Zobrazeno 1 - 2
of 2
pro vyhledávání: '"M. Rosa Sánchez-Casado"'
Autor:
José Manuel Bartolomé-Nebreda, Thomas Steckler, Susana Conde-Ceide, Colleen M. Niswender, Chrysa Malosh, María Piedrafita, Meredith J. Noetzel, Claire Mackie, Paige N. Vinson, Jerri M. Rook, Gregor James Macdonald, M. Rosa Sánchez-Casado, P. Jeffrey Conn, Shaun R. Stauffer, Carlos M. Martínez-Viturro, Hilde Lavreysen, J. Scott Daniels, Carrie K. Jones, Mark Turlington, Thomas M. Bridges, Craig W. Lindsley
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 25:5115-5120
We report the optimization of a series of metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulators (PAMs) from an acyl dihydropyrazolo[1,5-a]pyrimidinone class. Investigation of exocyclic amide transpositions with this unique 5,6-bicy
Autor:
Sánchez Casado, M. Rosa1 msanc117@its.jnj.com, Ciordia Jiménez, Myriam1, Ariza Bueno, Manuela2, Barriol, Morgane2, Leenaerts, Joseph E.2, Pagliuca, Chiara2, Martínez Lamenca, Carolina2, De Lucas, Ana Isabel1, García, Aránzazu1, Trabanco, Andrés A.1 atrabanc@its.jnj.com, Rombouts, Frederik J. R.2 frombout@its.jnj.com
Publikováno v:
European Journal of Organic Chemistry. Aug2015, Vol. 2015 Issue 23, p5221-5229. 9p.