Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Khammungkhune, Sak"'
Autor:
Adam Kois, Bernd Stein, Graciella Shevlin, May S Kung Sutherland, Steve Pierce, Shripad S. Bhagwat, Stephanie Lipps, Helen Brady, Leah M. Gayo-Fung, Matt Hickman, Mary Doubleday, David W. Anderson, Normand Richard, Khammungkhune Sak
Publikováno v:
Molecular Pharmacology. 61:562-568
We determined the differential response of a novel SERM, SP500263, on estrogen receptor (ER) alpha and the more recently cloned ER-beta. Because of the high homology of amino acid residues in the ligand-binding domain of ER-alpha and ER-beta, we were
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::31dffcef6a200a5684a7214a17de7d53
https://doi.org/10.1124/mol.61.3.562
https://doi.org/10.1124/mol.61.3.562
Autor:
Adam Kois, Normand Richard, Khammungkhune Sak, Graziella I. Shevlin, Shripad S. Bhagwat, John Sapienza, Helen Brady, Mathew Hickman, Jalluri Ravi Kumar, Deborah Mortensen, Gayo Leah M, Jeffrey A. Mckie, Mary Doubleday, May S Kung Sutherland, Bernd Stein
Publikováno v:
Bioorganicmedicinal chemistry letters. 14(13)
Starting from a phenol screening hit (6), three series of benzopyranone selective estrogen receptor modulators (SERMs) have been designed, synthesized, and analyzed for both estrogen receptor alpha binding affinity and in vitro activity in two cell a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5671bfae4e2deb683ad3fb739f4caaed
https://pubmed.ncbi.nlm.nih.gov/15177442
https://pubmed.ncbi.nlm.nih.gov/15177442
Autor:
McKie, Jeffrey A., Bhagwat, Shripad S., Brady, Helen, Doubleday, Mary, Gayo, Leah, Hickman, Mathew, Jalluri, Ravi K., Khammungkhune, Sak, Kois, Adam, Mortensen, Deborah, Richard, Normand, Sapienza, John, Shevlin, Graziella, Stein, Bernd, Sutherland, May
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 2004 14(13):3407-3410