Zobrazeno 1 - 10
of 91
pro vyhledávání: '"Leigh Zawel"'
Autor:
Robert N Booher, Harold Hatch, Brian M Dolinski, Thi Nguyen, Lauren Harmonay, Ali-Samer Al-Assaad, Mark Ayers, Michael Nebozhyn, Andrey Loboda, Heather A Hirsch, Theresa Zhang, Bin Shi, Carrie E Merkel, Minilik H Angagaw, Yaolin Wang, Brian J Long, Xianlu Q Lennon, Nathan Miselis, Vincenzo Pucci, James W Monahan, Junghoon Lee, Anna Georgieva Kondic, Eun Kyung Im, David Mauro, Rebecca Blanchard, Gary Gilliland, Stephen E Fawell, Leigh Zawel, Alwin G Schuller, Peter Strack
Publikováno v:
PLoS ONE, Vol 9, Iss 10, p e108371 (2014)
Dinaciclib is a potent CDK1, 2, 5 and 9 inhibitor being developed for the treatment of cancer. Additional understanding of antitumor mechanisms and identification of predictive biomarkers are important for its clinical development. Here we demonstrat
Externí odkaz:
https://doaj.org/article/b410584fec734e0e84be6d52d5590862
Autor:
Sriram Sathyanarayanan, Jon C. Aster, X. Shirley Liu, Warren S. Pear, Bradley E. Bernstein, Birgit Knoechel, Brandon E. Kremer, Theresa Zhang, Gary Gilliland, Stephen Fawell, Leigh Zawel, Christopher Moskaluk, Brian B. Haines, Jason Laskey, Michael Kluk, Philip W. Garrett-Engele, John MacLean, Chris Ware, Jing Yuan, Chongzhi Zang, Hongfang Wang, Li Pan, Andrew Truong, Serguei Lejnine, Alexander Stoeck
human Breast tumor Notch gene coverage annotations.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::772c70e0961cfb13b051a4fed2d019a3
https://doi.org/10.1158/2159-8290.22529885.v1
https://doi.org/10.1158/2159-8290.22529885.v1
Autor:
Sriram Sathyanarayanan, Jon C. Aster, X. Shirley Liu, Warren S. Pear, Bradley E. Bernstein, Birgit Knoechel, Brandon E. Kremer, Theresa Zhang, Gary Gilliland, Stephen Fawell, Leigh Zawel, Christopher Moskaluk, Brian B. Haines, Jason Laskey, Michael Kluk, Philip W. Garrett-Engele, John MacLean, Chris Ware, Jing Yuan, Chongzhi Zang, Hongfang Wang, Li Pan, Andrew Truong, Serguei Lejnine, Alexander Stoeck
S1: NOTCH gene rearrangement in breast cancer cell lines and human breast tumors. S2: NOTCH gene rearrangement and sensitivity to MRK-003. S3: HES4 expression is associated with NOTCH gene-rearrangement or activating mutation in NOTCH. S4: HES4 expre
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ba7e587c75653d144fc20a17c000c13a
https://doi.org/10.1158/2159-8290.22529894.v1
https://doi.org/10.1158/2159-8290.22529894.v1
Autor:
Yan Wang, Erick J. Morris, Richard E. Middleton, Paul T. Kirschmeier, Leigh Zawel, Cynthia Seidel-Dugan, Pasi A. Jánne, Kwok-Kin Wong, Kumiko Nagashima, Heather Hirsch, Steven Ripley, Chris Hulton, Weiqun Zhang, Rossana Chung, Stephen Wu, Peter Strack, Thi T. Nguyen, Brian Dolinski, Jongwon Lim, Rafael Fernandez, Haiyan Yan, Qi Pan, Asli Muvaffak
PDF file - 1334KB, S1. IC50 values of TBK1 inhibitors Compound number 5, Compound number 4 and Compound number 3 from the selected PDAC, colorectal cancer and NSCLC cancer cell lines using are shown. Table 1S. List of shRNAs Targeting TBK1 Table 2S.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::98442b5d4353d94a24d08eb4fa097ec2
https://doi.org/10.1158/1541-7786.22511083
https://doi.org/10.1158/1541-7786.22511083
Autor:
Stuart D. Shumway, D. Gary Gilliland, Stephen E. Fawell, Leigh Zawel, Carlo Toniatti, Yair Benita, Igor Feldman, Heather A. Hirsch, Brian Long, Alwin G. Schuller, Melissa S. Hurd, Yaping Liu, Jing Li, Amy D. Guertin
