Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency

Autor: Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.

Publikováno v: In Bioorganic & Medicinal Chemistry Letters 1999 9(9):1311-1316

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Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus

Autor: Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.

Publikováno v: In Bioorganic & Medicinal Chemistry Letters 1998 8(21):3081-3086

Benzodiazepines as potent and selective bradykinin B1 antagonists.

Autor: Wood MR; Department of Medicinal Chemistry, Merck Research Laboratories, P.O. Box 4, West Point, Pennsylvania 19486, USA. michael_wood2@merck.com, Kim JJ, Han W, Dorsey BD, Homnick CF, DiPardo RM, Kuduk SD, MacNeil T, Murphy KL, Lis EV, Ransom RW, Stump GL, Lynch JJ, O'Malley SS, Miller PJ, Chen TB, Harrell CM, Chang RS, Sandhu P, Ellis JD, Bondiskey PJ, Pettibone DJ, Freidinger RM, Bock MG

Publikováno v: Journal of medicinal chemistry [J Med Chem] 2003 May 08; Vol. 46 (10), pp. 1803-6.