Zobrazeno 1 - 10
of 5 365
pro vyhledávání: '"M4"'
Autor:
Cadeddu R; Department of Pharmacology and Toxicology, College of Pharmacy, University of Utah, Salt Lake City, Utah, USA., Braccagni G; Department of Pharmacology and Toxicology, College of Pharmacy, University of Utah, Salt Lake City, Utah, USA., Branca C; Department of Pharmacology and Toxicology, College of Pharmacy, University of Utah, Salt Lake City, Utah, USA., van Luik ER; Department of Pharmacology and Toxicology, College of Pharmacy, University of Utah, Salt Lake City, Utah, USA., Pittenger C; Department of Psychiatry, School of Medicine, Yale University, New Haven, Connecticut, USA.; Department of Psychology, School of Arts and Sciences, Yale University, New Haven, Connecticut, USA.; Child Study Center, School of Medicine, Yale University, New Haven, Connecticut, USA.; Center for Brain and Mind Health, School of Medicine, Yale University, New Haven, Connecticut, USA., Thomsen MS; Neuroscience Research, H. Lundbeck A/S, Valby, Copenhagen, Denmark., Bortolato M; Department of Pharmacology and Toxicology, College of Pharmacy, University of Utah, Salt Lake City, Utah, USA.
Publikováno v:
British journal of pharmacology [Br J Pharmacol] 2024 Sep; Vol. 181 (17), pp. 3064-3081. Date of Electronic Publication: 2024 Apr 30.
Autor:
Liu B; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia., Thompson G; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia., Jörg M; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia., Barnes N; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia., Thal DM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia.; Australian Research Council Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria 3052, Australia., Christopoulos A; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia.; Australian Research Council Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria 3052, Australia.; Neuromedicines Discovery Centre, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria 3052, Australia., Capuano B; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia., Valant C; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia.; Australian Research Council Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria 3052, Australia., Scammells PJ; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2024 Aug 08; Vol. 67 (15), pp. 13286-13304. Date of Electronic Publication: 2024 Jul 18.
Autor:
Belov V; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Guehl NJ; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Duvvuri S; Cerevel Therapeutics, LLC, Cambridge, MA, USA., Iredale P; Cerevel Therapeutics, LLC, Cambridge, MA, USA., Moon SH; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Dhaynaut M; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Chakilam S; Cerevel Therapeutics, LLC, Cambridge, MA, USA., MacDonagh AC; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Rice PA; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Yokell DL; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Renger JJ; Cerevel Therapeutics, LLC, Cambridge, MA, USA., El Fakhri G; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA., Normandin MD; Gordon Center for Medical Imaging, Massachusetts General Hospital, Harvard Medical School, Boston, MA, USA.
Publikováno v:
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism [J Cereb Blood Flow Metab] 2024 Aug; Vol. 44 (8), pp. 1329-1342. Date of Electronic Publication: 2024 Mar 13.
Autor:
Balakrishnan AS; Laboratory of Neuropsychiatry, Psychiatric Centre Copenhagen, Mental Health Services in the Capital Region of Denmark and Copenhagen University Hospital - Bispebjerg and Frederiksberg Hospital, Copenhagen, Denmark; Department of Neuroscience, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark., Johansen LBE; Laboratory of Neuropsychiatry, Psychiatric Centre Copenhagen, Mental Health Services in the Capital Region of Denmark and Copenhagen University Hospital - Bispebjerg and Frederiksberg Hospital, Copenhagen, Denmark., Lindsley CW; Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Vanderbilt University Medical Center, Nashville, TN, USA., Conn PJ; Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Vanderbilt University Medical Center, Nashville, TN, USA., Thomsen M; Laboratory of Neuropsychiatry, Psychiatric Centre Copenhagen, Mental Health Services in the Capital Region of Denmark and Copenhagen University Hospital - Bispebjerg and Frederiksberg Hospital, Copenhagen, Denmark; Department of Neuroscience, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark. Electronic address: morgan.hermann.thomsen@regionh.dk.
Publikováno v:
Progress in neuro-psychopharmacology & biological psychiatry [Prog Neuropsychopharmacol Biol Psychiatry] 2024 Aug 30; Vol. 134, pp. 111079. Date of Electronic Publication: 2024 Jun 29.
Autor:
Butler CR; Medicine Design, Medicinal Chemistry, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Popiolek M; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., McAllister LA; Medicine Design, Medicinal Chemistry, Pfizer Inc., Cambridge, Massachusetts 02139, United States., LaChapelle EA; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Kramer M; Medicine Design, Pharmacokinetics, Dynamics and Metabolism, Pfizer Inc., Groton, Connecticut 06340, United States., Beck EM; Medicine Design, Medicinal Chemistry, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Mente S; Medicine Design, Medicinal Chemistry, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Brodney MA; Medicine Design, Medicinal Chemistry, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Brown M; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Gilbert A; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Helal C; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Ogilvie K; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Starr J; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Uccello D; Medicine Design, Medicinal Chemistry, Pfizer Inc., Groton, Connecticut 06340, United States., Grimwood S; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Edgerton J; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Garst-Orozco J; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Kozak R; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Lotarski S; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Rossi A; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., Smith D; Internal Medicine, Pfizer Inc., Cambridge, Massachusetts 02139, United States., O'Connor R; Discovery Sciences, Primary Pharmacology, Pfizer Inc., Groton, Connecticut 06340, United States., Lazzaro J; Discovery Sciences, Primary Pharmacology, Pfizer Inc., Groton, Connecticut 06340, United States., Steppan C; Discovery Sciences, Primary Pharmacology, Pfizer Inc., Groton, Connecticut 06340, United States., Steyn SJ; Medicine Design, Pharmacokinetics, Dynamics and Metabolism, Pfizer Inc., Groton, Connecticut 06340, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2024 Jul 11; Vol. 67 (13), pp. 10831-10847. Date of Electronic Publication: 2024 Jun 18.
