Zobrazeno 1 - 10
of 11
pro vyhledávání: '"Kristen K. Ford"'
Autor:
Michelle R. Garnsey, Aaron C. Smith, Jana Polivkova, Autumn L. Arons, Guoyun Bai, Caroline Blakemore, Markus Boehm, Leanne M. Buzon, Sarah N. Campion, Matthew Cerny, Shiao-Chi Chang, Karen Coffman, Kathleen A. Farley, Kari R. Fonseca, Kristen K. Ford, Jeonifer Garren, Jimmy X. Kong, Martin R. M. Koos, Daniel W. Kung, Yajing Lian, Monica M. Li, Qifang Li, Luis A. Martinez-Alsina, Rebecca O’Connor, Kevin Ogilvie, Kiyoyuki Omoto, Brian Raymer, Matthew R. Reese, Tim Ryder, Lacey Samp, Kimberly A. Stevens, Daniel W. Widlicka, Qingyi Yang, Kaicheng Zhu, Jean-Philippe Fortin, Matthew F. Sammons
Publikováno v:
Journal of Medicinal Chemistry. 66:3195-3211
Autor:
David J. Matson, Daniel Broom, Michele Matchett, Robin Meade, David J. Wustrow, Marianne E. Buck, Weifeng Yu, Synthia H. Sun, Jun Yuan, Elizabeth Bradshaw, Susan Coombs, Kristen K. Ford, James E. Krause, Daniel N. Cortright, Ricardo Ochoa
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 327(3)
Recent evidence suggests that the P2X(7) receptor may play a role in the pathophysiology of preclinical models of pain and inflammation. Therefore, pharmacological agents that target this receptor may potentially have clinical utility as anti-inflamm
Publikováno v:
Molecular biology reports. 32(2)
Under conditions of genomic stress, the Mdm locus in human and in mouse is prone to instability manifested as amplification and oncogenesis. The Mdm2 gene is a known oncogene that is amplified in approximately one-third of sarcomas and whose protein
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 315(1)
P2X3 purinergic receptors are predominantly expressed in dorsal root ganglion (DRG) neurons and play an important role in pain sensation. P2X3-specific antagonists are currently being sought to ameliorate pain in several indications. Understanding ho
Publikováno v:
Molecular Biology Reports; Jun2005, Vol. 32 Issue 2, p95-101, 7p
Autor:
Dow RL; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Ammirati M; Pfizer Worldwide Research & Development , Groton , Connecticut 06340 , United States., Bagley SW; Pfizer Worldwide Research & Development , Groton , Connecticut 06340 , United States., Bhattacharya SK; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Buckbinder L; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Cortes C; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., El-Kattan AF; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Ford K; Pfizer Worldwide Research & Development , Groton , Connecticut 06340 , United States., Freeman GB; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Guimarães CRW; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Liu S; Pfizer Worldwide Research & Development , Groton , Connecticut 06340 , United States., Niosi M; Pfizer Worldwide Research & Development , Groton , Connecticut 06340 , United States., Skoura A; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States., Tess D; Pfizer Worldwide Research & Development , Cambridge , Massachusetts 02139 , United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2018 Apr 12; Vol. 61 (7), pp. 3114-3125. Date of Electronic Publication: 2018 Apr 03.
