Zobrazeno 1 - 10 of 59 pro vyhledávání: '"Ma, Sills"'
1
The unusual binding properties of the endothelin receptor antagonist CGS 27830 distinguishes receptor/agonist interactions
Autor: Mh, Chin, Cl, Cioffi, Garay M, Rf, Neale, Ss, Shetty, DelGrande D, Mugrage B, Ma, Sills, Kenneth Lipson
Publikováno v: Europe PubMed Central
CGS 27830 [meso-1,4-dihydro-5-methoxycarbonyl-2,6-dimethyl-4-(3- nitrophenyl)-3-pyridine carboxylic acid anhydride] is a nonpeptidic, insurmountable, endothelin (ET) receptor antagonist with approximately 10- to 20-fold selectivity for ETA receptors.
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::7b8d52b5a4d0915627493c0568b1ad9e
http://europepmc.org/abstract/med/8558459
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2
Akademický článek
Probing the primary screening efficiency by multiple replicate testing: a quantitative analysis of hit confirmation and false screening results of a biochemical assay.
Autor: Zhang JH; Novartis Institute for Biomedical Research, Cambridge, MA 02139, USA. ji-hu.zhang@novartis.com, Wu X, Sills MA
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 2005 Oct; Vol. 10 (7), pp. 695-704. Date of Electronic Publication: 2005 Aug 29.
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3
Akademický článek
Further comparison of primary hit identification by different assay technologies and effects of assay measurement variability.
Autor: Wu X; Novartis Institute for Biomedical Research, Cambridge, MA, USA., Sills MA, Zhang JH
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 2005 Sep; Vol. 10 (6), pp. 581-9. Date of Electronic Publication: 2005 Aug 15.
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4
Akademický článek
Comparison of assay technologies for a nuclear receptor assay screen reveals differences in the sets of identified functional antagonists.
Autor: Wu X; Exelixis, South San Francisco, CA 94083-0511, USA. swu@exelixis.com, Glickman JF, Bowen BR, Sills MA
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 2003 Aug; Vol. 8 (4), pp. 381-92.
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5
Akademický článek
Comparison of assay technologies for a tyrosine kinase assay generates different results in high throughput screening.
Autor: Sills MA; Novartis Institute for Biomedical Research, Summit, NJ 07901, USA. matthew.sills@pharma.novartis.com, Weiss D, Pham Q, Schweitzer R, Wu X, Wu JJ
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 2002 Jun; Vol. 7 (3), pp. 191-214.
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6
Akademický článek
Microxine, a new cdc2 kinase inhibitor from the Australian marine sponge Microxina species.
Autor: Killday KB; Division of Biomedical Marine Research, Harbor Branch Oceanographic Institution, Inc., 5600 US 1 North, Ft. Pierce, Florida 34946, USA., Yarwood D, Sills MA, Murphy PT, Hooper JN, Wright AE
Publikováno v: Journal of natural products [J Nat Prod] 2001 Apr; Vol. 64 (4), pp. 525-6.
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7
Akademický článek
The discovery and characterization of an interleukin 6 cytokine family antagonist protein from a marine sponge, Callyspongia sp.
Autor: Peppard JV, Loo P, Sills MA, Wennogle L, Wright A, Pomponi S, Cueto M
Publikováno v: Advances in experimental medicine and biology [Adv Exp Med Biol] 2001; Vol. 484, pp. 77-87.
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8
Akademický článek
Measurement of cdk4 kinase activity using an affinity peptide-tagging technology.
Autor: Wu JJ; Novartis Institute for Biomedical Research, Novartis Pharmaceuticals Corporation, Summit, NJ 07901, USA. jinzi.wu@phrma.novartis.com, Yarwood DR, Sills MA, Chaudhuri B, Muller L, Zurini M, Sills MA
Publikováno v: Combinatorial chemistry & high throughput screening [Comb Chem High Throughput Screen] 2000 Feb; Vol. 3 (1), pp. 27-36.
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9
Akademický článek
Identification of a high-affinity anti-phosphoserine antibody for the development of a homogeneous fluorescence polarization assay of protein kinase C.
Autor: Wu JJ; Immunex Corporation, Seattle, WA 98101, USA. jinziwu@yahoo.com, Yarwood DR, Pham Q, Sills MA
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 2000 Feb; Vol. 5 (1), pp. 23-30.
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10
Akademický článek
Digital Imaging as a Detection Method for a Fluorescent Protease Assay in 96-Well and Miniaturized Assay Plate Formats.
Autor: Abriola L; Novartis Institute of Biomedical Research, Summit, NJ., Chin M, Fuerst P, Schweitzer R, Sills MA
Publikováno v: Journal of biomolecular screening [J Biomol Screen] 1999; Vol. 4 (3), pp. 121-127.
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