XLSX file - 155K, Proliferation assay EC50 results for MK-1775 in diverse tumor cell lines.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::492fc6bcd867d365445a93212bebdc1b
https://doi.org/10.1158/1535-7163.22500334
https://doi.org/10.1158/1535-7163.22500334
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
HTRF and Biacore binding data for active and inactive ERK1 in the presence of SCH772984
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5a41d041f5824e4e438c00c030ecb53b
https://doi.org/10.1158/1535-7163.22509012.v1
https://doi.org/10.1158/1535-7163.22509012.v1
Autor:
Sriram Sathyanarayanan, Jon C. Aster, X. Shirley Liu, Warren S. Pear, Bradley E. Bernstein, Birgit Knoechel, Brandon E. Kremer, Theresa Zhang, Gary Gilliland, Stephen Fawell, Leigh Zawel, Christopher Moskaluk, Brian B. Haines, Jason Laskey, Michael Kluk, Philip W. Garrett-Engele, John MacLean, Chris Ware, Jing Yuan, Chongzhi Zang, Hongfang Wang, Li Pan, Andrew Truong, Serguei Lejnine, Alexander Stoeck
File includes genomic analysis, cell cycle and cell proliferation analysis.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::be61200c03fe3c0610304a985d3928e9
https://doi.org/10.1158/2159-8290.22529891.v1
https://doi.org/10.1158/2159-8290.22529891.v1
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
HTRF and Biacore binding data for active and inactive ERK1 in the presence of SCH772984
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3185945c7ae768bd2e93b8d986a09ade
https://doi.org/10.1158/1535-7163.22508997
https://doi.org/10.1158/1535-7163.22508997
Autor:
Sriram Sathyanarayanan, Jon C. Aster, X. Shirley Liu, Warren S. Pear, Bradley E. Bernstein, Birgit Knoechel, Brandon E. Kremer, Theresa Zhang, Gary Gilliland, Stephen Fawell, Leigh Zawel, Christopher Moskaluk, Brian B. Haines, Jason Laskey, Michael Kluk, Philip W. Garrett-Engele, John MacLean, Chris Ware, Jing Yuan, Chongzhi Zang, Hongfang Wang, Li Pan, Andrew Truong, Serguei Lejnine, Alexander Stoeck
Table S1: Analysis of Notch gene rearrangements in triple negative breast cancer subtypes. Table S2: Genes whose expression correlates with Notch gene-rearrangement status in cancer cell lines. Table S3: Genes whose expression correlates with Notch g
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dc068e95ade438f4b5a9a2cb23c5fe1
https://doi.org/10.1158/2159-8290.22529882.v1
https://doi.org/10.1158/2159-8290.22529882.v1
Autor:
Ahmed A. Samatar, Stephen Fawell, Leigh Zawel, Lata Jayaraman, D. Gary Gilliland, Daniel Hicklin, W. Robert Bishop, Paul Kirschmeier, David Witter, Phieng Siliphaivanh, Ulrike Philippar, Marc R. Pelletier, Bart A. Lutterbach, Ling Zhang, Pierre Daublain, Liang Zhu, Boga Sobhana Babu, Xiaolei Gao, Sunil Paliwal, Joe Kelly, James Wang, Alan Hruza, Gerald Shipps, Li Xiao, Jagdish Desai, Elaine M. Pinheiro, Minilik H. Angagaw, Shuxia Zhao, Rumin Zhang, William Windsor, Edward DiNunzio, Jenny Liu, Brian Long, Stuart Black, Weihong Jin, Yongi Deng, Donna Carr, Alan Cooper, Hugh Zhu, Priya Dayananth, Clifford R. Restaino, Sharda Jha, Erick J. Morris
Supplementary Figures - PDF file 1385K, File contains Supplementary figures of resistant cell lines, proliferation assay of a panel of cell lines, TdF binding assay transcriptional out and kinome selectivity
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::043d9dc9ddac3082860a77d7c7fbd235
https://doi.org/10.1158/2159-8290.22530809
https://doi.org/10.1158/2159-8290.22530809