Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Kikuko Kamisaka"'
Autor:
Chiduru Watanabe, Shigenori Tanaka, Yoshio Okiyama, Hitomi Yuki, Tatsuya Ohyama, Kikuko Kamisaka, Daisuke Takaya, Kaori Fukuzawa, Teruki Honma
Publikováno v:
The Journal of Physical Chemistry Letters. 14:3609-3620
Autor:
Chiduru Watanabe, Shigenori Tanaka, Yoshio Okiyama, Hitomi Yuki, Tatsuya Ohyama, Kikuko Kamisaka, Daisuke Takaya, Kaori Fukuzawa, Teruki Honma
A non-covalent oral drug targeting severe acute respiratory syndrome-coronavirus-2 (SARS-CoV-2) main protease (Mpro), ensitrelvir (brand name Xocova), has been developed by Unoh et al. (J. Med. Chem. 2022, 65, 9, 6499–6512) using structure-based dr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1092026b76b6be8c6f7183c157da27a3
https://doi.org/10.26434/chemrxiv-2022-drwc0
https://doi.org/10.26434/chemrxiv-2022-drwc0
Autor:
Shunpei Nagase, Hitomi Yuki, Noriyuki Kurita, Teruki Honma, Shigenori Tanaka, Daisuke Takaya, Kikuko Kamisaka, Yoshio Okiyama, Midori Takimoto-Kamimura, Hirotomo Moriwaki, Yoichiro Yagi, Tatsuya Takagi, Norihito Kawashita, Kenichiro Takaba, Tomohiro Sato, Tomonaga Ozawa, Chiduru Watanabe, Kaori Fukuzawa
Publikováno v:
Journal of Chemical Information and Modeling. 61:777-794
We developed the world's first web-based public database for the storage, management, and sharing of fragment molecular orbital (FMO) calculation data sets describing the complex interactions between biomacromolecules, named FMO Database (https://dru
Autor:
Nobuo Cho, Ko Kikuzato, Yushi Futamura, Takeshi Shimizu, Hiroki Hayase, Kikuko Kamisaka, Daisuke Takaya, Hitomi Yuki, Teruki Honma, Mamoru Niikura, Fumie Kobayashi, Nobumoto Watanabe, Hiroyuki Osada, Hiroo Koyama
Publikováno v:
Bioorganicmedicinal chemistry. 66
The identification, structure-activity relationships (SARs), and biological effects of new antimalarials consisting of a 2,3,4,9-tetrahydro-1H-β-carboline core, a coumarin ring, and an oxyalkanoyl linker are described. A cell-based phenotypic approa
Autor:
Kaori Fukuzawa, Atsushi Tokuhisa, Mitsunori Ikeguchi, Masuda Tomohide, Koichiro Kato, Satoshi Ono, Shumpei Nagase, Hiroshi Ueda, Kanji Oshima, Ryo Kanada, Masateru Ohta, Kikuko Kamisaka, Yasushi Okuno, Naoki Miyagawa, Teruki Honma, Hideo Mizouchi, Chiduru Watanabe
Publikováno v:
Journal of Chemical Information and Modeling. 60:3361-3368
Here, we have constructed neural network-based models that predict atomic partial charges with high accuracy at low computational cost. The models were trained using high-quality data acquired from quantum mechanics calculations using the fragment mo
Autor:
Kikuko Kamisaka, Tatsuya Ohyama, Chiduru Watanabe, Yuma Handa, Daisuke Takaya, Kaori Fukuzawa, Yusuke Kawashima, Koichiro Kato, Kazuki Watanabe, Ami Yamamoto, Teruki Honma
SARS-CoV-2 is the causative agent of coronavirus, globally known as COVID-19. There are ongoing researches to develop effective therapeutics and vaccines against COVID-19 using various methods. We currently conduct research based on the fragment mole
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::559c50451cf2575dc840236eaf084f1c
https://doi.org/10.33774/chemrxiv-2021-njqc8
https://doi.org/10.33774/chemrxiv-2021-njqc8
Publikováno v:
AINA (1)
Since IP-SAN allows us to reduce initial costs and management costs of storage by using IP networks, iSCSI, common protocol in IP-SAN, is becoming more important. Although one of the key issues for iSCSI is a security measure to access remote storage