Zobrazeno 1 - 10
of 20
pro vyhledávání: '"Krishna S. Ethiraj"'
Autor:
Rajesh Madhu, Yogeeswari Perumal, Krishna S. Ethiraj, Mallilkarjuna Reddy Guda, Rajkumar Veligeti, Naveen Polkam, Vijaya Kumar Reddy Avula, Sivaprasad Kasturi, Hasitha Shilpa Anantaraju, Grigory V. Zyryanov, Swetha Vallela, Visweswara Rao Pasupuleti, Jaya Shree Anireddy, Srinivas Uppalanchi
Publikováno v:
Scientific Reports, Vol 10, Iss 1, Pp 1-22 (2020)
Sci. Rep.
Scientific Reports
Sci. Rep.
Scientific Reports
Acridone based synthetic and natural products with inherent anticancer activity advancing the research and generating a large number of structurally diversified compounds. In this sequence we have designed, synthesized a series of tetracyclic acridon
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d76c07b6705f38e40b4277f9a25eb08d
https://doi.org/10.1038/s41598-020-77590-1
https://doi.org/10.1038/s41598-020-77590-1
Autor:
Dilep Kumar Sigalapalli, Sujatha Surarapu, Jaya Shree Anireddy, Krishna S. Ethiraj, Srinivas Uppalanchi, Perumal Yogeeswari, Shubham Dwivedi, Siva Prasad Kasturi, Nagendra Babu Bathini
Publikováno v:
European Journal of Medicinal Chemistry. 150:39-52
Biological evaluation of 3,4-dihydroxy piperidines as α-glucosidase inhibitors is being reported for the first time. Forty-five derivatives (amides, di-amides and sulfonamides) were made using cis and trans 3,4-dihydroxy piperidines to evaluate thei
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c41779a1626fc5548072433721c8fce1
https://doi.org/10.1016/j.ejmech.2018.02.072
https://doi.org/10.1016/j.ejmech.2018.02.072
Autor:
Shubham Dwivedi, Perumal Yogeeswari, Srinivas Uppalanchi, Jaya Shree Anireddy, Sivaprasad Kasturi, Hasitha Shilpa Anantaraju, Sujatha Surarapu, Krishna S. Ethiraj
Publikováno v:
Letters in Drug Design & Discovery. 15:181-192
Background: In the present study, new triazine derivatives 3, 4, 5, 6, 8 and 10 were synthesized starting from readily available cyanuric chloride 1 via nucleophilic displacement with morpholine followed by Suzuki or Stille coupling reactions and the
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::00f242338db751ff06dab4eb1fef4995
https://doi.org/10.2174/1570180814666170605115335
https://doi.org/10.2174/1570180814666170605115335
Autor:
Sujatha Surarapu, Dilep Kumar Sigalapalli, Shubham Dwivedi, Krishna S. Ethiraj, Yogeeswari Perumal, Hasitha Shilpa Anantaraju, Srinivas Uppalanchi, Sivaprasad Kasturi, Jaya Shree Anireddy, Bathini Nagendra Babu
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 27:2818-2823
A new series of Deacetylsarmentamide A and B derivatives, amides and sulfonamides of 3,4-dihydroxypyrrolidines as α-glucosidase inhibitors were designed and synthesized. The biological screening test against α-glucosidase showed that some of these
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::beef29f0ccc5c589f85dfece1d0dbf5a
https://doi.org/10.1016/j.bmcl.2017.04.078
https://doi.org/10.1016/j.bmcl.2017.04.078
Autor:
Dilep Kumar Sigalapalli, Yogeeswari Perumal, Shubham Dwivedi, Jaya Shree Anireddy, Krishna S. Ethiraj, Srinivas Uppalanchi, Sujatha Surarapu, Bathini Nagendra Babu, Sivaprasad Kasturi, Chandra Chary Bathoju
An efficient acid catalyzed methodology has been employed to synthesize a variety of aza-flavanones and their α-glucosidase inhibitory activity is evaluated using acarbose, miglitol and voglibose as reference standards. Molecular modeling studies we
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::96db4bda49a5dd49262416e727d7aa9f
https://europepmc.org/articles/PMC6072087/
https://europepmc.org/articles/PMC6072087/
Publikováno v:
Synthetic Communications. 37:2337-2343
A facile, mild, and efficient methodology for the ionic Diels–Alder reaction of acetals of α,β‐unsaturated ketones and aldehydes as dienophiles with various 1,3‐dienes employing MgBr2 as the Lewis acid catalyst to furnish corresponding Diels
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f1740b6ac30eeb51050685187ce44c76
https://doi.org/10.1080/00397910701410814
https://doi.org/10.1080/00397910701410814
Publikováno v:
Mini-Reviews in Medicinal Chemistry. 3:305-313
This Review contains our recent studies on evaluation of biological activities associated with monocyclic β-lactams and bicyclic β-lactam antibiotics containing various heteroatoms. A series of bicyclic β-lactams was synthesized, which possessed e
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a6a48a0941adff07e6173a71347061a5
https://doi.org/10.2174/1389557033488132
https://doi.org/10.2174/1389557033488132
Autor:
Subhash P. Chavan, Krishna S. Ethiraj
Publikováno v:
Tetrahedron Letters. 36:2281-2284
Facile intramolecular cyclisation of activated tethered dienes mediated by magnesium in methanol at room temperature is described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::baee861cc033b2d637fa4493b28cddea
https://doi.org/10.1016/0040-4039(95)00190-n
https://doi.org/10.1016/0040-4039(95)00190-n
Publikováno v:
Synlett. 2001:0857-0859
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::df5dd1de686b86d25c49415ccfa536a2
https://doi.org/10.1055/s-2001-14613
https://doi.org/10.1055/s-2001-14613
Publikováno v:
ChemInform. 28
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4d1d9433ce059c0c9ddd357e58293d58
https://doi.org/10.1002/chin.199706091
https://doi.org/10.1002/chin.199706091