Zobrazeno 1 - 10
of 66
pro vyhledávání: '"Legru A"'
Autor:
Legru, Alice, Batista, Fernando A., Puszko, Anna K., Bouillon, Anthony, Maurel, Manon, Martinez, Mariano, Ejjoummany, Abdelaziz, Ortega Varga, Laura, Adler, Pauline, Méchaly, Ariel, Hadjadj, Margot, Sosnowski, Piotr, Hopfgartner, Gérard, Alzari, Pedro M., Blondel, Arnaud, Haouz, Ahmed, Barale, Jean-Christophe, Hernandez, Jean-François
Publikováno v:
In European Journal of Medicinal Chemistry 5 April 2024 269
Autor:
Gavara, Laurent, Verdirosa, Federica, Sevaille, Laurent, Legru, Alice, Corsica, Giuseppina, Nauton, Lionel, Sandra Mercuri, Paola, Sannio, Filomena, De Luca, Filomena, Hadjadj, Margot, Cerboni, Giulia, Vo Hoang, Yen, Licznar-Fajardo, Patricia, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François
Publikováno v:
In Bioorganic & Medicinal Chemistry 15 October 2022 72
Autor:
Legru, Alice, Verdirosa, Federica, Hernandez, Jean-François, Tassone, Giusy, Sannio, Filomena, Benvenuti, Manuela, Conde, Pierre-Alexis, Bossis, Guillaume, Thomas, Caitlyn A., Crowder, Michael W., Dillenberger, Melissa, Becker, Katja, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean-Denis, Gavara, Laurent
Publikováno v:
In European Journal of Medicinal Chemistry 15 December 2021 226
Autor:
Gavara, Laurent, Legru, Alice, Verdirosa, Federica, Sevaille, Laurent, Nauton, Lionel, Corsica, Giuseppina, Mercuri, Paola Sandra, Sannio, Filomena, Feller, Georges, Coulon, Rémi, De Luca, Filomena, Cerboni, Giulia, Tanfoni, Silvia, Chelini, Giulia, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François
Publikováno v:
In Bioorganic Chemistry August 2021 113
Autor:
Gavara, Laurent, Sevaille, Laurent, De Luca, Filomena, Mercuri, Paola, Bebrone, Carine, Feller, Georges, Legru, Alice, Cerboni, Giulia, Tanfoni, Silvia, Baud, Damien, Cutolo, Giuliano, Bestgen, Benoît, Chelini, Giulia, Verdirosa, Federica, Sannio, Filomena, Pozzi, Cecilia, Benvenuti, Manuela, Kwapien, Karolina, Fischer, Marina, Becker, Katja, Frère, Jean-Marie, Mangani, Stefano, Gresh, Nohad, Berthomieu, Dorothée, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François
Publikováno v:
In European Journal of Medicinal Chemistry 15 December 2020 208
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Autor:
Laurent Gavara, Federica Verdirosa, Alice Legru, Paola Sandra Mercuri, Lionel Nauton, Laurent Sevaille, Georges Feller, Dorothée Berthomieu, Filomena Sannio, Francesca Marcoccia, Silvia Tanfoni, Filomena De Luca, Nohad Gresh, Moreno Galleni, Jean-Denis Docquier, Jean-François Hernandez
Publikováno v:
Biomolecules, Vol 10, Iss 8, p 1094 (2020)
To fight the increasingly worrying bacterial resistance to antibiotics, the discovery and development of new therapeutics is urgently needed. Here, we report on a new series of 1,2,4-triazole-3-thione compounds as inhibitors of metallo-β-lactamases
Externí odkaz:
https://doaj.org/article/0aebee0858594dab86b9fe9f6ecfb2af
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Autor:
Alice Legru, Federica Verdirosa, Yen Vo-Hoang, Giusy Tassone, Filippo Vascon, Caitlyn A. Thomas, Filomena Sannio, Giuseppina Corsica, Manuela Benvenuti, Georges Feller, Rémi Coulon, Francesca Marcoccia, Savannah Rowane Devente, Ezeddine Bouajila, Catherine Piveteau, Florence Leroux, Rebecca Deprez-Poulain, Benoît Deprez, Patricia Licznar-Fajardo, Michael W. Crowder, Laura Cendron, Cecilia Pozzi, Stefano Mangani, Jean-Denis Docquier, Jean-François Hernandez, Laurent Gavara
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, 2022, 65 (24), pp.16392-16419. ⟨10.1021/acs.jmedchem.2c01257⟩
Journal of Medicinal Chemistry, 2022, 65 (24), pp.16392-16419. ⟨10.1021/acs.jmedchem.2c01257⟩
International audience; Metallo-β-lactamases (MBLs) contribute to the resistance of Gram-negative bacteria to carbapenems, last-resort antibiotics at hospital, and MBL inhibitors are urgently needed to preserve these important antibacterial drugs. H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0a12a2619992adab250d34ee8e40f7d5
https://hdl.handle.net/11577/3465209
https://hdl.handle.net/11577/3465209
Autor:
Laurent, Gavara, Federica, Verdirosa, Laurent, Sevaille, Alice, Legru, Giuseppina, Corsica, Lionel, Nauton, Paola, Sandra Mercuri, Filomena, Sannio, Filomena, De Luca, Margot, Hadjadj, Giulia, Cerboni, Yen, Vo Hoang, Patricia, Licznar-Fajardo, Moreno, Galleni, Jean-Denis, Docquier, Jean-François, Hernandez
Publikováno v:
Bioorganic and Medicinal Chemistry
Bioorganic and Medicinal Chemistry, 2022, 72, pp.116964. ⟨10.1016/j.bmc.2022.116964⟩
Bioorganic and Medicinal Chemistry, 2022, 72, pp.116964. ⟨10.1016/j.bmc.2022.116964⟩
International audience; Metallo-β-lactamases (MBLs) represent an increasingly serious threat to public health because of their increased prevalence worldwide in relevant opportunistic Gram-negative pathogens. MBLs efficiently inactivate widely used
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a2ccc5a7fb5d5ee9e7946fc5eee59ccb
https://hal.science/hal-03767295/file/GavaraL_Manuscript.pdf
https://hal.science/hal-03767295/file/GavaraL_Manuscript.pdf