Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Katarina Vorcakova"'
Autor:
Andrzej Bak, Hana Pizova, Violetta Kozik, Katarina Vorcakova, Jiri Kos, Jakub Treml, Klara Odehnalova, Michal Oravec, Ales Imramovsky, Pavel Bobal, Adam Smolinski, Zdeněk Trávníček, Josef Jampilek
Publikováno v:
International Journal of Molecular Sciences, Vol 20, Iss 21, p 5385 (2019)
A set of 25 novel, silicon-based carbamate derivatives as potential acetyl- and butyrylcholinesterase (AChE/BChE) inhibitors was synthesized and characterized by their in vitro inhibition profiles and the selectivity indexes (SIs). The prepared compo
Externí odkaz:
https://doaj.org/article/30c6292c35bb4e59b0e38d4438424014
2-Hydroxy-N-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase
Autor:
Martin Krátký, Šárka Štěpánková, Neto-Honorius Houngbedji, Rudolf Vosátka, Katarína Vorčáková, Jarmila Vinšová
Publikováno v:
Biomolecules, Vol 9, Iss 11, p 698 (2019)
The development of novel inhibitors of acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE) represents a viable approach to alleviate Alzheimer’s disease. Thirty-six halogenated 2-hydroxy-N-phenylbenzamides (salicylanilides) with various s
Externí odkaz:
https://doaj.org/article/827e22d74bb147fc85350ec30870a88a
Autor:
Jarmila Vinšová, Martin Krátký, Markéta Komlóová, Echchukattula Dadapeer, Šárka Štěpánková, Katarína Vorčáková, Jiřina Stolaříková
Publikováno v:
Molecules, Vol 19, Iss 6, Pp 7152-7168 (2014)
A new series of 27 diethyl 2-(phenylcarbamoyl)phenyl phosphorothioates (thiophosphates) was synthesized, characterized by NMR, IR and CHN analyses and evaluated against Mycobacterium tuberculosis H37Rv, Mycobacterium avium and two strains of Mycobact
Externí odkaz:
https://doaj.org/article/61e6a30b8749480ba20de41b367501d3
Autor:
Eliška Kohelová, Rozálie Peřinová, Negar Maafi, Jan Korábečný, Daniela Hulcová, Jana Maříková, Tomáš Kučera, Loreto Martínez González, Martina Hrabinova, Katarina Vorčáková, Lucie Nováková, Angela De Simone, Radim Havelek, Lucie Cahlíková
Publikováno v:
Molecules, Vol 24, Iss 7, p 1307 (2019)
Twelve derivatives 1a–1m of the β-crinane-type alkaloid haemanthamine were developed. All the semisynthetic derivatives were studied for their inhibitory potential against both acetylcholinesterase and butyrylcholinesterase. In addition, glycogen
Externí odkaz:
https://doaj.org/article/e5c8419b582741039c32514f94ab04aa
Publikováno v:
Molecules, Vol 21, Iss 2, p 191 (2016)
Based on the presence of carbamoyl moiety, twenty salicylanilide N,N-disubstituted (thio)carbamates were investigated using Ellman’s method for their ability to inhibit acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). O-Aromatic (thio)
Externí odkaz:
https://doaj.org/article/1c358195046647c3a0b097c55cdc60a2