Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Keiichiro Tomita"'
Autor:
Yutaka Kawashima, Takehiro Yamagishi, Hamed I. Ali, Tomohisa Nagamatsu, Eiichi Akaho, Keiichiro Tomita, Hisao Ikeya, Munetaka Kunishima
Publikováno v:
European Journal of Medicinal Chemistry. 43:1376-1389
Various analogs of flavins, 5-deazaflavins, and flavin-5-oxides were docked into the binding site of protein tyrosine kinase pp60 c-src , and some of them were assayed for their potential antitumor and PKC (protein kinase C) inhibitory activities in
Autor:
Shinji Miura, Eiichi Akaho, Hiroyuki Hayakawa, Hamed I. Ali, Hiroto Kambara, Hisao Ikeya, Fumio Yoneda, Yutaka Kawashima, Tomohisa Nagamatsu, Keiichiro Tomita, Takehiro Yamagishi, Noriyuki Ashida
Publikováno v:
Bioorganic & Medicinal Chemistry. 15:242-256
Novel 2-deoxo-2-phenyl-5-deazaflavins and 2-deoxo-2-phenylflavin-5-oxides were prepared as a new class of antitumor agents and showed significant antitumor activities against NCI-H 460, HCT 116, A 431, CCRF-HSB-2, andKB cell lines. In vivo investigat
Publikováno v:
Japanese journal of medical sciencebiology. 5(5)