Zobrazeno 1 - 10 of 32 pro vyhledávání: '"Margolis BJ"'
1
Akademický článek
Positive allosteric modulators of the α7 nicotinic acetylcholine receptor: SAR investigation around PNU-120596.
Autor: Acker BA; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Badescu VO; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Berkenpas MB; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Groppi VE; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Hajós M; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Higdon NR; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Hurst RS; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Jon Jacobsen E; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Margolis BJ; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., McWhorter WW; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Myers JK; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Piotrowski DW; Pfizer Worldwide Research & Development, Groton, CT 06340, USA. Electronic address: david.w.piotrowski@comcast.net., Rogers BN; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Sarapa D; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Vetman TN; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Walker DP; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Wall TM; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Wilhite DM; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Wishka DG; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Xu W; Pfizer Worldwide Research & Development, Groton, CT 06340, USA., Yates KM; Pfizer Worldwide Research & Development, Groton, CT 06340, USA.
Publikováno v: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2023 Sep 01; Vol. 93, pp. 129433. Date of Electronic Publication: 2023 Aug 07.
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2
Akademický článek
Investigating the Behavior of Published PAINS Alerts Using a Pharmaceutical Company Data Set.
Autor: Vidler LR; Research and Development, Eli Lilly and Company, Ltd., Sunninghill Road, Windlesham, Surrey GU20 6PH, United Kingdom., Watson IA; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, Indiana 46285, United States., Margolis BJ; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, Indiana 46285, United States., Cummins DJ; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, Indiana 46285, United States., Brunavs M; Research and Development, Eli Lilly and Company, Ltd., Sunninghill Road, Windlesham, Surrey GU20 6PH, United Kingdom.
Publikováno v: ACS medicinal chemistry letters [ACS Med Chem Lett] 2018 Jul 10; Vol. 9 (8), pp. 792-796. Date of Electronic Publication: 2018 Jul 10 (Print Publication: 2018).
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3
Akademický článek
Discovery of N-(6-Fluoro-1-oxo-1,2-dihydroisoquinolin-7-yl)-5-[(3R)-3-hydroxypyrrolidin-1-yl]thiophene-2-sulfonamide (LSN 3213128), a Potent and Selective Nonclassical Antifolate Aminoimidazole-4-carboxamide Ribonucleotide Formyltransferase (AICARFT) Inhibitor Effective at Tumor Suppression in a Cancer Xenograft Model.
Autor: Fales KR; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Njoroge FG; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Brooks HB; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Thibodeaux S; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Torrado A; Centro de Investigación Lilly , S. A., Avda. de la Industria 30, 28108 Alcobendas, Madrid, Spain., Si C; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Toth JL; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Mc Cowan JR; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Roth KD; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Thrasher KJ; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Frimpong K; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Lee MR; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Dally RD; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Shepherd TA; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Durham TB; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Margolis BJ; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Wu Z; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Wang Y; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Atwell S; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Wang J; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Hui YH; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Meier TI; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Konicek SA; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States., Geeganage S; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285, United States.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2017 Dec 14; Vol. 60 (23), pp. 9599-9616. Date of Electronic Publication: 2017 Nov 09.
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4
Akademický článek
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5
Akademický článek
The Use of Nucleosome Substrates Improves Binding of SAM Analogs to SETD8.
Autor: Strelow JM; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA strelow_john_mark@lilly.com., Xiao M; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA., Cavitt RN; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA., Fite NC; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA., Margolis BJ; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA., Park KJ; Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA.
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 2016 Sep; Vol. 21 (8), pp. 786-94. Date of Electronic Publication: 2016 Jul 01.
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6
Akademický článek
Beyond PAINs: Chemotype Sensitivity of Protein Methyltransferases in Screens.
Autor: Gao C; Lilly Research Laboratories, Eli Lilly and Company , Lilly Corporate Center, Indianapolis, Indiana 46285, United States., Margolis BJ; Lilly Research Laboratories, Eli Lilly and Company , Lilly Corporate Center, Indianapolis, Indiana 46285, United States., Strelow JM; Lilly Research Laboratories, Eli Lilly and Company , Lilly Corporate Center, Indianapolis, Indiana 46285, United States., Vidler LR; Research and Development, Eli Lilly and Company Ltd. , Sunninghill Road, Windlesham, Surrey GU20 6PH, United Kingdom., Mader MM; Lilly Research Laboratories, Eli Lilly and Company , Lilly Corporate Center, Indianapolis, Indiana 46285, United States.
Publikováno v: ACS medicinal chemistry letters [ACS Med Chem Lett] 2015 Nov 19; Vol. 7 (2), pp. 156-61. Date of Electronic Publication: 2015 Nov 19 (Print Publication: 2016).
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8
Akademický článek
Affinity purification of a chimeric nicotinic acetylcholine receptor in the agonist and antagonist bound states.
Autor: Liu S; Pfizer Inc., Pfizer Global Research and Development, Groton, CT 06340, United States. shenping.liu@pfizer.com, Babcock MS, Bode J, Chang JS, Fischer HD, Garlick RL, Gill GS, Lund ET, Margolis BJ, Mathews WR, Rogers BN, Wolfe M, Groppi V, Baldwin ET
Publikováno v: Protein expression and purification [Protein Expr Purif] 2011 Sep; Vol. 79 (1), pp. 102-10. Date of Electronic Publication: 2011 Jun 02.
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9
Akademický článek
Assembly of 4-aminoquinolines via palladium catalysis: a mild and convenient alternative to SNAr methodology.
Autor: Margolis BJ; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana 46285, USA. margolis_brandon_j@lilly.com, Long KA, Laird DL, Ruble JC, Pulley SR
Publikováno v: The Journal of organic chemistry [J Org Chem] 2007 Mar 16; Vol. 72 (6), pp. 2232-5. Date of Electronic Publication: 2007 Feb 13.
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10
Akademický článek
Discovery of non-covalent dipeptidyl peptidase IV inhibitors which induce a conformational change in the active site.
Autor: Sheehan SM; Lilly Research Laboratories, A Division of Eli Lilly and Company, Indianapolis, IN 46285, USA. SHEEHAN_SCOTT@LILLY.COM, Mest HJ, Watson BM, Klimkowski VJ, Timm DE, Cauvin A, Parsons SH, Shi Q, Canada EJ, Wiley MR, Ruehter G, Evers B, Petersen S, Blaszczak LC, Pulley SR, Margolis BJ, Wishart GN, Renson B, Hankotius D, Mohr M, Zechel JC, Michael Kalbfleisch J, Dingess-Hammond EA, Boelke A, Weichert AG
Publikováno v: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2007 Mar 15; Vol. 17 (6), pp. 1765-8. Date of Electronic Publication: 2006 Dec 24.
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