Structure-activity relationship around PI-2620 highlights the importance of the nitrogen atom position in the tricyclic core

Autor: Kroth, Heiko, Oden, Felix, Serra, Andreia Monica, Molette, Jerome, Mueller, Andre, Berndt, Mathias, Capotosti, Francesca, Gabellieri, Emanuele, Schmitt-Willich, Heribert, Hickman, David, Pfeifer, Andrea, Dinkelborg, Ludger, Stephens, Andrew

Publikováno v: In Bioorganic & Medicinal Chemistry 15 December 2021 52

Position-Specific Trapping of Topoisomerase II by Benzo[a]pyrene Diol Epoxide Adducts: Implications for Interactions with Intercalating Anticancer Agents

Autor: Khan, Qasim A., Kohlhagen, Glenda, Marshall, Richard, Austin, Caroline A., Kalena, Govind P., Kroth, Heiko, Sayer, Jane M., Jerina, Donald M., Pommier, Yves

Publikováno v: Proceedings of the National Academy of Sciences of the United States of America, 2003 Oct . 100(21), 12498-12503.

Externí odkaz: https://www.jstor.org/stable/3147979

Position-Specific Trapping of Topoisomerase I-DNA Cleavage Complexes by Intercalated Benzo[a]-Pyrene Diol Epoxide Adducts at the 6-Amino Group of Adenine

Autor: Pommier, Yves, Laco, Gary S., Kohlhagen, Glenda, Sayer, Jane M., Kroth, Heiko, Jerina, Donald M.

Publikováno v: Proceedings of the National Academy of Sciences of the United States of America, 2000 Sep . 97(20), 10739-10744.

Externí odkaz: https://www.jstor.org/stable/123197

Discovery and preclinical characterization of [¹⁸F]PI-2620, a next-generation tau PET tracer for the assessment of tau pathology in Alzheimer's disease and other tauopathies.

Autor: Kroth, Heiko¹ (AUTHOR), Oden, Felix² (AUTHOR), Molette, Jerome¹ (AUTHOR), Schieferstein, Hanno^3,4 (AUTHOR), Capotosti, Francesca¹ (AUTHOR), Mueller, Andre² (AUTHOR), Berndt, Mathias² (AUTHOR), Schmitt-Willich, Heribert² (AUTHOR), Darmency, Vincent¹ (AUTHOR), Gabellieri, Emanuele¹ (AUTHOR), Boudou, Cédric¹ (AUTHOR), Juergens, Tanja¹ (AUTHOR), Varisco, Yvan¹ (AUTHOR), Vokali, Efthymia¹ (AUTHOR), Hickman, David T.¹ (AUTHOR), Tamagnan, Gilles^5,6 (AUTHOR), Pfeifer, Andrea¹ (AUTHOR), Dinkelborg, Ludger² (AUTHOR), Muhs, Andreas¹ (AUTHOR), Stephens, Andrew² (AUTHOR) a.stephens@life-mi.com

Publikováno v: European Journal of Nuclear Medicine & Molecular Imaging. Sep2019, Vol. 46 Issue 10, p2178-2189. 12p. 4 Diagrams, 2 Charts, 1 Graph.

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