Zobrazeno 1 - 10
of 66
pro vyhledávání: '"Makoto Shimazaki"'
Autor:
Taisei Iwasa, Seiji Adachi, Yusuke Oyama, Yusuke Suzuki, Masatoshi Mabuchi, Hironori Nakamura, Makoto Shimazaki, Shinji Nishiwaki, Takuji Iwashita, Masahito Shimizu
Publikováno v:
Internal Medicine; 2024, Vol. 63 Issue 8, p1099-1103, 5p
Autor:
Taisei Iwasa, Seiji Adachi, Yusuke Suzuki, Eri Takada, Kana Matsuura, Masatoshi Mabuchi, Hironori Nakamura, Makoto Shimazaki, Shinji Nishiwaki, Takashi Ibuka, Takuji Iwashita, Masahito Shimizu
Publikováno v:
Internal Medicine; 2024, Vol. 63 Issue 13, p1879-1881, 3p
Autor:
Hironori Nakamura, Seiji Adachi, Yukari Uno, Masatoshi Mabuchi, Makoto Shimazaki, Shinji Nishiwaki, Masahito Shimizu
Publikováno v:
American Journal of Case Reports; 11/28/2023, Vol. 24, p1-10, 10p
Autor:
Masatoshi Mabuchi, Seiji Adachi, Yukari Uno, Hironori Nakamura, Makoto Shimazaki, Shinji Nishiwaki, Iwao Kumazawa, Takuji Iwashita, Masahito Shimizu
Publikováno v:
Internal Medicine; 2023, Vol. 62 Issue 16, p2355-2359, 5p
Autor:
Makoto Shimazaki, Yuka Shogase, Miyuki Tatsuta, Klaus Urbahns, Kayo Yasoshima, Noriyuki Yamamoto, Sachiko Sakakibara, Jang Bahadur Gupta, Takeshi Yura, Li Yingfu, Mikayo Kataoka
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 15:2265-2269
1-(1H-Benzimidazol-5-yl)-3-tert-butylurea derivatives have been identified as a novel class of non-peptide luteinizing hormone-releasing hormone (LHRH) antagonists. Herein, we disclose the synthesis and structure–activity relationships (SAR) of thi
Autor:
Kinji Fuchikami, Sachiko Sakakibara, Tsutomu Masuda, Takuya Shintani, Mitsuyuki Shimada, Karl Ziegelbauer, Yoshino Takashi, Kevin Bacon, Timothy B. Lowinger, Makoto Shimazaki, Toshiki Murata, Hiroshi Kadono
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 14:4013-4017
A series of 2-amino-3-cyano-4-alkyl-6-(2-hydroxyphenyl)pyridine derivatives was synthesized and evaluated as IkappaB kinase beta (IKK-beta) inhibitors. Substitution of an aminoalkyl group for the aromatic group at the 4-position on the core pyridine
Autor:
Yoshino Takashi, Keisuke Takeshita, Hiroshi Kadono, Sachiko Sakakibara, Kevin Bacon, Makoto Shimazaki, Mitsuyuki Shimada, Takuya Shintani, Katsuya Sakai, Toshiro Niki, Toshiki Murata, Tsutomu Masuda, Masaomi Umeda, Timothy B. Lowinger, Hisayo Inbe, Karl Ziegelbauer, Kinji Fuchikami
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 13:913-918
IkappaB kinase beta (IKK-beta) is a serine-threonine protein kinase critically involved in the activation of the transcription factor Nuclear Factor kappa B (NF-kappaB) in response to various inflammatory stimuli. We have identified a small molecule
Autor:
Miyuki Funabashi Yoh, Katsuhisa Toda, Makoto Shimazaki, Toshiyuki Nakamura, Yoichiro Ito, Eri Morita
Publikováno v:
Journal of Infection and Chemotherapy. 8:256-261
We report a case of a 71-year-old man with staphylococcal scalded-skin syndrome (SSSS). The patient, with a chronic history of diabetes mellitus, was admitted to our hospital with lumbago, and a diagnosis of renal-cell carcinoma with bone metastasis
Autor:
Masanobu Uchiyama, Yuki Shimogaichi, Makoto Shimazaki, Atsushi Ohta, Naoko Yokota, Nobuo Katoh, Rio Mimura
Publikováno v:
Tetrahedron: Asymmetry. 8:3467-3474
Asymmetric reduction of symmetrical diacetylaromatics ( 1a , 1b , and 1d-g ) with baker's yeast ( Saccharomyces cerevisiae ) provided the corresponding alcohols of high enantiomeric purity. By choosing appropriate reaction conditions, the products we
Autor:
Yoshinori Nishino, Hiroto Shima, Takashi Deguchi, Hisataka Moriwaki, Hiromi Mohri, Takaya Ohnishi, Yoichiro Ito, Makoto Shimazaki, Mori Yasuda, Toshiyuki Nakamura, Shigeru Fujihiro, Yasutoshi Muto, Tomomichi Matsushita
Publikováno v:
Journal of Gastroenterology. 32:236-240
An extremely rare case of esophageal metastasis from prostate cancer is reported. A 65-year-old man presented with anorexia and back pain. Upper gastrointestinal X-ray fluoroscopy and endoscopy revealed a shallow longitudinal ulcer, with converging m