Zobrazeno 1 - 1
of 1
pro vyhledávání: '"M. Gabriella Brasca"'
Autor:
Paolo Polucci, Suzanne Metz, Anna Vulpetti, Antonella Ermoli, M. Gabriella Brasca, Roberto D'Alessio, Alberto Bargiotti, Marcellino Tibolla, Alexander D. Cameron, Paolo Pevarello, Vazquez Michael L, Aurelio Marsiglio, Fulvia Roletto
Publikováno v:
Bioorganicmedicinal chemistry letters. 15(5)
The synthesis and the preliminary expansion of this new class of CDK2 inhibitors are presented. The synthesis was accomplished using a solution-phase protocol amenable to rapid parallel expansion and suitable to be scaled-up in view of possible lead