Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Kephart SE"'
Autor:
Meador J rd, Clifford E. Ford, Edward L. Brown, Chan F, Johnson T, Reich Siegfried Heinz, Kephart Se, Rose Ann Ferre, D. M. Delisle, David A. Matthews, Susan L. Binford, Shella A. Fuhrman, Amy K. Patick, Thomas F. Hendrickson, Stephen T. Worland, Wallace Michael B
Publikováno v:
Journal of Medicinal Chemistry. 43:1670-1683
A series of nonpeptide benzamide-containing inhibitors of human rhinovirus (HRV) 3C protease was identified using structure-based design. The design, synthesis, and biological evaluation of these inhibitors are reported. A Michael acceptor was combin
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Autor:
Jensen-Pergakes K; Oncology Research Division, Pfizer Inc.; San Diego, California., Tatlock J; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Maegley KA; Oncology Research Division, Pfizer Inc.; San Diego, California., McAlpine IJ; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., McTigue M; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Xie T; Oncology Research Division, Pfizer Inc.; San Diego, California., Dillon CP; Oncology Research Division, Pfizer Inc.; San Diego, California., Wang Y; Oncology Research Division, Pfizer Inc.; San Diego, California., Yamazaki S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Inc., San Diego, California., Spiegel N; Oncology Research Division, Pfizer Inc.; San Diego, California., Shi M; Oncology Research Division, Pfizer Inc.; San Diego, California., Nemeth A; Oncology Research Division, Pfizer Inc.; San Diego, California., Miller N; Oncology Research Division, Pfizer Inc.; San Diego, California., Hendrickson E; Oncology Research Division, Pfizer Inc.; San Diego, California., Lam H; Oncology Research Division, Pfizer Inc.; San Diego, California., Sherrill J; Oncology Research Division, Pfizer Inc.; San Diego, California., Chung CY; Oncology Research Division, Pfizer Inc.; San Diego, California., McMillan EA; Oncology Research Division, Pfizer Inc.; San Diego, California., Bryant SK; Oncology Research Division, Pfizer Inc.; San Diego, California., Palde P; Oncology Research Division, Pfizer Inc.; San Diego, California., Braganza J; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Brooun A; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Deng YL; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Goshtasbi V; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Kephart SE; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Kumpf RA; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Liu W; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Patman RL; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Rui E; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Scales S; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Tran-Dube M; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Wang F; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Wythes M; Oncology Medicinal Chemistry, Pfizer Inc.; San Diego, California., Paul TA; Oncology Research Division, Pfizer Inc.; San Diego, California. Thomas.A.Paul@pfizer.com.
Publikováno v:
Molecular cancer therapeutics [Mol Cancer Ther] 2022 Jan; Vol. 21 (1), pp. 3-15. Date of Electronic Publication: 2021 Nov 04.
Autor:
Freeman-Cook K; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Hoffman RL; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Miller N; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Almaden J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Chionis J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Zhang Q; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Eisele K; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Liu C; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Zhang C; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Huser N; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Nguyen L; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Costa-Jones C; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Niessen S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Carelli J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Lapek J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Weinrich SL; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Wei P; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., McMillan E; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Wilson E; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Wang TS; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., McTigue M; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Ferre RA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., He YA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Ninkovic S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Behenna D; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Tran KT; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Sutton S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Nagata A; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Ornelas MA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Kephart SE; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Zehnder LR; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Murray B; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Xu M; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Solowiej JE; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Visswanathan R; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Boras B; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Looper D; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Lee N; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Bienkowska JR; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Zhu Z; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Kan Z; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Ding Y; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Mu XJ; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Oderup C; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., Salek-Ardakani S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., White MA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA., VanArsdale T; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA. Electronic address: todd.vanarsdale@pfizer.com., Dann SG; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, CA 92121, USA. Electronic address: stephen@genesistherapeutics.ai.
Publikováno v:
Cancer cell [Cancer Cell] 2021 Oct 11; Vol. 39 (10), pp. 1404-1421.e11. Date of Electronic Publication: 2021 Sep 13.
Autor:
Freeman-Cook KD; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Hoffman RL; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Behenna DC; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Boras B; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Carelli J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Diehl W; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Ferre RA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., He YA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Hui A; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Huang B; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Huser N; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Jones R; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Kephart SE; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Lapek J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., McTigue M; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Miller N; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Murray BW; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Nagata A; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Nguyen L; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Niessen S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Ninkovic S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., O'Doherty I; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Ornelas MA; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Solowiej J; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Sutton SC; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Tran K; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Tseng E; Pfizer Global Research and Development, Eastern Point Road, Groton, Connecticut 06340, United States., Visswanathan R; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Xu M; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Zehnder L; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Zhang Q; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Zhang C; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States., Dann S; Pfizer Global Research and Development La Jolla, 10770 Science Center Drive, San Diego, California 92121, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2021 Jul 08; Vol. 64 (13), pp. 9056-9077. Date of Electronic Publication: 2021 Jun 10.
Autor:
Cheng H; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Orr STM; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Bailey S; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Brooun A; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Chen P; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Deal JG; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Deng YL; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Edwards MP; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Gallego GM; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Grodsky N; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Huang B; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Jalaie M; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Kaiser S; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Kania RS; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Kephart SE; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Lafontaine J; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Ornelas MA; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Pairish M; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Planken S; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Shen H; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Sutton S; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Zehnder L; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Almaden CD; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Bagrodia S; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Falk MD; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Gukasyan HJ; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Ho C; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Kang X; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Kosa RE; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Liu L; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Spilker ME; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Timofeevski S; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Visswanathan R; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Wang Z; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States., Meng F; Wuxi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Ren S; Wuxi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Shao L; Wuxi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Xu F; Wuxi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Kath JC; La Jolla Laboratories, Pfizer Worldwide Research and Development, 10770 Science Center Drive, San Diego, California 92121, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2021 Jan 14; Vol. 64 (1), pp. 644-661. Date of Electronic Publication: 2020 Dec 24.
Autor:
Kung PP, Bingham P, Brooun A, Collins M, Deng YL, Dinh D, Fan C, Gajiwala KS, Grantner R, Gukasyan HJ, Hu W, Huang B, Kania R, Kephart SE, Krivacic C, Kumpf RA, Khamphavong P, Kraus M, Liu W, Maegley KA, Nguyen L, Ren S; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Richter D, Rollins RA; Pfizer Global Research and Development , 401 N. Middletown Road, Pearl River, New York 10965, United States., Sach N, Sharma S, Sherrill J, Spangler J, Stewart AE, Sutton S, Uryu S, Verhelle D, Wang H, Wang S; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Wythes M, Xin S; WuXi AppTec , 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China., Yamazaki S, Zhu H, Zhu J, Zehnder L, Edwards M
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2018 Feb 08; Vol. 61 (3), pp. 650-665. Date of Electronic Publication: 2017 Dec 27.
Autor:
Murray BW; Pfizer Oncology, Pfizer, San Diego, CA 92121, USA. brion.murray@pfizer.com, Guo C, Piraino J, Westwick JK, Zhang C, Lamerdin J, Dagostino E, Knighton D, Loi CM, Zager M, Kraynov E, Popoff I, Christensen JG, Martinez R, Kephart SE, Marakovits J, Karlicek S, Bergqvist S, Smeal T
Publikováno v:
Proceedings of the National Academy of Sciences of the United States of America [Proc Natl Acad Sci U S A] 2010 May 18; Vol. 107 (20), pp. 9446-51. Date of Electronic Publication: 2010 May 03.