Zobrazeno 1 - 10
of 948
pro vyhledávání: '"Ladds, G."'
Autor:
de Vries T; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., Labruijere S; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., Rivera-Mancilla E; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., Garrelds IM; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., de Vries R; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., Schutter D; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., van den Bogaerdt A; Heart Valve Department, ETB-BISLIFE, Beverwijk, The Netherlands., Poyner DR; School of Life and Health Sciences, Aston University, Aston Triangle, Birmingham, UK., Ladds G; Department of Pharmacology, University of Cambridge, Cambridge, UK., Danser AHJ; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands., MaassenVanDenBrink A; Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, Rotterdam, The Netherlands.
Publikováno v:
British journal of pharmacology [Br J Pharmacol] 2024 Aug; Vol. 181 (15), pp. 2478-2491. Date of Electronic Publication: 2024 Apr 07.
Autor:
Malcharek MA; M Malcharek, Pharmacology, University of Cambridge, Cambridge, United Kingdom of Great Britain and Northern Ireland., Pearce A; A Pearce, Pharmacology, University of Cambridge, Cambridge, United Kingdom of Great Britain and Northern Ireland., Brighton CA; C Brighton, Research and Early Development, Cardiovascular, Renal and Metabolism (CVRM), BioPharmaceuticals RandD, AstraZeneca UK Limited, Cambridge, United Kingdom of Great Britain and Northern Ireland., Hornigold DC; D Hornigold, Research and Early Development, Cardiovascular, Renal and Metabolism (CVRM), BioPharmaceuticals RandD, AstraZeneca UK Limited, Cambridge, United Kingdom of Great Britain and Northern Ireland., Ladds G; G Ladds, Pharmacology, University of Cambridge, Cambridge, United Kingdom of Great Britain and Northern Ireland.
Publikováno v:
Journal of molecular endocrinology [J Mol Endocrinol] 2024 Sep 01. Date of Electronic Publication: 2024 Sep 01.
Autor:
Huang X; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge CB2 1PD, U.K., Chorianopoulou A; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Kalkounou P; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Georgiou M; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Pousias A; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Davies A; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge CB2 1PD, U.K., Pearce A; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge CB2 1PD, U.K., Harris M; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge CB2 1PD, U.K., Lambrinidis G; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Marakos P; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Pouli N; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Kolocouris A; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Lougiakis N; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou 15771, Athens, Greece., Ladds G; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge CB2 1PD, U.K.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2024 Aug 08; Vol. 67 (15), pp. 13117-13146. Date of Electronic Publication: 2024 Jul 29.
Autor:
Gandasi NR; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden.; Cell Metabolism Lab (GA-08), Department of Developmental Biology and Genetics, Indian Institute of Science, Bangalore, India., Gao R; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Kothegala L; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden., Pearce A; Department of Pharmacology, University of Cambridge, Cambridge, UK., Santos C; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden., Acreman S; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden.; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Basco D; Center for Integrative Genomics, University of Lausanne, Lausanne, Switzerland., Benrick A; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden., Chibalina MV; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Clark A; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Guida C; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Harris M; Department of Pharmacology, University of Cambridge, Cambridge, UK., Johnson PRV; Nuffield Department of Surgical Sciences, John Radcliffe Hospital, Oxford, UK.; Biomedical Research Centre, Oxford National Institute for Health Research, Churchill Hospital, Oxford, UK., Knudsen JG; Section for Cell Biology and Physiology, Department of Biology, University of Copenhagen, Copenhagen, Denmark., Ma J; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Miranda C; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden.; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Shigeto M; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Tarasov AI; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK.; School of Biomedical Sciences, University of Ulster, Coleraine, Northern Ireland, UK., Yeung HY; Department of Pharmacology, University of Cambridge, Cambridge, UK., Thorens B; Center for Integrative Genomics, University of Lausanne, Lausanne, Switzerland., Asterholm IW; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden., Zhang Q; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Ramracheya R; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK., Ladds G; Department of Pharmacology, University of Cambridge, Cambridge, UK., Rorsman P; Metabolic Physiology Unit, Department of Physiology, Institute of Neuroscience and Physiology, Sahlgrenska Academy, Gothenburg, Sweden. patrik.rorsman@drl.ox.ac.uk.; Oxford Centre for Diabetes, Endocrinology and Metabolism, University of Oxford, Churchill Hospital, Oxford, UK. patrik.rorsman@drl.ox.ac.uk.; Biomedical Research Centre, Oxford National Institute for Health Research, Churchill Hospital, Oxford, UK. patrik.rorsman@drl.ox.ac.uk.; School of Biomedical Sciences, University of Ulster, Coleraine, Northern Ireland, UK. patrik.rorsman@drl.ox.ac.uk.