Autor:
Kung DW; Worldwide Medicinal Chemistry, Groton, CT 06340, United States. Electronic address: daniel.w.kung@pfizer.com., Griffith DA; Worldwide Medicinal Chemistry, Cambridge, MA 02139, United States. Electronic address: david.a.griffith@pfizer.com., Esler WP; Cardiovascular, Metabolic and Endocrine Diseases Research Unit, Cambridge, MA 02139, United States., Vajdos FF; Structural Biology, Groton, CT 06340, United States., Mathiowetz AM; Worldwide Medicinal Chemistry, Cambridge, MA 02139, United States., Doran SD; Pharmacokinetics, Dynamics and Metabolism, Groton, CT 06340, United States., Amor PA; Cardiovascular, Metabolic and Endocrine Diseases Research Unit, Cambridge, MA 02139, United States., Bagley SW; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Banks T; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Cabral S; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Ford K; Primary Pharmacology Group, Groton, CT 06340, United States., Garcia-Irizarry CN; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Landis MS; Pharmaceutical Sciences Research Formulations, Pfizer Worldwide Research and Development, Cambridge, MA 02139, United States., Loomis K; Cardiovascular, Metabolic and Endocrine Diseases Research Unit, Groton, CT 06340, United States., McPherson K; Cardiovascular, Metabolic and Endocrine Diseases Research Unit, Groton, CT 06340, United States., Niosi M; Pharmacokinetics, Dynamics and Metabolism, Groton, CT 06340, United States., Rockwell KL; Primary Pharmacology Group, Groton, CT 06340, United States., Rose C; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Smith AC; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Southers JA; Worldwide Medicinal Chemistry, Groton, CT 06340, United States., Tapley S; Cardiovascular, Metabolic and Endocrine Diseases Research Unit, Groton, CT 06340, United States., Tu M; Worldwide Medicinal Chemistry, Cambridge, MA 02139, United States., Valentine JJ; Primary Pharmacology Group, Groton, CT 06340, United States.
Publikováno v:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2015 Nov 15; Vol. 25 (22), pp. 5352-6. Date of Electronic Publication: 2015 Sep 15.
Autor:
Ammirati M; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Bagley SW; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Bhattacharya SK; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Buckbinder L; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Carlo AA; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Conrad R; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Cortes C; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Dow RL; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Dowling MS; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., El-Kattan A; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Ford K; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Guimarães CR; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Hepworth D; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Jiao W; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., LaPerle J; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Liu S; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Londregan A; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Loria PM; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Mathiowetz AM; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Munchhof M; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Orr ST; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Petersen DN; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Price DA; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Skoura A; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Smith AC; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Wang J; Worldwide Medicinal Chemistry, Cardiovascular and Metabolic Research Unit, External Research Solutions, Primary Pharmacology Group, and Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States.
Publikováno v:
ACS medicinal chemistry letters [ACS Med Chem Lett] 2015 Oct 06; Vol. 6 (11), pp. 1128-33. Date of Electronic Publication: 2015 Oct 06 (Print Publication: 2015).
Autor:
Osuch E; Department of Psychiatry, Schulich School of Medicine and Dentistry, University of Western Ontario, London, ON, Canada N6A 4G5; Department of Medical Biophysics, University of Western Ontario, London, ON, Canada. Electronic address: Elizabeth.osuch@lhsc.on.ca., Ford K; Department of Psychiatry, Schulich School of Medicine and Dentistry, University of Western Ontario, London, ON, Canada N6A 4G5., Wrath A; Department of Psychiatry, Schulich School of Medicine and Dentistry, University of Western Ontario, London, ON, Canada N6A 4G5., Bartha R; Department of Medical Biophysics, University of Western Ontario, London, ON, Canada., Neufeld R; Department of Psychiatry, Schulich School of Medicine and Dentistry, University of Western Ontario, London, ON, Canada N6A 4G5; Department of Psychology, University of Western Ontario, London, ON, Canada; Program in Neuroscience, University of Western Ontario, London, ON, Canada.
Publikováno v:
Psychiatry research [Psychiatry Res] 2014 Aug 30; Vol. 223 (2), pp. 104-12. Date of Electronic Publication: 2014 May 14.
Autor:
Khan SA; Department of Psychology, The University of Western Ontario, Social Science Centre, London, Ontario, N6A 5C2, Canada., Ford K, Timney B, Everling S
Publikováno v:
Experimental brain research [Exp Brain Res] 2003 May; Vol. 150 (1), pp. 68-74. Date of Electronic Publication: 2003 Mar 04.