Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Kelly M. DiMattio"'
Autor:
Chongguang Chen, Jeffrey J. Liu, Taylor A. Gentile, John W. Muschamp, Peng Huang, Matthias Mann, Lee-Yuan Liu-Chen, Kelly M. DiMattio, Yi-Ting Chiu, Alan Cowan
Kappa opioid receptor (KOR) agonists produce analgesic and anti-pruritic effects, but their clinical application was limited by dysphoria and hallucinations. Nalfurafine, a clinically used KOR agonist, does not cause dysphoria or hallucinations at th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0e7bc3e2dddc0581bf0355721702049f
https://europepmc.org/articles/PMC6462019/
https://europepmc.org/articles/PMC6462019/
Publikováno v:
European Journal of Pharmacology. 748:93-100
β-funaltrexamine (β-FNA) is an irreversible μ opioid (MOP) receptor antagonist and a reversible agonist of κ opioid (KOP) receptor. β-FNA binds covalently to the MOP receptor at Lys233 5.39 , which is conserved among opioid receptors. Molecular
Publikováno v:
Neuroscience Letters. 563:155-159
It has been shown previously that norbinaltorphimine (norBNI) and 5′-guanidinonaltrindole (5′-GNTI), long-acting kappa opioid receptor (KOPR) antagonists, cause frenzied scratching in mice [1] , [2] . In the current study, we examined if zyklophi
Publikováno v:
European journal of pharmacology. 761
Several investigators recently identified biased κ opioid receptor (KOP receptor) agonists. However, no comprehensive study of the functional selectivity of available KOP receptor agonists at the human and mouse KOP receptors (hKOP receptor and mKOP
Autor:
Jian-Guo Li, Lee-Yuan Liu-Chen, Chongguang Chen, Ellen M. Unterwald, Yujun Wang, Kelly M. DiMattio, Wei Xu
Chronic administration of cocaine attenuates delta opioid receptor (DOPR) signaling in the striatum and the desensitization is mediated by the indirect actions of cocaine on dopamine D1 receptors (D1R). In addition, DOPR and D1R co-exist in some rat
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6916a2ef25e2021f05b38f0805f48ca1
https://europepmc.org/articles/PMC3805374/
https://europepmc.org/articles/PMC3805374/