Zobrazeno 1 - 10
of 67
pro vyhledávání: '"Lucien Stella"'
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 103:361-366
The methyl N-(1-phenylethyl)-α-iminoacetate undergoes zinc iodide activated aza-Diels-Alder cycloaddition reactions with electron rich conjugated dienes. Cyclic α-amino-acids are formed in good yields, with complete regioselectivity, but the extent
Publikováno v:
Tetrahedron. 63:3205-3216
Selected N-sulfenylimines act as good nucleophilic partners in the Staudinger reaction with methoxy- and benzyloxy-ketenes. The choice of diisopropylethylamine as a non-nucleophilic Lewis base for the generation of ketenes from acid chlorides is a de
Autor:
Lucien Stella
Publikováno v:
Angewandte Chemie. 95:368-380
Viele N-Chlor-alkylamine mit Doppelbindung(en) im Alkylrest zerfallen homolytisch in Chloratome und Aminylradikale, die unter intramolekularer Addition cyclisieren. Die Natur der Aminylradikale (neutral, protoniert oder an Metallsalze gebunden) schei
Publikováno v:
Tetrahedron. 59:3719-3727
We report the use of 19 F NMR as a simple means to monitor reactions on a solid phase. Multi-step sequences including protection, coupling, deprotection, condensation, cycloaddition and cleavage steps are described in the case of multicomponent react
Publikováno v:
Synthetic Communications. 30:3685-3691
The reaction of chloroacetyl chloride and triethylamine with a chiral imine derived from the combination of methyl glyoxylate and protected L-threonine gave two optically active α-amino acid derivatives with a cis-substituted β-lactam skeleton in a
Autor:
Alain Commercon, Dominique Mouysset, Patricia Perfetti, Serge Mignani, Lucien Stella, Michel Barreau
Publikováno v:
Scopus-Elsevier
Selected imines of methyl glyoxylate act as good partners in the Staudinger cycloaddition reaction with a series of substituted ketenes. The cis stereoselectivity is almost complete with electron-donor substituted ketenes, but the asymmetric inductio
Publikováno v:
Tetrahedron. 54:4579-4590
A new series of conformationally restricted retinoids (3-aryl-3-methyl-2,3-dihydro-benzofurans) have been prepared through a palladium-catalyzed tandem cyclisation-hydride capture. The use of enantiopure BINAP-Pd catalyst allowed asymmetric synthesis
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 7:2289-2294
A series of 3-aryl-2H-1-benzopyrancarboxylic acid derivatives was synthesized and evaluated as Retinoic Acid Receptor (RAR) agonists. By modifications of the 3-aryl group, we have obtained new retinoids exhibiting potent cellular differentiating acti
Publikováno v:
Tetrahedron. 49:8397-8406
Treatment of the acyclic allyl-octa-4,7-dienyl N-chloroamine 5 by titanium trichloride induces a chain process including three consecutive regio- and stereo-selective homolytic cyclisations. As a result of these selectivities, the main product of the
Autor:
H. Abraham, Lucien Stella
Publikováno v:
ChemInform. 22