Zobrazeno 1 - 10
of 19
pro vyhledávání: '"Lisa Kindler"'
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
Supplementary Methods
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::38d0dc26b8998855020bf945222d1189
https://doi.org/10.1158/1535-7163.22507273.v1
https://doi.org/10.1158/1535-7163.22507273.v1
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
In vivo effect of treatment on body weight loss.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::952c561d8520c3c104049374b206e09a
https://doi.org/10.1158/1535-7163.22507276.v1
https://doi.org/10.1158/1535-7163.22507276.v1
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
Generation of vemurafenib-resistant A375 model in vivo.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::282e0d00cc1b76255f633d6c5a03ff19
https://doi.org/10.1158/1535-7163.22507279
https://doi.org/10.1158/1535-7163.22507279
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
Summary of antitumor activity of LY3214996 and other MAPK pathway inhibitors in cancer models with dominant MAPK pathway alterations
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1f6c4588b08e0998a9a4807fcc3a711c
https://doi.org/10.1158/1535-7163.22507261.v1
https://doi.org/10.1158/1535-7163.22507261.v1
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
Biochemical and cellular selectivity profile of LY3214996 (DiscoveRx and ActiveX data)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::833c6a5db8886d95637d97ec87b52a9f
https://doi.org/10.1158/1535-7163.22507267
https://doi.org/10.1158/1535-7163.22507267
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
Time-dependent increase in apoptosis induction by LY3214996, pan-RAF inhibitor LY3009120 and MEK inhibitor trametinib in KRAS-mutant HCT116 colorectal cancer cells.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04e72d719f970d347e2ae4c00c36677b
https://doi.org/10.1158/1535-7163.22507294
https://doi.org/10.1158/1535-7163.22507294
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
Inhibition of downstream signaling by LY3214996 in a BRAF-mutant A375 melanoma cells (A) and MEK1 mutant SW48 colorectal cancer cells (B).
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1e3699d33e036f707d9247a30025ba8e
https://doi.org/10.1158/1535-7163.22507288
https://doi.org/10.1158/1535-7163.22507288
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
pan-RAF inhibitor can block increase in ERK phosphorylation due to inhibition of negative feedback on CRAF by ERK inhibitor.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0595bf4108d4385cc3a3e7ed92a8b16a
https://doi.org/10.1158/1535-7163.22507291.v1
https://doi.org/10.1158/1535-7163.22507291.v1
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
The ERK pathway is critical in oncogenesis; aberrations in components of this pathway are common in approximately 30% of human cancers. ERK1/2 (ERK) regulates cell proliferation, differentiation, and survival and is the terminal node of the pathway.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7b6b83642603b80faa51fcf05c737a2b
https://doi.org/10.1158/1535-7163.c.6538636.v1
https://doi.org/10.1158/1535-7163.c.6538636.v1
Autor:
Sheng-Bin Peng, Sajan Joseph, Ramon V. Tiu, Gregory D. Plowman, Michael J. Rodriguez, Eunice Yuen, Jennie Walgren, Jason Manro, Andrew J. Dropsey, Denis McCann, Xi Rao, Robert D. Van Horn, Meghann Pogue, Xiu-Juan Yuan, Yan Zhai, Bryan Anderson, Wenjuan Wu, Robert S. Flack, Lisa Kindler, Weihua Shen, Matthew Whitesell, Baohui Zhao, Shufen Cai, William T. McMillen, Shripad V. Bhagwat
In vivo effect of treatment on body weight loss.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::92f5878656a7dcf087ed5e9f7e535f63
https://doi.org/10.1158/1535-7163.22507282.v1
https://doi.org/10.1158/1535-7163.22507282.v1