Zobrazeno 1 - 1
of 1
pro vyhledávání: '"Manuel Alunno"'
Autor:
Manuel Alunno, Francesco Antonio Greco, Emidio Camaioni, Andrea Carotti, Giorgio Saluti, Roccaldo Sardella, Paride Liscio, Antonio Macchiarulo, Andrea Mammoli, Martina Ferri
Publikováno v:
Bioorganic & Medicinal Chemistry. 28:115731
The medicinal chemist toolbox is plenty of (bio)isosteres when looking for a carboxylic acid replacement. However, systematic assessment of acid surrogates is often time consuming and expensive, while prediction of both physicochemical properties (lo