Zobrazeno 1 - 9
of 9
pro vyhledávání: '"M. J. Kates"'
Autor:
J. H. Schauble, M. J. Kates
Publikováno v:
The Journal of Organic Chemistry. 61:4164-4167
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::add9dd1813c9e92a0e97e0db98c2800f
https://doi.org/10.1021/jo9601977
https://doi.org/10.1021/jo9601977
Autor:
M. J. Kates, J. Herman Schauble
Publikováno v:
Journal of Heterocyclic Chemistry. 32:971-978
Reaction of five-membered ring anhydrides with sodium sulfide has previously been employed for synthesis of the corresponding thioanhydrides in low yields. Re-examination of the stoichiometry reveals reaction of cyclic anhydride with sodium sulfide (
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a3e1a3ff6573d2764a6fdbed2c854e64
https://doi.org/10.1002/jhet.5570320350
https://doi.org/10.1002/jhet.5570320350
Autor:
M. J. Kates, J. H. Schauble
Publikováno v:
ChemInform. 26
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::84b53878ca336d5720906fc60d2fcd0a
https://doi.org/10.1002/chin.199545075
https://doi.org/10.1002/chin.199545075
Autor:
J. H. Schauble, M. J. Kates
Publikováno v:
ChemInform. 27
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::21732037647b888397ff48f24d6961bc
https://doi.org/10.1002/chin.199610117
https://doi.org/10.1002/chin.199610117
Autor:
J. H. Schauble, M. J. Kates
Publikováno v:
ChemInform. 27
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::52ecc8eef177c8b74783896d82679ac7
https://doi.org/10.1002/chin.199641248
https://doi.org/10.1002/chin.199641248
Autor:
M. J. Kates, J. Herman Schauble
Publikováno v:
The Journal of Organic Chemistry. 59:494-496
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5c75569e40081653d121ecd0776d0ea0
https://doi.org/10.1021/jo00081a037
https://doi.org/10.1021/jo00081a037
Autor:
Thomas J. Caggiano, John J. Fitzgerald, Thomas E. Christos, John M. Kulishoff, Michael L. McCaleb, Kurt E. Steiner, M. J. Kates, Robin Moore, Kenneth L. Kees
Publikováno v:
Journal of medicinal chemistry. 38(4)
Bioisosteric substitution was used as a tool to generate several new structural alternatives to the thiazolidine-2,4-dione and tetrazole heterocycles as potential antidiabetic agents. Among the initial leads that emerged from this strategy, a family
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fcc8a8e8b5fad755d07884ec21585358
https://pubmed.ncbi.nlm.nih.gov/7861410
https://pubmed.ncbi.nlm.nih.gov/7861410
Autor:
Kenneth Keavey, Russell J. Thomas, Thomas McDonagh, Hamelin Estelle, Rory A. J. Curtis, Jonathan Barker, Peter S. DiStefano, Patricia Amouzegh, Jean-François Pons, Wei Tsung Yau, Andrew Napper, Jeffrey Hixon, M. J. Kates, Stephen Jones, Jeffrey O. Saunders, Manuel A. Navia, Adam Flegg
Publikováno v:
Journal of Medicinal Chemistry. 50:1086-1086
High-throughput screening against the human sirtuin SIRT1 led to the discovery of a series of indoles as potent inhibitors that are selective for SIRT1 over other deacetylases and NAD-processing enzymes. The most potent compounds described herein inh
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::688909b83bf7f2eb12f50310167448a1
https://doi.org/10.1021/jm061430o
https://doi.org/10.1021/jm061430o
Autor:
M. J. Kates, J. Herman Schauble
Publikováno v:
The Journal of Organic Chemistry. 60:6676-6677
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::110d346cde50f16868dc9971b4e2f052
https://doi.org/10.1021/jo00126a013
https://doi.org/10.1021/jo00126a013