Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Konghua Jing"'
Autor:
Chulho Choi, Anthony A. Carlo, Ciarán N. Cronin, Konghua Jing, Daniel W. Kung, Jianhua Liu, Vincent M. Lombardo, Abigail R. Turco, Juxing Yin, Aijia Yu, Stephen W. Wright
Publikováno v:
ACS Medicinal Chemistry Letters. 13:250-256
Autor:
Chulho, Choi, Anthony A, Carlo, Ciarán N, Cronin, Konghua, Jing, Daniel W, Kung, Jianhua, Liu, Vincent M, Lombardo, Abigail R, Turco, Juxing, Yin, Aijia, Yu, Stephen W, Wright
Publikováno v:
ACS Med Chem Lett
[Image: see text] The metabolic oxidation of drug-like small molecules by aldehyde oxidase (AO) has commonly been mitigated through the incorporation of deuterium at the oxidation site. We report that dimethylformamide dimethyl acetal and related com
Autor:
W. Lynn Rogers, Brian F. Mcguinness, Kurt W. Saionz, Steven G. Kultgen, Vikash Srivastava, Hema Desai, Hao Yan, Tara M. Stauffer, Samiran Saha, Koc-Kan Ho, Shengting Zhang, Neelima Mannava, Yan Jiang, Anthony E. Klon, Tailong Li, Juxing Yin, Weiqing Chen, Konghua Jing, Maria L. Webb, Kanak Kanti Majumdar, Laura L. Rokosz
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 20:7414-7420
A novel series of quinolinone-based adenosine A2B receptor antagonists was identified via high throughput screening of an encoded combinatorial compound collection. Synthesis and assay of a series of analogs highlighted essential structural features