Zobrazeno 1 - 10
of 31
pro vyhledávání: '"Maddamsetty V. Rao"'
Publikováno v:
Journal of Pharmacy & Pharmaceutical Sciences, Vol 11, Iss 2 (2008)
Development of new chemotherapeutic drugs is the need of the hour to improve tuberculosis control, particularly in the developing world. In the last fourty years no new compound has been brought to the market for the treatment of tuberculosis. Howeve
Externí odkaz:
https://doaj.org/article/a357df13116d46ccb3a3b51d99fc587e
Publikováno v:
Current Medicinal Chemistry-Anti-Cancer Agents. 2:215-254
Pyrrolo[2,1-c][1,4]benzodiazepines (PBDs) are naturally occurring compounds isolated from various Streptomyces species. The PBDs exert their biological activity through covalent binding and exhibit cytotoxicity. Extensive studies have been carried ou
Publikováno v:
The Journal of Organic Chemistry. 66:997-1001
A facile synthesis of bronchodilatory pyrrolo[2,1-b]quinazoline alkaloids by azidoreductive cyclization strategy employing TMSCl-NaI and bakers' yeast is described. Both the chemical and enzymatic methods are mild and take place at room temperature i
Publikováno v:
Tetrahedron: Asymmetry. 10:4261-4264
The ring opening of epoxides with nucleophiles such as TMSN 3 and isopropylamine takes place enantioselectively in the presence of β-cyclodextrin under extremely mild conditions and the azido alcohols and amino alcohols are formed as ( S )-isomers.
Publikováno v:
Chemistry of Heterocyclic Compounds. 34:1342-1358
Modern synthetic approaches to DNA binding pyrrolobenzodiazepine antibiotics have been discussed.
Publikováno v:
ChemInform. 22
o-Cyanophenyl allyl carbamate (3), 3-allyl-3,4-dihydro-4-imino-2H-1,3-benzoxazine-2-thione (8a), and -quinazoline-2(1H)-thiones (8b–d) have been cyclized to 2,3-dihydro-2-methyl-5H-imidazo[1,2-c][1,3]benzoxazin-5-one (5), the corresponding 5-thione
Publikováno v:
ChemInform. 23
Autor:
Maddamsetty V. Rao, Ahmed Kamal
Publikováno v:
ChemInform. 22
Porcine pancreatic lipase catalyzes the specific hydroxyl acylation of 2-propanol amines with enantioselectivity employing trichloroacetic anhydride in organic solvents.
Publikováno v:
ChemInform. 22
The enzymatic conversion of oximes by ultrasonically stimulated baker's yeast yields the corresponding aldehydes and ketones in high yields.
Publikováno v:
ChemInform. 24
The ring opening of epoxides with 2-propylamine in presence of lipase in organic solvents affords selectively (S)-propanol amines. The effect of solvents towards selectivity has also been examined.