Autor:
Madrid LI; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia., Hafey K; Mater Research Institute - The University of Queensland, Translational Research Institute, Brisbane QLD 4102, Queensland, Australia., Bandhavkar S; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia.; Mater Research Institute - The University of Queensland, Translational Research Institute, Brisbane QLD 4102, Queensland, Australia., Bodea GO; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia.; Mater Research Institute - The University of Queensland, Translational Research Institute, Brisbane QLD 4102, Queensland, Australia., Jimenez-Martin J; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia., Milne M; School of Biomedical Sciences, The University of Queensland, Brisbane QLD 4072, Queensland, Australia., Walker TL; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia., Faulkner GJ; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia.; Mater Research Institute - The University of Queensland, Translational Research Institute, Brisbane QLD 4102, Queensland, Australia., Coulson EJ; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia.; School of Biomedical Sciences, The University of Queensland, Brisbane QLD 4072, Queensland, Australia., Jhaveri DJ; Queensland Brain Institute, The University of Queensland, Brisbane QLD 4072, Queensland, Australia.; Mater Research Institute - The University of Queensland, Translational Research Institute, Brisbane QLD 4102, Queensland, Australia.
Publikováno v:
Development (Cambridge, England) [Development] 2024 Jan 01; Vol. 151 (1). Date of Electronic Publication: 2024 Jan 02.
Autor:
Vuckovic Z; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Wang J; Center for Computational Biology and Department of Molecular Biosciences, University of Kansas, Lawrence, United States., Pham V; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Mobbs JI; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Belousoff MJ; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Bhattarai A; Center for Computational Biology and Department of Molecular Biosciences, University of Kansas, Lawrence, United States., Burger WAC; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Thompson G; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Yeasmin M; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Nawaratne V; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Leach K; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., van der Westhuizen ET; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Khajehali E; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Liang YL; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Glukhova A; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Wootten D; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Lindsley CW; Department of Pharmacology, Warren Center for Neuroscience Drug Discovery and Department of Chemistry, Warren Center for Neuroscience Drug Discovery, Vanderbilt University, Nashville, United States., Tobin A; The Centre for Translational Pharmacology, Advanced Research Centre (ARC), College of Medical, Veterinary and Life Sciences, University of Glasgow, Glasgow, United Kingdom., Sexton P; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Danev R; Graduate School of Medicine, University of Tokyo, Tokyo, Japan., Valant C; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Miao Y; Center for Computational Biology and Department of Molecular Biosciences, University of Kansas, Lawrence, United States., Christopoulos A; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; Neuromedicines Discovery Centre, Monash University, Parkville, Australia., Thal DM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.
Publikováno v:
ELife [Elife] 2023 May 30; Vol. 12. Date of Electronic Publication: 2023 May 30.
Autor:
Tsotsokou G; Laboratory of Physiology, University of Patras, Department of Medicine, Rion, Greece., Trompoukis G; Laboratory of Physiology, University of Patras, Department of Medicine, Rion, Greece., Papatheodoropoulos C; Laboratory of Physiology, University of Patras, Department of Medicine, Rion, Greece. Electronic address: cepapath@upatras.gr.
Publikováno v:
Molecular and cellular neurosciences [Mol Cell Neurosci] 2024 Jun; Vol. 129, pp. 103935. Date of Electronic Publication: 2024 May 03.
Autor:
Fu L; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China., Luo Y; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China., Niu L; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China., Lin Y; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China., Chen X; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China., Zhang J; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China., Tang W; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China.. Electronic address: twf@cpu.edu.cn., Chen Y; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China.. Electronic address: ydchen@cpu.edu.cn., Jiao Y; School of Science, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, PR China.. Electronic address: jiaoyu923@126.com.
Publikováno v:
Bioorganic & medicinal chemistry [Bioorg Med Chem] 2024 May 01; Vol. 105, pp. 117728. Date of Electronic Publication: 2024 Apr 16.
Autor:
Russell JK; Department of Pharmacology, Warren Center for Neuroscience Drug Discovery, and Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States., Ingram SM; Department of Pharmacology, Warren Center for Neuroscience Drug Discovery, and Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States., Teal LB; Department of Pharmacology, Warren Center for Neuroscience Drug Discovery, and Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States., Lindsley CW; Department of Pharmacology, Warren Center for Neuroscience Drug Discovery, and Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States., Jones CK; Department of Pharmacology, Warren Center for Neuroscience Drug Discovery, and Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States.
Publikováno v:
ACS chemical neuroscience [ACS Chem Neurosci] 2023 Feb 01; Vol. 14 (3), pp. 435-457. Date of Electronic Publication: 2023 Jan 19.