Zobrazeno 1 - 10
of 11
pro vyhledávání: '"Kang-Po Li"'
Autor:
Kang-Po Li, Ming-Kuan Hu, Cheng-Yi Cheng, Li-Fan Hsu, Ta-Kai Chou, Chyng-Yann Shiue, Daniel H Shen
Publikováno v:
Journal of Medical Sciences, Vol 37, Iss 1, Pp 7-11 (2017)
Aims: 11C-L-methionine, an amino acid tracer used to delineate certain tumor tissues, has proven to be a prevailing nonfluorodeoxyglucose positron emission tomography (PET) radiopharmaceutical. We intended to prepare 11C-L-methionine by following mod
Externí odkaz:
https://doaj.org/article/36f51549f8794eeca8acb1049956a544
Autor:
Wei Chen, Xuedan Wu, Joshua B. McManus, Gerald T. Bida, Kang-Po Li, Zhanhong Wu, David A. Nicewicz, Zibo Li
Publikováno v:
Organic Letters. 24:9316-9321
Innovative labeling methods to incorporate the short-lived positron emitter carbon-11(
Autor:
Mei Luo, Jing-Cheng Zhang, Hao Yin, Cheng-Ming Wang, Lan Xie, Kang-Po Li, Masuo Goto, Susan L. Morris-Natschke, Kuo-Hsiung Lee, Jia-Hai Zhang, Yan-Min Zhang, Xue-Ru Zhang
Publikováno v:
Journal of inorganic biochemistry. 239
Six new Pd(II), Pt(II) and Ag(I) complexes, (1);{Pd (L
Autor:
Susan L. Morris-Natschke, Pei Ling Hsu, Dongqing Zhu, Kang-Po Li, Lan Xie, Xiaoyang He, Li Jiang, Kuo Hsiung Lee, Masuo Goto, Mutian Cui
Publikováno v:
ACS Medicinal Chemistry Letters. 11:83-89
Scaffold hopping-driven lead optimizations were performed based on our prior lead 7-methoxy-4-(2-methylquinazolin-4-yl)-3,4-dihydroquinoxalin-2(1H)-one (2a) by C-ring expansion and isometric replacement of the A/B-ring, successively, aimed at finding
Autor:
Kang-Po Li, Nicholas E. S. Tay, Zhanhong Wu, Hui Wang, Zibo Li, Wei Chen, David A. Nicewicz, Vincent A Pistritto, Tao Zhang
Publikováno v:
Nat Chem
Positron emission tomography (PET) is a powerful imaging technology that could visualize and measure metabolic processes in vivo and/or obtain unique information about drug candidates at early stages. Identification of new and improved molecular prob
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2dddbe56ea479419d563ce0f67f489bd
Autor:
Kuo Hsiung Lee, Kan-Yen Hsieh, Masuo Goto, Kang-Po Li, Stephen J. Capuzzi, Jizhen Li, Ying-Chao Zhang, Pei Ling Hsu, Susan L. Morris-Natschke, Ling-Chu Chang
Publikováno v:
Bioorganic & Medicinal Chemistry. 27:2871-2882
Betulinic acid (BA), a pentacyclic triterpenoid, exhibits broad spectrum antiproliferative activity, but generally with only modest potency. To improve BA’s pharmacological properties, fluorine was introduced as a single atom at C-2, creating two d
Autor:
Nami Kusanagi, Koji Wada, Takahiro Shimizu, Megumi Mizukami, Yuji Suzuki, Kang-Po Li, Hiroshi Yamashita, Masuo Goto, Kuo Hsiung Lee
Publikováno v:
J Nat Med
Diterpenoid alkaloids with remarkable chemical properties and biological activities are frequently found in plants of the genera Aconitum, Delphinium, and Garrya. However, little information has been reported on the antiproliferative effects of the d
Autor:
Ming-Kuan Hu, Cheng-Yi Cheng, Li-Fan Hsu, Chyng-Yann Shiue, Kang-Po Li, Daniel H. Shen, Ta-Kai Chou
Publikováno v:
Journal of Medical Sciences, Vol 37, Iss 1, Pp 7-11 (2017)
Aims: 11C-L-methionine, an amino acid tracer used to delineate certain tumor tissues, has proven to be a prevailing nonfluorodeoxyglucose positron emission tomography (PET) radiopharmaceutical. We intended to prepare 11C-L-methionine by following mod
Autor:
Li, Jiang, Masuo, Goto, Dong-Qing, Zhu, Pei-Ling, Hsu, Kang-Po, Li, Mutian, Cui, Xiaoyang, He, Susan Lynne, Morris-Natschke, Kuo-Hsiung, Lee, Lan, Xie
Publikováno v:
ACS Med Chem Lett
[Image: see text] Scaffold hopping-driven lead optimizations were performed based on our prior lead 7-methoxy-4-(2-methylquinazolin-4-yl)-3,4-dihydroquinoxalin-2(1H)-one (2a) by C-ring expansion and isometric replacement of the A/B-ring, successively
Autor:
Clifton K.-F. Shen, Cheng Yi Cheng, Wei-Yu Lin, Libo Zhao, Shuang Hou, Daniel H. Shen, Kang-Po Li, Ming-Kuan Hu
Publikováno v:
Applied Radiation and Isotopes. 94:113-117
N-Succinimidyl-4-[(18)F]fluorobenzoate ([(18)F]SFB) is a potential prosthetic agent for novel tracer development in positron emission tomography (PET). Previously, we reported a microwave-assisted one-pot synthesis of [(18)F]SFB with high efficacy. H