Zobrazeno 1 - 6
of 6
pro vyhledávání: '"M. Joelle Dill"'
Autor:
Matthew W. Carson, Robert J. Barr, Dana Sindelar, Daniel Timothy Kohlman, Bradley Condon, David K. Clawson, A. Pustilnik, M. Joelle Dill, James S. Bean, John G. Luz, Michael J. Coghlan, Milan Maletic
Publikováno v:
Journal of Medicinal Chemistry. 58:6607-6618
To further elucidate the structural activity correlation of glucocorticoid receptor (GR) antagonism, the crystal structure of the GR ligand-binding domain (GR LBD) complex with a nonsteroidal antagonist, compound 8, was determined. This novel indole
Publikováno v:
Pharmacology Biochemistry and Behavior. 112:1-8
Serotonin acts through receptors controlling several physiological functions, including energy homeostasis regulation and food intake. Recent experiments demonstrated that 5-HT1A receptor antagonists reduce food intake. We sought to examine the micro
Autor:
Jesline T. Alexander-Chacko, Traci A. Czyzyk, Dana Sindelar, Michael A. Statnick, M. Joelle Dill
Publikováno v:
Neuromethods ISBN: 9781627031035
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::334b70169b77891ad0b1b021be860993
https://doi.org/10.1007/978-1-62703-104-2_5
https://doi.org/10.1007/978-1-62703-104-2_5
Autor:
Samuel W. Oldham, M. Joelle Dill, Brian Morgan Watson, Craig W. Lindsley, Don Richard Finley, Dana Sindelar, Lisa Selsam Beavers, Cynthia Darshini Jesudason, Philip Arthur Hipskind, Robert Alan Gadski, Ajay Singh, Christopher Stephen Siedem, Jeffrey W Cramer, R. Todd Pickard, F. Craig Stevens
Publikováno v:
Bioorganicmedicinal chemistry letters. 16(13)
The synthesis and biological evaluation of novel tetrahydroisoquinoline, tetrahydroquinoline, and tetrahydroazepine antagonists of the human and rat H(3) receptors are described. The substitution around these rings as well as the nature of the substi
Autor:
Richard Todd Pickard, Robert Alan Gadski, Jesline T. Alexander-Chacko, Dennis P. Smith, Mary L Shepperd, Jeffrey W Cramer, M. Joelle Dill, Dana Sindelar
Publikováno v:
Pharmacology, biochemistry, and behavior. 78(2)
The central histamine 3 receptor (H3R) is a presynaptic autoreceptor that regulates neuronal release and synthesis of histamine, and is thought to play a key role in controlling numerous central nervous system (CNS)-mediated parameters, including ene
Autor:
John G. Luz, MatthewW. Carson, Bradley Condon, David Clawson, Anna Pustilnik, Daniel T. Kohlman, Robert J. Barr, James S. Bean, M. Joelle Dill, Dana K Sindelar, Milan Maletic, Michael J. Coghlan
Publikováno v:
Journal of Medicinal Chemistry; Aug2015, Vol. 58 Issue 16, p6607-6618, 12p