Zobrazeno 1 - 10 of 159 pro vyhledávání: '"Krámos B"'
1
Akademický článek
Ligand Binding and Functional Effect of Novel Bicyclic α5 GABA A Receptor Negative Allosteric Modulators.
Autor: Krámos B; Spectroscopic Research Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary., Béni Z; Spectroscopic Research Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary., Túrós GI; Medicinal Chemistry Laboratory II, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary., Éliás O; Medicinal Chemistry Laboratory II, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary., Potor A; Medicinal Chemistry Laboratory II, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary., Kapus GL; Proprietary R&D Coordination Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary., Szabó G; Medicinal Chemistry Laboratory II, Gedeon Richter Plc., Gyömrői út 19-21, Budapest 1103, Hungary.
Publikováno v: Journal of chemical information and modeling [J Chem Inf Model] 2024 Dec 17. Date of Electronic Publication: 2024 Dec 17.
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2
Akademický článek
Development of dual V1a/V2 antagonists containing triazolobenzazepine scaffold.
Autor: Varró G; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary. Electronic address: varrog@gedeonrichter.com., Bozó É; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Vukics K; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Baska F; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Szántó G; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Krámos B; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Domány-Kovács K; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Kordás KS; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Vastag M; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Magdó I; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Bata I; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary.
Publikováno v: European journal of medicinal chemistry [Eur J Med Chem] 2024 Nov 28; Vol. 283, pp. 117069. Date of Electronic Publication: 2024 Nov 28.
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3
Akademický článek
Novel-Type GABA B PAMs: Structure-Activity Relationship in Light of the Protein Structure.
Autor: Krámos B; Spectroscopic Research Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Hadady Z; Chemistry Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Makó A; Chemistry Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Szántó G; Chemistry Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Felföldi N; Chemistry Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Magdó I; Spectroscopic Research Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Bobok AÁ; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Bata I; Chemistry Department, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Román V; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Visegrády A; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Keserű GM; Medicinal Chemistry Research Group, Research Centre for Natural Sciences, Magyar tudósok krt. 2, Budapest, 1117 Hungary., Greiner I; Research and Development Director, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary., Éles J; Head of Medicinal Chemistry, Gedeon Richter Plc., Gyömrői út 19-21, Budapest, 1103 Hungary.
Publikováno v: ACS medicinal chemistry letters [ACS Med Chem Lett] 2024 Mar 01; Vol. 15 (3), pp. 396-405. Date of Electronic Publication: 2024 Mar 01 (Print Publication: 2024).
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4
Akademický článek
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5
Akademický článek
Optimization of Novel α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulators and the Discovery of a Preclinical Development Candidate Molecule (RGH-560).
Autor: Ledneczki I; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Némethy Z; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Molnár KD; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Tapolcsányi P; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Ilkei V; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Vágó I; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Kolok S; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Thán M; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Laszy J; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Balázs O; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Krámos B; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Szigetvári Á; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Bata I; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Makó A; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Visegrády A; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Fodor L; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Vastag M; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Lévay G; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Lendvai B; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Greiner I; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary., Éles J; Gedeon Richter Plc, 19-21 Gyömői útca, Budapest H-1103, Hungary.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2023 Dec 14; Vol. 66 (23), pp. 16276-16302. Date of Electronic Publication: 2023 Nov 21.
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6
Akademický článek
Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM.
Autor: Károlyi BI; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary. Electronic address: karolyibi@richter.hu., Potor A; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Kapus GL; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Fodor L; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Bobok A; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Krámos B; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Magdó I; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Bata I; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary., Szabó G; Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary.
Publikováno v: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2023 Jan 15; Vol. 80, pp. 129107. Date of Electronic Publication: 2022 Dec 19.
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7
Akademický článek
Potential Mechanisms for Why Not All Antipsychotics Are Able to Occupy Dopamine D 3 Receptors in the Brain in vivo .
Autor: Kiss B; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Krámos B; Spectroscopic Research Department, Gedeon Richter Plc., Budapest, Hungary., Laszlovszky I; Global Medical Division, Gedeon Richter Plc., Budapest, Hungary.
Publikováno v: Frontiers in psychiatry [Front Psychiatry] 2022 Mar 24; Vol. 13, pp. 785592. Date of Electronic Publication: 2022 Mar 24 (Print Publication: 2022).
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8
Akademický článek
HTS-based discovery and optimization of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor.
Autor: Ledneczki I; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary. Electronic address: ledneczki@richter.hu., Horváth A; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary., Tapolcsányi P; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary., Éles J; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary., Molnár KD; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary., Vágó I; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary., Visegrády A; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Kiss L; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Szigetvári Á; Spectroscopic Research Department, Gedeon Richter Plc., Budapest, Hungary., Kóti J; Spectroscopic Research Department, Gedeon Richter Plc., Budapest, Hungary., Krámos B; Spectroscopic Research Department, Gedeon Richter Plc., Budapest, Hungary., Mahó S; Department of Chemistry, Gedeon Richter Plc., Budapest, Hungary., Holm P; Orion Corporation, Turku, Finland., Kolok S; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Fodor L; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Thán M; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Kostyalik D; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Balázs O; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Vastag M; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Greiner I; Research Management, Gedeon Richter Plc., Budapest, Hungary., Lévay G; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Lendvai B; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary., Némethy Z; Pharmacological and Drug Safety Research, Gedeon Richter Plc., Budapest, Hungary.
Publikováno v: European journal of medicinal chemistry [Eur J Med Chem] 2021 Oct 15; Vol. 222, pp. 113560. Date of Electronic Publication: 2021 May 29.
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9
Akademický článek
Synthesis and Characterization of New V 1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers.
Autor: Szeleczky Z; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Szakács Z; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Bozó É; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Baska F; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Vukics K; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Lévai S; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Temesvári K; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Vass E; Institute of Chemistry, Eötvös Loránd University, Pázmány Péter sétány 1/A, Budapest H-1117, Hungary., Béni Z; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Krámos B; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Magdó I; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Szántay C Jr; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Kóti J; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Domány-Kovács K; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Greiner I; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary., Bata I; Gedeon Richter Plc., 19-21 Gyömrői út, Budapest 1103, Hungary.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2021 Jul 22; Vol. 64 (14), pp. 10445-10468. Date of Electronic Publication: 2021 Jul 13.
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10
Akademický článek
Blockade of dopamine D3 receptors improves hippocampal synaptic function and rescues age‐related cognitive phenotype.
Autor: Tropea, Maria Rosaria1 (AUTHOR), Melone, Marcello2,3 (AUTHOR), Li Puma, Domenica Donatella4,5 (AUTHOR), Vacanti, Valeria1 (AUTHOR), Aceto, Giuseppe4,5 (AUTHOR), Bandiera, Bruno4 (AUTHOR), Trovato, Roberta Carmela1 (AUTHOR), Torrisi, Sebastiano Alfio1 (AUTHOR), Leggio, Gian Marco1 (AUTHOR), Palmeri, Agostino1 (AUTHOR), D'Ascenzo, Marcello4,5 (AUTHOR), Conti, Fiorenzo2,3 (AUTHOR), Grassi, Claudio4,5 (AUTHOR), Puzzo, Daniela1,6 (AUTHOR) danypuzzo@yahoo.it
Publikováno v: Aging Cell. Nov2024, Vol. 23 Issue 11, p1-16. 16p.
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