Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Mahesh G. Jadhav"'
Autor:
Ravindra Dattatraya Gupte, Mahesh G. Jadhav, Prabhu Dutt Mishra, Asha Kulkarni-Almeida, Bindu Hegde, Shruta Dadarkar, Meet Shah, Girish B Mahajan, Nilesh M Dagia, Jacqueline Trivedi
Publikováno v:
International Immunopharmacology. 33:63-69
Rheumatoid arthritis (RA), an autoimmune-inflammatory disease is characterized by dysregulation of signal transduction pathways, increased production of pro-inflammatory cytokines, enhanced leukocyte infiltration into synovial microvascular endotheli
Autor:
Lyle C. Fonseca, Shruta Dadarkar, Asha Almeida, Firuza Kharas, Aurelio S. Lobo, Ashish Suthar, Mahesh G. Jadhav, Sapna Parikh, Roda Dalal, Jacqueline Trivedi, Ankita Srivastava
Publikováno v:
Pharmacology & Pharmacy. :106-116
Tumor necrosis factor (TNF-α) is a key regulator of the inflammatory and tissue destruc-tive pathways in rheumatoid arthritis (RA). The clinical success of anti-TNF-α and an-ti-IL-17 biologics has validated the concept that cytokine blockade is ben
Autor:
Sanjay Kumar, Lyle C. Fonseca, Nilesh M. Dagia, Mahesh G. Jadhav, Shruta S. Dadarkar, Asha Kulkarni-Almeida, Ravindra Dattatraya Gupte, Mandar R. Bhonde, Anshu Chetrapal-Kunwar, Divya V. Kamath, Gautam Agarwal, Firuza Kharas, Jacqueline Trivedi
Publikováno v:
American journal of physiology. Cell physiology. 298(4)
A promising therapeutic approach to diminish pathological inflammation is to inhibit the increased production and/or biological activity of proinflammatory cytokines (e.g., TNF-alpha, IL-6). The production of proinflammatory cytokines is controlled a
Autor:
Vijaykumar Deore, Shruta S. Dadarkar, Pooja Bhatt, Dimple Bhatia, Kumar V.S. Nemmani, Nilesh M. Dagia, Sanjay Kumar, Mandar R. Bhonde, Abhijit Roychowdhury, Ravindra Dattatraya Gupte, Nilambari Yewalkar, Somesh Sharma, Nikesh Desai, Mahesh G. Jadhav, Ram A. Vishwakarma, Aditi Amol Tannu
Publikováno v:
Bioorganicmedicinal chemistry letters. 19(11)
A series of novel cyanopyridyl based molecules ( 1 – 14 ) were designed, synthesized and probed for inhibition of mammalian target of rapamycin (mTOR) activity. Compound 14 was found to be a potent inhibitor of mTOR activity as assessed by enzyme-l
Autor:
Sanjay Kumar, Somesh Sharma, Nilesh M Dagia, Dimple Bhatia, Aditi Amol Tannu, Ram A. Vishwakarma, Mahesh G. Jadhav, Nilambari Yewalkar, Shruta Dadarkar, Vijaykumar Deore, Nikesh Desai, Pooja Bhatt, Ravindra Dattatraya Gupte, Mandar R. Bhonde
Publikováno v:
American journal of physiology. Gastrointestinal and liver physiology. 295(6)
Ulcerative colitis is an autoimmune-inflammatory disease characterized by increased proliferation of colonic epithelial cells, dysregulation of signal transduction pathways, elevated mucosal T cell activation, increased production of proinflammatory