Publikováno v:
Diabetologia [Diabetologia] 2024 Mar; Vol. 67 (3), pp. 528-546. Date of Electronic Publication: 2023 Dec 21.
Autor:
Jones AJY; Department of Biochemistry, University of Cambridge, 80 Tennis Court Road, Cambridge, CB2 1GA, UK., Harman TH; Department of Biochemistry, University of Cambridge, 80 Tennis Court Road, Cambridge, CB2 1GA, UK., Harris M; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge, CB2 1PD, UK., Lewis OE; Department of Biochemistry, University of Cambridge, 80 Tennis Court Road, Cambridge, CB2 1GA, UK., Ladds G; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge, CB2 1PD, UK., Nietlispach D; Department of Biochemistry, University of Cambridge, 80 Tennis Court Road, Cambridge, CB2 1GA, UK. dn206@cam.ac.uk.
Publikováno v:
Nature communications [Nat Commun] 2024 Feb 13; Vol. 15 (1), pp. 1334. Date of Electronic Publication: 2024 Feb 13.
Autor:
Stampelou M; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou, 15771 Athens, Greece., Ladds G; Department of Pharmacology, University of Cambridge, Tennis Court Road, Cambridge CB2 1PD, U.K., Kolocouris A; Laboratory of Medicinal Chemistry, Section of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou, 15771 Athens, Greece.
Publikováno v:
The journal of physical chemistry. B [J Phys Chem B] 2024 Feb 01; Vol. 128 (4), pp. 914-936. Date of Electronic Publication: 2024 Jan 18.
Autor:
Pan D; Sackler Institute of Pulmonary Pharmacology, Institute of Pharmaceutical Science, King's College London, London, UK., Ladds G; Department of Pharmacology, University of Cambridge, Cambridge, UK., Rahman KM; Chemical Biology Group, Institute of Pharmaceutical Science, King's College London, London, UK., Pitchford SC; Sackler Institute of Pulmonary Pharmacology, Institute of Pharmaceutical Science, King's College London, London, UK.
Publikováno v:
British journal of pharmacology [Br J Pharmacol] 2024 Feb; Vol. 181 (4), pp. 580-592. Date of Electronic Publication: 2023 Aug 02.
The adenosine A3 receptor (A3R) belongs to a family of four adenosine receptor (AR) subtypes which all play distinct roles throughout the body. A3R antagonists have been described as potential treatments for numerous diseases including asthma. Given
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=od______2127::121d56c430c2691df184d6ac7cf199a5
https://pergamos.lib.uoa.gr/uoa/dl/object/uoadl:3056323
https://pergamos.lib.uoa.gr/uoa/dl/object/uoadl:3056323
Publikováno v:
Journal of Theoretical Biology
Highlights • A new ordinary differential equation model for biased agonism dynamics at a G protein-coupled receptor (GPCR) is presented. • The model is general in the number of G proteins and active receptor. • Numerical simulations reveal new
Autor:
Preti B; Institute of Biochemistry and Molecular Medicine, University of Bern, Bühlstrasse 28, 3012Bern, Switzerland., Suchankova A; Department of Pharmacology, University of Cambridge, Tennis Court Road, CambridgeCB2 1PD, U.K., Deganutti G; Centre for Sport, Exercise and Life Sciences, Faculty of Health and Life Sciences, Coventry University, CoventryCV1 5FB, U.K., Leuenberger M; Institute of Biochemistry and Molecular Medicine, University of Bern, Bühlstrasse 28, 3012Bern, Switzerland., Barkan K; Department of Pharmacology, University of Cambridge, Tennis Court Road, CambridgeCB2 1PD, U.K., Manulak I; Department of Pharmacology, University of Cambridge, Tennis Court Road, CambridgeCB2 1PD, U.K., Huang X; Department of Pharmacology, University of Cambridge, Tennis Court Road, CambridgeCB2 1PD, U.K., Carvalho S; Department of Pharmacology, University of Cambridge, Tennis Court Road, CambridgeCB2 1PD, U.K., Ladds G; Department of Pharmacology, University of Cambridge, Tennis Court Road, CambridgeCB2 1PD, U.K., Lochner M; Institute of Biochemistry and Molecular Medicine, University of Bern, Bühlstrasse 28, 3012Bern, Switzerland.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2022 Nov 10; Vol. 65 (21), pp. 14864-14890. Date of Electronic Publication: 2022 Oct 21.