Zobrazeno 1 - 10 of 18 pro vyhledávání: '"Małgorzata Dukat"'
1
Akademický článek
Binding and functional structure-activity similarities of 4-substituted 2,5-dimethoxyphenyl isopropylamine analogues at 5-HT2A and 5-HT2B serotonin receptors
Autor: Prithvi Hemanth, Pallavi Nistala, Vy T. Nguyen, Jose M. Eltit, Richard A. Glennon, Małgorzata Dukat
Publikováno v: Frontiers in Pharmacology, Vol 14 (2023)
Certain 4-substituted analogs of 1-(2,5-dimethoxyphenyl)isopropylamine (2,5-DMA) are psychoactive classical hallucinogens or serotonergic psychedelic agents that function as human 5-HT2A (h5-HT2A) serotonin receptor agonists. Activation of a related
Externí odkaz: https://doaj.org/article/f2f80a56888b4989a6bc29f6d4529f18
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4
X-Ray Crystal Structure of a 2-Amino-3,4-dihydroquinazoline 5-HT
Autor: Ahmed S, Abdelkhalek, Faik N, Musayev, Kavita A, Iyer, Prithvi, Hemanth, Martin K, Safo, Małgorzata, Dukat
Publikováno v: J Mol Struct
Certain 2-amino-3,4-dihydroquinazolines bind at 5-HT(3) serotonin receptors and act as antagonists (e.g. 6-chloro) whereas others bind with little to no affinity and lack functional activity (e.g. 8-chloro). The purpose of this investigation was to g
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::011c444f37ad436d72c39ed6264a4fd7
https://pubmed.ncbi.nlm.nih.gov/32616964
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6
Akademický článek
Merging cultures and disciplines to create a drug discovery ecosystem at Virginia commonwealth university: Medicinal chemistry, structural biology, molecular and behavioral pharmacology and computational chemistry
Autor: Glen E. Kellogg, Yana Cen, Malgorzata Dukat, Keith C. Ellis, Youzhong Guo, Jiong Li, Aaron E. May, Martin K. Safo, Shijun Zhang, Yan Zhang, Umesh R. Desai
Publikováno v: SLAS Discovery, Vol 28, Iss 6, Pp 255-269 (2023)
The Department of Medicinal Chemistry, together with the Institute for Structural Biology, Drug Discovery and Development, at Virginia Commonwealth University (VCU) has evolved, organically with quite a bit of bootstrapping, into a unique drug discov
Externí odkaz: https://doaj.org/article/96b02476711041fea6a676aac62c3785
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8
Synthetic Cathinones: A Brief Overview of Overviews with Applications to the Forensic Sciences
Autor: Richard A, Glennon, Małgorzata, Dukat
Publikováno v: Annals of forensic research and analysis. 4(2)
Catha edulis, the fresh leaves of which (i.e., khat) are used for their central stimulant actions, has been known for many hundreds of years. S(−)Cathinone was identified as a centrally-active khat constituents >30 years ago. Although khat use was
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::b21b34910a5a203c77e40f19317b4bd5
https://pubmed.ncbi.nlm.nih.gov/30288398
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