Zobrazeno 1 - 10
of 24
pro vyhledávání: '"Kazutaka TACHIBANA"'
Publikováno v:
Journal of The Surface Finishing Society of Japan. 73:128-129
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::11c8e21bbda17de2c1029a699d52c685
https://doi.org/10.4139/sfj.73.128
https://doi.org/10.4139/sfj.73.128
Autor:
Hiromitsu Kawata, Ayako Nishimoto, Nobuyuki Ishikura, Takao Houjo, Robert L. Vessella, Hitoshi Yoshino, Takashi Emura, Toshito Nakagawa, Kazutaka Tachibana, Haruhiko Sato, Miho Watanabe, Ryo Nakamura, Takuya Shiraishi, Masateru Ohta, Toshiaki Tsunenari, Yuko Aoki, Akie Honma, Eva Corey
Publikováno v:
International Journal of Oncology. 46:1560-1572
Resistance of prostate cancer to castration is currently an unavoidable problem. The major mechanisms underlying such resistance are androgen receptor (AR) overexpression, androgen-independent activation of AR, and AR mutation. To address this proble
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e627101cf3300cee571ab61aa5f6c0ee
https://doi.org/10.3892/ijo.2015.2860
https://doi.org/10.3892/ijo.2015.2860
Publikováno v:
Materials Science and Engineering: A. 528:8100-8105
This study was conducted to clarify the effects of grain boundaries and precipitates on room-temperature hydrogen transport in two types of austenitic stainless steels with ultrafine-grained structures produced by high-pressure torsion (HPT) and subs
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::17b1d850f2fbd2d8a6f1a537436a3203
https://doi.org/10.1016/j.msea.2011.07.031
https://doi.org/10.1016/j.msea.2011.07.031
Autor:
Hitoshi Yoshino, Muraoka Terushige, Kazutaka Tachibana, Akemi Mizutani, Takashi Emura, Takuya Shiraishi, Akie Honma
Publikováno v:
Synlett. 2011:1117-1120
Short-step and scalable transformations from 2,6-dibromopyridine to 6-bromopyridine-2-sulfonamide by means of halogen―metal exchange and subsequent reaction with sulfuryl chloride followed by amidation are established. Application of the method for
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8f57d2427a2ebbaa8de45489e989321e
https://doi.org/10.1055/s-0030-1259953
https://doi.org/10.1055/s-0030-1259953
Autor:
Takuya Shiraishi, Ayako Nishimoto, Hitoshi Yoshino, Hiromitsu Kawata, Shinichi Arai, Haruhiko Sato, Kazutaka Tachibana, Toshito Nakagawa, Nobuyuki Ishikura, Ryo Nakamura
Publikováno v:
The Prostate. 71:1344-1356
BACKGROUND Castration-resistant prostate cancer (CRPC) is still dependent on androgen receptor (AR) signaling. We previously reported that a novel nonsteroidal AR pure antagonist, CH4933468, which is a thiohydantoin derivative with a sulfonamide side
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::96e9b7a016491ae90c43166f8992ac64
https://doi.org/10.1002/pros.21351
https://doi.org/10.1002/pros.21351
Autor:
Takuya Shiraishi, Ayako Nishimoto, Toshito Nakagawa, Akie Honma, Masateru Ohta, Hitoshi Yoshino, Kazutaka Tachibana, Nobuyuki Ishikura, Toshiaki Tsunenari, Kentaro Furumoto, Ryo Nakamura, Kazuya Kimura, Hiromitsu Kawata, Haruhiko Sato, Miho Watanabe, Noriyuki Takata, Takashi Emura
Publikováno v:
Bioorganic & Medicinal Chemistry. 18:8150-8157
A series of 5,5-dimethylthiohydantoin derivatives were synthesized and evaluated for androgen receptor pure antagonistic activities for the treatment of castration-resistant prostate cancer. Since CH4933468, which we reported previously, had a proble
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8b8d5bf575f9424ec05177698a77a811
https://doi.org/10.1016/j.bmc.2010.10.023
https://doi.org/10.1016/j.bmc.2010.10.023
Publikováno v:
Metallurgical and Materials Transactions A. 41:3110-3120
The effect of high-pressure torsion (HPT) and annealing on hydrogen embrittlement (HE) of a type 304 stainless steel was studied by metallographic characterization and tensile test after hydrogen gas charging. A volume fraction of ~78 pct of the aust
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a10fd3c791d77c59e783de73d4383880
https://doi.org/10.1007/s11661-010-0394-0
https://doi.org/10.1007/s11661-010-0394-0
Autor:
Hiromitsu Kawata, Hitoshi Yoshino, Haruhiko Sato, Nobuyuki Ishikura, Masateru Ohta, Etsuro Onuma, Takuya Shiraishi, Kyung-Yun Jung, Mitsuaki Nakamura, Masahiro Nagamuta, Kazutaka Tachibana, Toshito Nakagawa, Shinichi Arai, Koo-Hyeon Ahn
Publikováno v:
Bioorganic & Medicinal Chemistry. 18:3159-3168
A series of 5,5-dimethylthiohydantoin derivatives were synthesized and evaluated for androgen receptor pure antagonistic activities for the treatment of hormone refractory prostate cancer. CH4933468 (32d) with a sulfonamide side chain not only exhibi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5ba02e5f233be169acfa3c16fe8e8218
https://doi.org/10.1016/j.bmc.2010.03.036
https://doi.org/10.1016/j.bmc.2010.03.036
Autor:
Muraoka Terushige, Akemi Mizutani, Hitoshi Yoshino, Takashi Emura, Kazutaka Tachibana, Akie Honma, Takuya Shiraishi
Publikováno v:
ChemInform. 42
A scalable one-pot transformation via halogen—metal exchange allows the preparation of various title compounds and analogues as important intermediates in drug synthesis.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::31055d5136b669874da3afc331bac712
https://doi.org/10.1002/chin.201138138
https://doi.org/10.1002/chin.201138138
Publikováno v:
Chemistry Letters. 22:937-940
γ-Trialkylstannyl ketones underwent cyclobutanation, C-C bond cleavage, or 1,5-hydride shift, depending upon the substitution pattern of the substrates.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2065358c05c89b32accbb136db82e1d9
https://doi.org/10.1246/cl.1993.937
https://doi.org/10.1246/cl.1993.937