Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Luca G. Moccia"'
Autor:
Ilaria Sartori, Laura Zonzini, Laurie J. Gordon, Angela Worby, Stefano Fontana, Manuela Borriello, Silvia Bison, Jeannette M. Watson, Steven Mark Bromidge, Giovanna Dal Forno, Colin Philip Leslie, Alessandra Pasquarello, Anna Sava, Luca G. Moccia, Barbara Bertani, Roberto Arban, Daniele Donati, Enrica Granci, Valeria Zucchelli, Paolo Cavanni, Massimo Gianotti, Romano Di-Fabio
Publikováno v:
Journal of Medicinal Chemistry. 53:5827-5843
Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of fused tricyclic benzoxazines which are potent 5-HT1A/B/D receptor antagonists with and wit
Autor:
Davide Pozzi, Olivier Corminboeuf, Eric A. Ertel, Thomas Pfeifer, Catherine Roch, Bibia Heidmann, Ruben de Kanter, Melanie Kessler, Bruno Capeleto, Michael Toeroek-Schafroth, Jacques Mawet, Isabelle Reymond, Simon Stamm, Romain Siegrist, Olivier Bezencon, Richard Moon, Sylvia Richard, Elvire Fournier, Markus Rey, Luca G. Moccia
Publikováno v:
Journal of Medicinal Chemistry. 60:9769
We report here the discovery and pharmacological characterization of N-(1-benzyl-1H-pyrazol-3-yl)-2-phenylacetamide derivatives as potent, selective, brain-penetrating T-type calcium channel blockers. Optimization focused mainly on solubility, brain