novel set of long-chain arylpiperazines with the purpose of elucidating if some structural modifications in the te
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1bcf83e202d65212582e50c8beb4eabd
http://hdl.handle.net/20.500.11769/18852
http://hdl.handle.net/20.500.11769/18852
Autor:
Sebastiano, Intagliata, Maria N, Modica, Valeria, Pittalà, Loredana, Salerno, Maria A, Siracusa, Alfredo, Cagnotto, Mario, Salmona, Rafał, Kurczab, Giuseppe, Romeo
Publikováno v:
Bioorganicmedicinal chemistry. 25(3)
Based on our earlier studies of structure activity relationships on 4-substituted piperazine derivatives, in this work we synthesized a novel set of long-chain arylpiperazines with the purpose of elucidating if some structural modifications in the te
Autor:
Valeria Pittalà, Loredana Salerno, Alfredo Cagnotto, Tiziana Mennini, Giulio Vistoli, Giuseppe Romeo, Maria Angela Siracusa, Maria N. Modica, Alessandro Pedretti
Publikováno v:
Bioorganic & Medicinal Chemistry. 19:5260-5276
Three different series of 1H-pyrrolopyrimidine-2,4-dione derivatives were designed and synthesized as ligands for the α(1)-adrenergic receptors (α(1)-ARs). A microwave-assisted protocol was developed in order to improve purity and yields of some fi
Autor:
Kenneth P. Minneman, Maria Angela Siracusa, Maurizio Botta, Loredana Salerno, Luisa Materia, Valeria Pittalà, Fabrizio Manetti, Giuseppe Romeo, Maria N. Modica
Publikováno v:
European Journal of Medicinal Chemistry. 46:2676-2690
A number of new 4-phenylpiperidine-2,6-diones bearing at the 1-position an ω-[4-(substituted phenyl)piperazin-1-yl]alkyl moiety were designed and synthesized as ligands for the α1-adrenergic receptor (α1-AR) subtypes. Some synthesized compounds, t
Autor:
Kenneth P. Minneman, Giuseppe Romeo, Gabriella Marucci, Valeria Pittalà, Maria Angela Siracusa, Maria N. Modica, Piero Angeli, Luisa Materia, Loredana Salerno, Michela Buccioni
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 16:6200-6203
A number of new pyrimido[5,4-b]indole and [1]benzothieno[3,2-d]pyrimidine derivatives were synthesized and evaluated for their binding and functional properties at alpha(1)-adrenergic receptor (alpha(1)-AR) subtypes. They behaved as potent alpha(1)-A