Zobrazeno 1 - 10 of 137 pro vyhledávání: '"M. Loriga"'
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Quinoxaline 1,4-dioxide: a versatile scaffold endowed with manifold activities
Autor: M. Loriga, Antonio Carta, P. Corona
Publikováno v: Current medicinal chemistry. 12(19)
Since 1940s, Quinoxaline 1,4-dioxides (QdNOs) are known as potent antibacterial agents, and subtherapeutic levels have been used to promote growth and improve efficiency of feed conversion in animal feed. They have also shown a selective cytotoxicity
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1c777514d2793c98dca3a2eab34b22e1
https://pubmed.ncbi.nlm.nih.gov/16178784
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Quinoxaline chemistry. Part 8. 2-[Anilino]-3-[carboxy]-6(7)-substituted quinoxalines as non classical antifolate agents. Synthesis and evaluation of in vitro anticancer, anti-HIV and antifungal activity
Autor: M, Loriga, P, Moro, P, Sanna, G, Paglietti, S, Zanetti
Publikováno v: Farmaco (Societa chimica italiana : 1989). 52(8-9)
Thirty quinoxalines bearing a substituted anilino group on position 2, a carboethoxy or carboxy group on position 3 and a trifluoromethyl group on position 6 or 7 of the heterocycle were prepared in order to evaluate in vitro anticancer activity. Pre
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::9bdccbe2bc4d9b3efaf76cbc9474c99c
https://pubmed.ncbi.nlm.nih.gov/9507661
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Quinoxaline chemistry. Part 7. 2-[aminobenzoates]- and 2-[aminobenzoylglutamate]-quinoxalines as classical antifolate agents. Synthesis and evaluation of in vitro anticancer, anti-HIV and antifungal activity
Autor: M, Loriga, S, Piras, P, Sanna, G, Paglietti
Publikováno v: Farmaco (Societa chimica italiana : 1989). 52(3)
Thirty-three quinoxalines bearing an aminobenzoyl or aminobenzoylglutamate group on position 2 and various substituents on position 3,6,7 of the heterocycle were prepared in order to evaluate in vitro anticancer activity. Preliminary screening perfor
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::97f4751e846e140b3da3cdbf96d9e8de
https://pubmed.ncbi.nlm.nih.gov/9212450
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Quinoxaline chemistry. Part 5. 2-(R)-benzylaminoquinoxalines as nonclassical antifolate agents. Synthesis and evaluation of in vitro anticancer activity
Autor: M, Loriga, M, Fiore, P, Sanna, G, Paglietti
Publikováno v: Farmaco (Societa chimica italiana : 1989). 51(8-9)
Thirty-one quinoxalines bearing a substituted benzylamino group on position 2 and various substituents on position 3,6,7 and 8 of the heterocycle were prepared in order to evaluate in vitro anticancer activity. Preliminary screening performed at NCI
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::eeacad9ad7937aff5fa88069ea4a791a
https://pubmed.ncbi.nlm.nih.gov/8930109
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Quinoxaline chemistry. Part 4. 2(R)-anilinoquinoxalines as nonclassical antifolate agents. Synthesis, structure elucidation and evaluation of in vitro anticancer activity
Autor: M, Loriga, M, Fiore, P, Sanna, G, Paglietti
Publikováno v: Farmaco (Societa chimica italiana : 1989). 50(5)
Thirty-five quinoxalines bearing a substituted aniline group on position 2 and various substituents on positions 3,6,7 and 8 were prepared in order to evaluate in vitro anticancer activity. Structural elucidation of some isomeric quinoxalinones forme
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::bd4f6fa65d9089e61fa649d4eb6576f5
https://pubmed.ncbi.nlm.nih.gov/7626163
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Synthesis and evaluation of gastroprotective activity of omeprazole related benzimidazole, imidazo[4,5-b]pyridine and quinoxaline 2-substituted derivatives
Autor: S, Piras, M, Loriga, G, Paglietti, F, Sparatore, M P, Demontis, M V, Varoni, M C, Fattaccio, V, Anania
Publikováno v: Farmaco (Societa chimica italiana : 1989). 48(9)
Twenty compounds possessing benzimidazole, imidazo[4,5-b]pyridine and quinoxaline structure bearing either a substituted arylmethylmercapto- or an arylmethylsulfinyl group in position 2 were prepared in order to evaluate an antiulcer and gastroprotec
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::526b50ceec9277223dcb38fda45e002e
https://pubmed.ncbi.nlm.nih.gov/8259982
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Synthesis of substituted DL-3(5-benzazolyl)alanines as dopa and alpha-methyldopa analogs and their effects on dopamine beta-hydroxylase, tyrosinase and diphenoloxidase
Autor: M, Loriga, G, Paglietti, F, Sparatore, G, Pinna, A, Sisini
Publikováno v: Farmaco (Societa chimica italiana : 1989). 47(4)
The influence of bioisosteric replacement of catechol moiety of L-Dopa and alpha-Methyldopa with benzimidazole and benzotriazole ring has been examined on dopamine beta-hydroxylase and tyrosinase, in order to evidentiate an inhibitory activity on the
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::62684fa7fcd3abf71ae32786c5490b3c
https://pubmed.ncbi.nlm.nih.gov/1388592
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Synthesis and evaluation of gastroprotective and antiulcer activity of some 2-substituted-1H-imidazo[4,5-b] pyridines and -1H-benzimidazoles
Autor: M, Loriga, G, Paglietti, S, Piras, F, Sparatore, V, Anania, M P, Demontis, M V, Varoni, M C, Fattaccio
Publikováno v: Farmaco (Societa chimica italiana : 1989). 47(3)
Several compounds possessing imidazo[4,5-b]pyridine and benzimidazole structure bearing substituents in position 2 were prepared in order to evaluate an anti-ulcer and gastroprotective activity in rat pylorus ligature, in comparison with omeprazole.
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::7660d20edb3707d5c986efabd1548bcf
https://pubmed.ncbi.nlm.nih.gov/1503593
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