Zobrazeno 1 - 10 of 22 pro vyhledávání: '"Kaiss Aouadi"'
1
Akademický článek
Synthesis, optical properties, DNA, β-cyclodextrin interactions, and antioxidant evaluation of novel isoxazolidine derivative (ISoXD2): A multispectral and computational analysis
Autor: Ibrahim A. Alhagri, Raghad Alsowayan, Siwar Ghannay, Sadeq M. Al-Hazmy, Iqrar Ahmad, Harun Patel, Adel Kadri, Kaiss Aouadi
Publikováno v: Heliyon, Vol 10, Iss 14, Pp e34561- (2024)
ISoXD2 are well explored among versatile and outstanding class of pharmacophores for the preparation and discovery of drugs. Herein, the electronic absorption and emission spectra of ISoXD2 were investigated in three different solvents. The observed
Externí odkaz: https://doaj.org/article/a36b8883e1054e94abc53d2be7c13ff6
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2
Akademický článek
Synthesis, optical properties, DNA, β-cyclodextrin interaction, hydrogen isotope sensor and computational study of new enantiopure isoxazolidine derivative (ISoXD)
Autor: Afnan Alotayeq, Siwar Ghannay, Ibrahim A. Alhagri, Iqrar Ahmed, Bechir Hammami, Abuzar E. A. E. Albadri, Harun Patel, Sabri Messaoudi, Adel Kadri, Sadeq M. Al-Hazmy, Kaiss Aouadi
Publikováno v: Heliyon, Vol 10, Iss 4, Pp e26341- (2024)
A novel isoxazolidine derivative (ISoXD) dye was successfully synthesized and comprehensively characterized. In this study, we conducted a thorough examination of its various properties, including optical characteristics, interactions with DNA and β
Externí odkaz: https://doaj.org/article/85114b3456b34620b87f569e76278d79
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3
Akademický článek
Identification of dual-target isoxazolidine-isatin hybrids with antidiabetic potential: Design, synthesis, in vitro and multiscale molecular modeling approaches
Autor: Siwar Ghannay, Budur Saleh Aldhafeeri, Iqrar Ahmad, Abuzar E.A.E. Albadri, Harun Patel, Adel Kadri, Kaiss Aouadi
Publikováno v: Heliyon, Vol 10, Iss 4, Pp e25911- (2024)
In the development of novel antidiabetic agents, a novel series of isoxazolidine-isatin hybrids were designed, synthesized, and evaluated as dual α‐amylase and α-glucosidase inhibitors. The precise structures of the synthesized scaffolds were cha
Externí odkaz: https://doaj.org/article/856612864df54719ab96211353e9e49d
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4
Akademický článek
In Silico Design, Synthesis, and Evaluation of Novel Enantiopure Isoxazolidines as Promising Dual Inhibitors of α-Amylase and α-Glucosidase
Autor: Fahad Alhawday, Fahad Alminderej, Siwar Ghannay, Bechir Hammami, Abuzar E. A. E. Albadri, Adel Kadri, Kaiss Aouadi
Publikováno v: Molecules, Vol 29, Iss 2, p 305 (2024)
Isoxazolidine derivatives were designed, synthesized, and characterized using different spectroscopic techniques and elemental analysis and then evaluated for their ability to inhibit both α-amylase and α-glucosidase enzymes to treat diabetes. All
Externí odkaz: https://doaj.org/article/97c16e76fc5e4b79aa0a493f1a1bc1fa
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5
Mechanochemical Promoted Heterocycles: A Solvent-free Route to Triazole Carbohydrates as Glycogen Phosphorylase Inhibitors
Autor: Ahlem Guesmi, Wesam Abdulfattah, Manel Ben Ticha, Faisal K. Algathami, Kaiss Aouadi, Ammar Houas, Lotfi Khezami, Naoufel Ben Hamadi
Publikováno v: Current Organic Synthesis. 19:930-936
Aims: This study aimed to recommend a novel way for the preparation of carbohydrates containing triazole derivatives. Background: Triazoles containing derivatives have numerous biological activities. Ball milling is a fast, modest, green process with
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::7d191728eea6b06c1aa240f9520ba242
https://doi.org/10.2174/1570179419666220420133644
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6
Akademický článek
Crystal structure of 2-isopropyl-5,7′-dimethyl-1′,3′,3a',6′,8a',8b'-hexahydrospiro[cyclohexane-1,6′-furo[3,4-d]imidazo[1,5-b]isoxazol]-8′(7′H)-one
Autor: Heithem Abda, Khaireddine Ezzayani, Kaiss Aouadi, Taha Guerfel, Sebastien Vidal, Moncef Msaddek
Publikováno v: Acta Crystallographica Section E: Crystallographic Communications, Vol 72, Iss 8, Pp 1150-1152 (2016)
In the title compound, C17H28N2O3, the isoxazolidine ring adopts an envelope conformation with the O atom deviating from the mean plane of the other four ring atoms by 0.617 (1) Å. In the crystal, molecules are linked via weak C—H...O hydrogen bon
Externí odkaz: https://doaj.org/article/3dadfc939bd24ca19d87ce70799af4c9
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7
Akademický článek
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8
Akademický článek
In Silico Design, Synthesis, and Evaluation of Novel Enantiopure Isoxazolidines as Promising Dual Inhibitors of α-Amylase and α-Glucosidase.
Autor: Alhawday, Fahad1 (AUTHOR) 431114194@qu.edu.sa, Alminderej, Fahad1 (AUTHOR) f.alminderej@qu.edu.sa, Ghannay, Siwar1 (AUTHOR) s.ghannay@qu.edu.sa, Hammami, Bechir1,2 (AUTHOR) b.hammami@qu.edu.sa, Albadri, Abuzar E. A. E.1 (AUTHOR) aa.albadri@qu.edu.sa, Kadri, Adel3,4 (AUTHOR) lukadel@yahoo.fr, Aouadi, Kaiss1,5 (AUTHOR) lukadel@yahoo.fr
Publikováno v: Molecules. Jan2024, Vol. 29 Issue 2, p305. 19p.
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9
Akademický článek
New Synthetic Routes toward Enantiopure (2S,3R,4R)-4-Hydroxyisoleucine by 1,3-Dipolar Cycloaddition of a Chiral Nitrone to C4 Alkenes.
Autor: Kaiss Aouadi
Publikováno v: Synthesis; Nov2007, Vol. 2007 Issue 21, p3399-3405, 7p
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10
Akademický článek
Crystal structure of 2-isopropyl-5,7'-dimethyl-1',3',3a',6',8a',8b'-hexahydrospiro[cyclohexane-1,6'-furo[3,4-d]imidazo[1,5-b]isoxazol]-8'(7'H)-one.
Autor: Abda, Heithem, Ezzayani, Khaireddine, Aouadi, Kaiss, Guerfel, Taha, Vidal, Sebastien, Msaddek, Moncef
Publikováno v: Acta Crystallographica Section E: Crystallographic Communications; Aug2016, Vol. 72 Issue 8, p1150-1153, 9p
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